Copper(II) triflate promoted multicomponent catalytic clubbing of piperazinyl-thiazoloquinolines and thiazolocoumarins as antimicrobials

Archiv der Pharmazie

Volumn 346, Issue 3, 2013, Pages 221-231

  Patel, Rahul V ^a   Patel, Jigar K ^a   Nile, Shivraj H ^b   Park, Se Won ^b  

^a SARDAR VALLABHBHAI NATIONAL INSTITUTE OF TECHNOLOGY   (India)

^b Konkuk University   (South Korea)

Author keywords

Antimicrobial activity; Coumarin; Piperazine; Quinoline; Thiazole

Indexed keywords

2 (3,5 DIMETHYLPIPERIDIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 ACETYLPIPERAZIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 BENZHYDRYLPIPERAZIN 1 YL) 7H CHROMENO [6,5 D]THIAZOL 7 ONE; 2 (4 BENZYLPIPERAZIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 BENZYLPIPERIDIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 ETHYLPIPERAZIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 ISOPROPYLPIPERAZIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 METHYLPIPERAZIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 (4 PHENYLPIPERAZIN 1 YL) 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 (2 FLUOROPHENYL)PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 (2,3 DICHLOROPHENYL)PIPERAZIN 1 YL] 7H CHROMENONE [6,5 D]THIAZOL 7 ONE; 2 [4 (2,3,4 TRIMETHOXYBENZYL)PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 (3 CHLOROPHENYL)PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 (4 FLUOROPHENYL)PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 (4 METHOXYPHENYL)PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 (PYRIDIN 2 YL)PIPERAZIN 1 YL] 7H CHROMENO [6,5 D]THIAZOL 7 ONE; 2 [4 (PYRIMIDIN 2 YL)PIPERAZIN 1 YL] 7H CHROMENO [6,5 D]THIAZOL 7 ONE; 2 [4 [(4 CHLOROPHENYL)(PHENYL)METHYL]PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; 2 [4 [3 (TRIFLUOROMETHYL)PHENYL]PIPERAZIN 1 YL] 7H CHROMENO[6,5 D]THIAZOL 7 ONE; ANTIINFECTIVE AGENT; COUMARIN; CUPRIC ION; CUPRIC ION TRIFLUOROMETHANESULFONIC ACID; PIPERAZINE; PIPERAZINYL THIAZOLOQUINOLINE DERIVATIVE; QUINOLINE; QUINOLINE DERIVATIVE; THIAZOLOCOUMARIN DERIVATIVE; TRIFLUOROMETHANESULFONIC ACID; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ANNULATION REACTION; ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS NIGER; BACILLUS CEREUS; CANDIDA ALBICANS; CARBON NUCLEAR MAGNETIC RESONANCE; CATALYSIS; CONTROLLED STUDY; DRUG SCREENING; ESCHERICHIA COLI; FINITE ELEMENT ANALYSIS; INFRARED SPECTROSCOPY; KLEBSIELLA PNEUMONIAE; MINIMUM INHIBITORY CONCENTRATION; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; ANTI-INFECTIVE AGENTS; ANTIFUNGAL AGENTS; ASPERGILLUS NIGER; CANDIDA ALBICANS; CATALYSIS; COUMARINS; DRUG DESIGN; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; MESYLATES; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; PIPERAZINES; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 84875228758     PISSN: 03656233     EISSN: 15214184     Source Type: Journal    
DOI: 10.1002/ardp.201200383     Document Type: Article

References (13)

1. J. Davies, Nature 1996, 383, 219-220.
2. P. Vicini, A. Geronikaki, K. Anastasia, M. Incerti, F. Zani, Bioorg. Med. Chem. 2006, 14, 3859-3864.
3. B. W. Caprathe, J. C. Jaen, L. D. Wise, T. G. Heffner, T. A. Pugsley, L. T. Meltzer, M. J. Parvez, Med. Chem. 1991, 34, 2736-2746.
4. C. J. Paget, K. Kisner, R. L. Stone, D. C. DeLong, J. Med. Chem. 1969, 12, 1016-1018.
5. G. J. Keating, R. O'Kennedy, in Coumarins: Biology, Applications and Mode of Action (Eds.:, R. O'Kennedy, R. D. Thornes,), Wiley, Chichester, UK 1997, p. 23.
6. Q. Z. Li, X. Y. Nie, J. Liang, Lett. Drug. Des. Discov. 2011, 8, 558-561.
7. O. H. Hishmat, J. A. A. Miky, A. A. Farrag, E. M. Fadl-Allah, Arch. Pharm. Res. 2008, 12, 181-185.
8. R. V. Patel, P. Kumari, D. P. Rajani, K. H. Chikhalia, J. Fluorine Chem. 2011, 132, 617-627.
9. R. V. Patel, P. Kumari, D. P. Rajani, K. H. Chikhalia, Eur. J. Med. Chem. 2011, 46, 4354-4365.
10. R. V. Patel, J. K. Patel, P. Kumari, K. H. Chikhalia, Lett. Org. Chem. 2012, 9, 478-486.
11. R. V. Patel, P. Kumari, D. P. Rajani, K. H. Chikhalia, Med. Chem. Res. 2013, 22, 195-210.
12. K. C. Majumdar, N. De, D. Ghosh, S. Ponra, B. Roya, Synthesis 2012, 1, 87-92.
13. G. W. Clause, Understanding Microbes: A Laboratory Textbook for Microbiology, W.H. Freeman and Company, New York, USA 1989.