Benzophenone derivatives of pyrimidines as effective non-nucleoside inhibitors of wild-type and drug-resistant HIV-1 reverse transcriptase

Doklady Biochemistry and Biophysics

Volumn 447, Issue 1, 2012, Pages 280-281

  Prokofjeva, M M ^a   Valuev Elliston, V T ^a   Ivanov, A V ^a   Kochetkov, S N ^a   Novikov, M S ^b   Prassolov, V S ^a  

^a ENGELHARDT INSTITUTE OF MOLECULAR BIOLOGY   (Russian Federation)

^b VOLGOGRAD STATE MEDICAL UNIVERSITY   (Russian Federation)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOPHENONE; BENZOPHENONE DERIVATIVE; ENZYME INHIBITOR; NUCLEOSIDE; PYRIMIDINE DERIVATIVE; REVERSE TRANSCRIPTASE, HUMAN IMMUNODEFICIENCY VIRUS 1; RNA DIRECTED DNA POLYMERASE;

ANTIVIRAL RESISTANCE; ARTICLE; CHEMISTRY; DRUG ANTAGONISM; DRUG EFFECT;

BENZOPHENONES; DRUG RESISTANCE, VIRAL; ENZYME INHIBITORS; HIV REVERSE TRANSCRIPTASE; NUCLEOSIDES; PYRIMIDINES;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 84871953342     PISSN: 16076729     EISSN: None     Source Type: Journal    
DOI: 10.1134/S160767291206004X     Document Type: Article

References (5)

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3. Novikov, M. S., Ivanova, O. N., Ivanov, A. V., Ozerov, A. A., Valuev-Elliston, V. T., Gurskaya, G. V., Kochetkov, S. N., Pannecouque, C., Balzarini, J., and Seley-Radtke, K. L., Bioorg. Med. Chem., 2011, vol. 19, no. 19, pp. 5794-5802.
4. Ren, J., Chamberlain, P. P., Stamp, A., Short, S. A., Weaver, K. L., Romines, K. R., Hazen, R., Freeman, A., Ferris, R. G., Andrews, C. W., Boone, L., Chan, J. H., and Stammers, D. K., J. Med. Chem., 2008, vol. 51, no. 16, pp. 5000-5008.
5. Prokof'eva, M. M., Spirin, P. V., Yanvarev, D. V., Ivanov, A. V., Novikov, M. S., Stepanov, O. A., Gottikh, M. B., Kochetkov, S. N., Fehse, B., Stocking, C., and Prasolov, V. S., Acta Nat., 2011, vol. 3, no. 4, pp. 61-71.