Blockade of insect odorant receptor currents by amiloride derivatives

Chemical Senses

Volumn 38, Issue 3, 2013, Pages 221-229

  Pask, Gregory M ^a   Bobkov, Yuriy V ^b   Corey, Elizabeth A ^b   Ache, Barry W ^b   Zwiebel, Laurence J ^a,c  

^a VANDERBILT UNIVERSITY   (United States)

^b UNIVERSITY OF FLORIDA   (United States)

^c VANDERBILT UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Amiloride; Channel blocker; Insect; Odorant receptor

Indexed keywords

3',4' DICHLOROBENZAMIL; 5 (N ETHYL N ISOPROPYL)AMILORIDE; 5 (N ISOBUTYL N METHYL)AMILORIDE; 5 (N,N DIMETHYL)AMILORIDE; 5 (N,N HEXAMETHYLENE)AMILORIDE; AMILORIDE; AMILORIDE DERIVATIVE; ION CHANNEL; N (4 ETHYLPHENYL) 2 [[4 ETHYL 5 (3 PYRIDINYL) 4H 1,2,4 TRIAZOL 3 YL]THIO]ACETAMIDE; ORCO CHANNEL SUBUNIT; PHENAMIL; THIOACETAMIDE DERIVATIVE; UNCLASSIFIED DRUG;

ANOPHELES GAMBIAE; ARTICLE; CHEMICAL STRUCTURE; CONTROLLED STUDY; EMBRYO; HARPEGNATHOS SALTATOR; HELIOTHIS VIRESCENS; HEMIPTERA; HUMAN; HUMAN CELL; HYMENOPTERA; IC 50; INHIBITION KINETICS; ION CURRENT; LEPIDOPTERA; LYGUS HESPERUS; NONHUMAN; OLFACTORY RECEPTOR; PRIORITY JOURNAL; RECEPTOR BINDING; RECEPTOR BLOCKING;

AMILORIDE; ANIMALS; ANOPHELES GAMBIAE; CELL LINE; HEK293 CELLS; HUMANS; INSECT PROTEINS; PATCH-CLAMP TECHNIQUES; RECEPTORS, ODORANT; THIOGLYCOLATES; TRANSFECTION; TRIAZOLES;

EID: 84874037047     PISSN: 0379864X     EISSN: 14643553     Source Type: Journal    
DOI: 10.1093/chemse/bjs100     Document Type: Article

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