Structure-based fragment screening is demonstrated to be a practical lead discovery method for a representative g-protein-coupled receptor

Journal of Medicinal Chemistry

Volumn 56, Issue 9, 2013, Pages 3444-3445

  Stevens, Benjamin D ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

G PROTEIN COUPLED RECEPTOR;

BIOPHYSICS; DRUG SCREENING; FRAGMENTATION REACTION; NOTE; PROCESS OPTIMIZATION; STRUCTURE ANALYSIS;

DRUG EVALUATION, PRECLINICAL; LIGANDS; RECEPTORS, G-PROTEIN-COUPLED;

EID: 84877694782     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm400561w     Document Type: Note

References (9)

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