Synthetic peptide octarphin (TPLVTLFK) inhibits the activity of the hypothalamus-pituitary-adrenal axis through nonopioid β-endorphin receptor

Regulatory Peptides

Volumn 183, Issue 1, 2013, Pages 23-26

  Nekrasova, Yuliia N ^a   Zolotarev, Yury A ^b   Navolotskaya, Elena V ^a  

^a SHEMYAKIN OVCHINNIKOV INSTITUTE OF BIOORGANIC CHEMISTRY   (Russian Federation)

^b INSTITUTE OF MOLECULAR GENETICS   (Russian Federation)

Author keywords

Endorphin; Adrenal; Hypothalamus; Peptide; Pituitary; Receptor

Indexed keywords

ADENYLATE CYCLASE; BETA ENDORPHIN; BETA ENDORPHIN RECEPTOR; CORTICOSTERONE; NALOXONE; OCTARPHIN; OPIATE RECEPTOR; SYNTHETIC PEPTIDE; TRITIUM; UNCLASSIFIED DRUG; OLIGOPEPTIDE;

ADRENAL CORTEX; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BLOOD FLOW; CONTROLLED STUDY; DRUG MECHANISM; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME REGULATION; HYPOPHYSIS ADRENAL SYSTEM; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN SECRETION; RAT; AMINO ACID SEQUENCE; ANIMAL; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; HYPOTHALAMUS HYPOPHYSIS SYSTEM; INTRAMUSCULAR DRUG ADMINISTRATION; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS; WISTAR RAT;

RATTUS;

AMINO ACID SEQUENCE; ANIMALS; BETA-ENDORPHIN; DOSE-RESPONSE RELATIONSHIP, DRUG; HYPOTHALAMO-HYPOPHYSEAL SYSTEM; INJECTIONS, INTRAMUSCULAR; MALE; OLIGOPEPTIDES; PITUITARY-ADRENAL SYSTEM; RATS; RATS, WISTAR; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84875769441     PISSN: 01670115     EISSN: 18731686     Source Type: Journal    
DOI: 10.1016/j.regpep.2013.03.002     Document Type: Article

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