Radiosynthesis of [18F]FEt-Tyr-urea-Glu ([18F]FEtTUG) as a new PSMA ligand

Journal of Radioanalytical and Nuclear Chemistry

Volumn 295, Issue 3, 2013, Pages 2289-2294

  Al Momani, E ^a,b   Malik, N ^a,b   Machulla, H J ^a,b   Reske, S N ^a   Solbach, C ^a  

^a UNIVERSITY OF ULM   (Germany)

^b UNIVERSITY OF TÜBINGEN   (Germany)

Author keywords

18F FEtTUG; 18F Fluoroethyl tosylate; Indirect radiofluorination; Prostate cancer; PSMA

Indexed keywords

ACETONITRILE; BASE; FLUOROETHYL TYROSINE UREA GLUTAMATE PEPTIDE; FLUOROETHYLTOSYLATE F 18; FLUOROETHYLTOSYLATE TYROSINE UREA GLUTAMIC ACID F 18; LIGAND; PEPTIDE DERIVATIVE; PROSTATE SPECIFIC MEMBRANE ANTIGEN; RADIOPHARMACEUTICAL AGENT; SODIUM HYDROXIDE; SOLVENT; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG FORMULATION; DRUG PURIFICATION; DRUG PURITY; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HYDROLYSIS; ISOTOPE LABELING; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE; REACTION TIME; TEMPERATURE;

EID: 84876280603     PISSN: 02365731     EISSN: 15882780     Source Type: Journal    
DOI: 10.1007/s10967-012-2293-x     Document Type: Article

References (12)

1. Kularatne SA, Zhou Z, Yang J, Post CB, Low PS (2009) Mol Pharm 6(3):790-800
2. Kularatne SA, Venkatesh C, Santhapuram H-KR, Wang K, Vaitilingam B, Henne WA, Low PS (2010) J Med Chem 53(21):7767-7777
3. Chen Y, Pullambhatla M, Foss CA, Byun Y, Nimmagadda S, Senthamizhchelvan S, Sgouros G, Mease RC, Pomper MG (2011) Clin Cancer Res 17(24):7645-7653
4. Olberg DE, Arukwe JM, Grace D, Hjelstuen OK, Solbakken M, Kindberg GM, Cuthbertson A (2010) J Med Chem 53(4):1732-1740
5. Malik N, Machulla H-J, Solbach C, Winter G, Reske SN, Zlatopolskiy B (2011) Appl Radiat Isot 69(7):1014-1018
6. Glaser M, Årstad E, Luthra SK, Robins EG (2009) J Label Compd Radiopharm 52(8):327-330
7. Scott PJH, Shao X (2010) J Label Compd Radiopharm 53(9):586-591
8. Becaud J, Mu L, Karramkam M, Schubiger PA, Ametamey SM, Graham K, Stellfeld T, Lehmann L, Borkowski S, Berndorff D, Dinkelborg L, Srinivasan A, Smits R, Koksch B (2009) Bioconjug Chem 20(12):2254-2261
9. Wester HJ, Hertz M, Weber W, Heiss P, Senekowitsch-Schmidtke R, Schwaiger M, Stöcklin G (1999) J Nucl Med 40(1):205-212
10. Kozikowski AP, Zhang J, Nan F, Petukhov PA, Grajkowska E, Wroblewski JT, Yamamoto T, Bzdega T, Wroblewska B, Neale JH (2004) J Med Chem 47(7):1729-1738
11. Holschbach M, Schirrmacher R, Solbach C, Hamkens W, Coenen HH (1997) J Lab Comp Radiopharm 40(11):762-763
12. Solbach C (1996) Diploma thesis: Zur selektiven n.c.a. Markierung polyfunktioneller Moleküle mit Kohlenstoff-11 (Towards the selective n.c.a. labelling of polyfunctional molecules with carbon-11). Research Centre Jülich, University of Köln, Germany