Nicotinic acid hydrazone: A novel anticonvulsant pharmacophore
Dimmock JR, Pandeya SN, Quail JW, Pugazhenthi U, Allen TM, Kao GY, Balzarini J, DeClereq E. Nicotinic acid hydrazone: A novel anticonvulsant pharmacophore. Eur J Med Chem 1995;30:303-314.
Antiepileptic Drug Device Trials XI Conference. Aventura, FL, April 27-29
Antiepileptic Drug and Device Trials XI Conference. (2011). CPP-115 for refractory complex partial seizures and infantile spasm. Aventura, FL, April 27-29.
Syntheses and evaluation of 3-(3-bromo phenyl)-5-phenyl-1-(thiazolo [4,5-b] quinoxaline-2-yl)-2-pyrazoline derivatives
Budakoti A, Bhat AR, Athar F, Azam A. Syntheses and evaluation of 3-(3-bromo phenyl)-5-phenyl-1-(thiazolo [4,5-b] quinoxaline-2-yl)-2-pyrazoline derivatives. Eur J Med Chem 2008;43:1749-1757.
Poly(ethylene glycol) (PEG-400) as an alternative reaction solvent for the synthesis of some new 1-(4-(4?-chlorophenyl)-2-thiazolyl)-3-aryl-5-(2-butyl- 4-chloro-1H-imidazol-5-l)-2-pyrazolines and their in vitro antimicrobial evaluation
Dawane BS, Konda SG, Mandawad GG, Shaikh BM. Poly(ethylene glycol) (PEG-400) as an alternative reaction solvent for the synthesis of some new 1-(4-(4?-chlorophenyl)-2-thiazolyl)-3-aryl-5-(2-butyl-4-chloro-1H-imidazol-5-l) -2-pyrazolines and their in vitro antimicrobial evaluation. Eur J Med Chem 2010;45:387-392.
Synthesis and biological evaluation of some pyrazolylpyrazolines as anti-inflammatory-antimicrobial agents
Sharma PK, Kumar S, Kumar P, Kaushik P, Kaushik D, Dhingra Y et al. Synthesis and biological evaluation of some pyrazolylpyrazolines as anti-inflammatory-antimicrobial agents. Eur J Med Chem 2010;45:2650-2655.
Studies on the synthesis and antidepressant activity of some 1-thiocarbamoyl-3,5-diphenyl-2-pyrazolines
Bilgin AA, Palaska E, Sunal R. Studies on the synthesis and antidepressant activity of some 1-thiocarbamoyl-3,5-diphenyl-2-pyrazolines. Arzneimittelforschung 1993;43:1041-1044.
Synthesis of some thiazolyl-pyrazoline derivatives and preliminary investigation of their hypotensive activity
Turan-Zitouni G, Chevallet P, Kiliç FS, Erol K. Synthesis of some thiazolyl-pyrazoline derivatives and preliminary investigation of their hypotensive activity. Eur J Med Chem 2000;35:635-641.
Synthesis of N-1 acidic functionality affording analogues with enhanced antiviral activity against HIV
Mui MS, Siew BN, Buss AD, Crasta SC, Kah LG, Sue KL. Synthesis of N-1 acidic functionality affording analogues with enhanced antiviral activity against HIV. Bioorg Med Chem Lett 2002;12: 679-699.
Synthesis of some pyrazole derivatives and preliminary investigation of their affinity binding to P-glycoprotein
Manna F, Chimenti F, Fioravanti R, Bolasco A, Secci D, Chimenti P et al. Synthesis of some pyrazole derivatives and preliminary investigation of their affinity binding to P-glycoprotein. Bioorg Med Chem Lett 2005;15:4632-4635.
Syn thesis, structural activity relationship and anti-tubercular activity of novel pyrazoline derivatives
Ali MA, Shaharyar M, Siddiqui AA. Synthesis, structural activity relationship and anti-tubercular activity of novel pyrazoline derivatives. Eur J Med Chem 2007;42:268-275.
Design, synthesis and antimycobacterial evaluation of novel 3-substituted-N-aryl-6,7-dimethoxy-3a,4-dihydro-3Hindeno[1,2-c] pyrazole-2-carboxamide analogues
Ahsan MJ, Samy JG, Dutt KR, Agrawal UK, Yadav BS, Vyas S et al. Design, synthesis and antimycobacterial evaluation of novel 3-substituted-N-aryl-6,7- dimethoxy-3a,4-dihydro-3Hindeno[1,2-c]pyrazole-2-carboxamide analogues. Bioorg Med Chem Lett 2011;21:4451-4453.
Discovery of novel antitubercular 3a,4-dihydro-3H-indeno[1,2-c] pyrazole-2-carboxamide/carbothioamide analogues
Ahsan MJ, Samy JG, Soni S, Jain N, Kumar L, Sharma LK et al. Discovery of novel antitubercular 3a,4-dihydro-3H-indeno[1,2-c] pyrazole-2-carboxamide/ carbothioamide analogues. Bioorg Med Chem Lett 2011;21:5259-5261.
Synthesis of N1-(3-chloro-4-fluorophenyl)-N4-substituted semicarbazones as novel anticonvulsant agents
Amir M, Ahsan MJ, Ali I. Synthesis of N1-(3-chloro-4-fluorophenyl)-N4- substituted semicarbazones as novel anticonvulsant agents. Ind J Chem 2010;49B:1509-1514.
General principles: Experimental selection, quantification, and evaluation of anticonvulsants
Levy RH,Mattson RH, Melmm B, Penry JK, Dreifuss FE, ed. New York: Raven Press, 85-102
Swinyard EA, Woodhead JH, White HS, Franklin MR. (1989). General principles: Experimental selection, quantification, and evaluation of anticonvulsants. In: Levy RH,Mattson RH, Melmm B, Penry JK, Dreifuss FE, ed. Antiepileptic Drugs. New York: Raven Press, 85-102.
The early identification of anticonvulsant activity: Role of the maximal electroshock and subcutaneous pentylenetetrazol seizure models
White HS, Johnson M, Wolf HH, Kupferberg HJ. The early identification of anticonvulsant activity: Role of the maximal electroshock and subcutaneous pentylenetetrazol seizure models. Ital J Neurol Sci 1995;16:73-77.
In: Levy RH,Mattson RH, Meldrum B, ed. Antiepileptic Drugs. New York: Raven Press
White HS, Woodhead JH, Franklin MR. (1995). General principles: Experimental selection, quantification, and evaluation of antiepileptic drugs. In: Levy RH,Mattson RH, Meldrum B, ed. Antiepileptic Drugs. New York: Raven Press, 99-110.
A note on a simple apparatus for detecting neurological deficit in rats and mice
DUNHAM NW, MIYA TS. A note on a simple apparatus for detecting neurological deficit in rats and mice. J Am Pharm Assoc Am Pharm Assoc (Baltim) 1957;46:208-209.
Pharmacological characterization of the 6 Hz psychomotor seizure model of partial epilepsy
Barton ME, Klein BD, Wolf HH, White HS. Pharmacological characterization of the 6 Hz psychomotor seizure model of partial epilepsy. Epilepsy Res 2001;47:217-227.
Organotypic hippocampal slice cultures for studies of brain damage, neuroprotection and neurorepair
Noraberg J, Poulsen FR, Blaabjerg M, Kristensen BW, Bonde C, Montero M et al. Organotypic hippocampal slice cultures for studies of brain damage, neuroprotection and neurorepair. Curr Drug Targets CNS Neurol Disord 2005;4:435-452.