Development of a novel class of pyrrolo-[1,2,5]benzothiadiazepine derivatives as potential anti-schistosomal agents

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 13, 2013, Pages 3785-3787

  Chen, Jinglei ^a   Sun, Weizhen ^a   Yang, Jingjing ^a   Sun, Huan ^a   Wang, Zhixia ^a   Dong, Lanlan ^a   Qiao, Chunhua ^a   Xia, Chao Ming ^a  

^a SOOCHOW UNIVERSITY   (China)

Author keywords

Anti schistosomal; Benzothiadiazepine derivatives

Indexed keywords

ANTISCHISTOSOMAL AGENT; BENZODIAZEPINE DERIVATIVE; PYRROLO[1,2,5]BENZOTHIADIAZEPINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CHLORINATION; CONTROLLED STUDY; DRUG EFFICACY; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; MOUSE; NONHUMAN; SCHISTOSOMA JAPONICUM; SCHISTOSOMIASIS JAPONICA;

ANIMALS; DRUG DESIGN; MOLECULAR STRUCTURE; PYRROLES; SCHISTOSOMA JAPONICUM; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZEPINES;

SCHISTOSOMA JAPONICUM;

EID: 84878860347     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.04.085     Document Type: Article

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