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Volumn 8, Issue 3, 2013, Pages 415-425

Synthesis and Biological Evaluation of Purine 2′-Fluoro-2′-deoxyriboside ProTides as Anti-influenza Virus Agents

(6) Meneghesso, Silvia a Vanderlinden, Evelien b Brancale, Andrea a Balzarini, Jan b Naesens, Lieve b Mcguigan, Christopher a

a CARDIFF UNIVERSITY (United Kingdom)

b REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

Author keywords

2 fluoro 2 deoxyguanosine; Antiviral agents; Influenza; Nucleosides; ProTides

Indexed keywords

ANTIVIRUS AGENT; CARBOXYPEPTIDASE C; DEOXYGUANOSINE DERIVATIVE; PHOSPHORAMIDIC ACID DERIVATIVE; RIBAVIRIN;

ANIMAL CELL; ARTICLE; BIOLOGICAL ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME ASSAY; INFLUENZA VIRUS A; MDCK CELL; NONHUMAN; PRIORITY JOURNAL;

ADENOSINE DEAMINASE; ANIMALS; ANTIVIRAL AGENTS; BINDING SITES; CATALYTIC DOMAIN; DNA-DIRECTED RNA POLYMERASES; DOGS; DRUG EVALUATION, PRECLINICAL; FLUORINE; HEK293 CELLS; HUMANS; MADIN DARBY CANINE KIDNEY CELLS; MOLECULAR DOCKING SIMULATION; NUCLEOSIDES; ORTHOMYXOVIRIDAE; PURINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84874328316 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201200562 Document Type: Article

Times cited : (18)

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