Comparison and systematic optimization of synthetic protocols for DOTA-hydrazide generation

Tetrahedron Letters

Volumn 54, Issue 8, 2013, Pages 918-920

  Fuge, Felix ^a   Weiler, Marek ^a   Gätjens, Jessica ^a   Lammers, Twan ^a,b,c   Kiessling, Fabian ^a  

^a RWTH AACHEN UNIVERSITY   (Germany)

^b UNIVERSITY OF TWENTE   (Netherlands)

^c UTRECHT UNIVERSITY   (Netherlands)

Author keywords

Alkylation; Cyclen; DOTA; Hydrazide; Lanthanides

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECAN N,N',N'',N''' TETRAACETIC ACID; CHELATING AGENT; GADOLINIUM; GALLIUM; HYDRAZIDE DERIVATIVE; INDIUM; ORGANOMETALLIC COMPOUND; UNCLASSIFIED DRUG; YTTRIUM;

ARTICLE; COMPARATIVE STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; MOLECULAR IMAGING; PROCESS OPTIMIZATION; RADIOIMMUNOTHERAPY; REACTION TIME; THERMODYNAMICS;

EID: 84872351786     PISSN: 00404039     EISSN: 18733581     Source Type: Journal    
DOI: 10.1016/j.tetlet.2012.11.151     Document Type: Article

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