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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 13, 2013, Pages 3891-3895

Discovery of a small molecular compound simultaneously targeting RXR and HADC: Design, synthesis, molecular docking and bioassay

(10) Chen, Guo Liang a Wang, Li Hui a Wang, Jian a Chen, Kang a Zhao, Man b Sun, Zhao Zhu a Wang, Shuang a Zheng, Hong Li a Yang, Jing Yu a Wu, Chun Fu a

a SHENYANG PHARMACEUTICAL UNIVERSITY (China)

b NONE

Author keywords

Anti cancer; Dual target; Histone deacetylase; Retinoid X receptors

Indexed keywords

ANTINEOPLASTIC AGENT; HISTONE DEACETYLASE; HISTONE DEACETYLASE INHIBITOR; HYDROXAMIC ACID DERIVATIVE; RECEPTOR BLOCKING AGENT; RETINOID DERIVATIVE; RETINOID X RECEPTOR;

ANTINEOPLASTIC ACTIVITY; ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BIOASSAY; CANCER CELL CULTURE; CONTROLLED STUDY; DRUG DESIGN; DRUG SYNTHESIS; DRUG TARGETING; FEMALE; HUMAN; HUMAN CELL; IC 50; MOLECULAR DOCKING;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DISCOVERY; DRUG SCREENING ASSAYS, ANTITUMOR; HELA CELLS; HISTONE DEACETYLASES; HL-60 CELLS; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; RETINOID X RECEPTORS; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84878875803 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.04.067 Document Type: Article

Times cited : (19)

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