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Volumn 14, Issue 6, 2012, Pages 743-752

Quantitative analysis and parametric imaging of 18F-labeled monomeric and dimeric RGD peptides using compartment model

Author keywords

Integrin; Kinetic modeling; Positron emission tomography; Quantitative analysis; RGD peptide

Indexed keywords

FLUORINE FPPRGD2 F 18; FLUORINE FPRGD F 18; RADIOPHARMACEUTICAL AGENT; TRACER; UNCLASSIFIED DRUG;

EID: 84870470028     PISSN: 15361632     EISSN: 18602002     Source Type: Journal    
DOI: 10.1007/s11307-012-0541-7     Document Type: Article
Times cited : (29)

References (35)
  • 1
    • 52549109852 scopus 로고    scopus 로고
    • Imaging of integrin alphavbeta3 expression
    • Beer AJ, Schwaiger M (2008) Imaging of integrin alphavbeta3 expression. Cancer Metastasis Rev 27:631-644
    • (2008) Cancer Metastasis Rev , vol.27 , pp. 631-644
    • Beer, A.J.1    Schwaiger, M.2
  • 2
    • 65549092007 scopus 로고    scopus 로고
    • Engineered knottin peptides: A new class of agents for imaging integrin expression in living subjects
    • Kimura RH, Cheng Z, Gambhir SS et al (2009) Engineered knottin peptides: a new class of agents for imaging integrin expression in living subjects. Cancer Res 69:2435-2442
    • (2009) Cancer Res , vol.69 , pp. 2435-2442
    • Kimura, R.H.1    Cheng, Z.2    Gambhir, S.S.3
  • 3
    • 0036488589 scopus 로고    scopus 로고
    • Role of integrins in cell invasion and migration
    • Hood JD, Cheresh DA (2002) Role of integrins in cell invasion and migration. Nat Rev Cancer 2:91-100
    • (2002) Nat Rev Cancer , vol.2 , pp. 91-100
    • Hood, J.D.1    Cheresh, D.A.2
  • 4
    • 0035266374 scopus 로고    scopus 로고
    • Noninvasive imaging of αvβ3 integrin expression using 18F-labeled RGD-containing glycopeptide and positron emission tomography
    • Haubner R, Wester HJ, Weber WA et al (2001) Noninvasive imaging of αvβ3 integrin expression using 18F-labeled RGD-containing glycopeptide and positron emission tomography. Cancer Res 61:1781-1785
    • (2001) Cancer Res , vol.61 , pp. 1781-1785
    • Haubner, R.1    Wester, H.J.2    Weber, W.A.3
  • 5
    • 79959271064 scopus 로고    scopus 로고
    • Why integrin as a primary target for imaging and therapy
    • Niu G, Chen X (2011) Why integrin as a primary target for imaging and therapy. Theranostics 1:30-47
    • (2011) Theranostics , vol.1 , pp. 30-47
    • Niu, G.1    Chen, X.2
  • 6
    • 80255141418 scopus 로고    scopus 로고
    • PET imaging of integrin αvβ3 expression
    • Beer AJ, Kessler H, Wester HJ et al (2011) PET imaging of integrin αvβ3 expression. Theranostics 1:48-57
    • (2011) Theranostics , vol.1 , pp. 48-57
    • Beer, A.J.1    Kessler, H.2    Wester, H.J.3
  • 7
    • 33646057302 scopus 로고    scopus 로고
    • Multimodality imaging of tumor integrin αvβ3 expression
    • Chen X (2006) Multimodality imaging of tumor integrin αvβ3 expression. Mini Rev Med Chem 6:227-234
    • (2006) Mini Rev Med Chem , vol.6 , pp. 227-234
    • Chen, X.1
  • 8
    • 80051700245 scopus 로고    scopus 로고
    • Novel 64Cu-and 68Ga-labeled RGD conjugates show improved PET imaging of αvβ3 integrin expression and facile radiosynthesis
    • Dumont RA, Deininger F, Haubner R et al (2011) Novel 64Cu-and 68Ga-labeled RGD conjugates show improved PET imaging of αvβ3 integrin expression and facile radiosynthesis. J Nucl Med 52:1276-1284
    • (2011) J Nucl Med , vol.52 , pp. 1276-1284
    • Dumont, R.A.1    Deininger, F.2    Haubner, R.3
  • 9
    • 79959567221 scopus 로고    scopus 로고
    • Pilot pharmacokinetic and dosimetric studies of 18F-FPPRGD2: A PET radiopharmaceutical agent for imaging αvβ3 integrin levels
    • Mittra ES, Goris ML, Iagaru AH et al (2011) Pilot pharmacokinetic and dosimetric studies of 18F-FPPRGD2: a PET radiopharmaceutical agent for imaging αvβ3 integrin levels. Radiology 260:182-191
    • (2011) Radiology , vol.260 , pp. 182-191
    • Mittra, E.S.1    Goris, M.L.2    Iagaru, A.H.3
  • 10
    • 84861481740 scopus 로고    scopus 로고
    • First experience with clinical-grade [18F]FPP(RGD) 2 an automated multi-step radiosynthesis for clinical PET studies
    • Chin FT, Shen B, Liu S et al (2012) First experience with clinical-grade [18F]FPP(RGD)2: an automated multi-step radiosynthesis for clinical PET studies. Mol Imaging Biol 14:88-95.
    • (2012) Mol Imaging Biol , vol.14 , pp. 88-95
    • Chin, F.T.1    Shen, B.2    Liu, S.3
  • 11
    • 79952784609 scopus 로고    scopus 로고
    • Monitoring tumor response to antiangiogenic sunitinib therapy with 18F-fluciclatide, an 18F-labeled αvβ3-integrin and αvβ5-integrin imaging agent
    • Battle MR, Goggi JL, Allen L et al (2011) Monitoring tumor response to antiangiogenic sunitinib therapy with 18F-fluciclatide, an 18F-labeled αvβ3-integrin and αvβ5-integrin imaging agent. J Nucl Med 52:424-430
    • (2011) J Nucl Med , vol.52 , pp. 424-430
    • Battle, M.R.1    Goggi, J.L.2    Allen, L.3
  • 12
    • 72449156995 scopus 로고    scopus 로고
    • Radiolabeled cyclic RGD peptides as integrin αvβ3-targeted radiotracers: Maximizing binding affinity via bivalency
    • Liu S (2009) Radiolabeled cyclic RGD peptides as integrin αvβ3-targeted radiotracers: maximizing binding affinity via bivalency. Bioconjug Chem 20:2199-2213
    • (2009) Bioconjug Chem , vol.20 , pp. 2199-2213
    • Liu, S.1
  • 13
    • 67651122837 scopus 로고    scopus 로고
    • Ligands for mapping αvβ3-integrin expression in vivo
    • Schottelius M, Laufer B, Kessler H et al (2009) Ligands for mapping αvβ3-integrin expression in vivo. Acc Chem Res 42:969-980
    • (2009) Acc Chem Res , vol.42 , pp. 969-980
    • Schottelius, M.1    Laufer, B.2    Kessler, H.3
  • 14
    • 38149039498 scopus 로고    scopus 로고
    • Preparation of peptide-conjugated quantum dots for tumor vasculature-targeted imaging
    • Cai W, Chen X (2008) Preparation of peptide-conjugated quantum dots for tumor vasculature-targeted imaging. Nat Protoc 3:89-96
    • (2008) Nat Protoc , vol.3 , pp. 89-96
    • Cai, W.1    Chen, X.2
  • 15
    • 44149120982 scopus 로고    scopus 로고
    • Preparation of a promising angiogenesis PET imaging agent: 68Ga-labeled c(RGDyK)-isothiocyanatobenzyl-1,4,7-triazacyclononane-1,47-triacetic acid and feasibility studies in mice
    • Jeong JM, Hong MK, Chang YS et al (2008) Preparation of a promising angiogenesis PET imaging agent: 68Ga-labeled c(RGDyK)-isothiocyanatobenzyl-1,4, 7-triazacyclononane-1,4,7-triacetic acid and feasibility studies in mice. J Nucl Med 49:830-836
    • (2008) J Nucl Med , vol.49 , pp. 830-836
    • Jeong, J.M.1    Hong, M.K.2    Chang, Y.S.3
  • 16
    • 27944457471 scopus 로고    scopus 로고
    • MicroPET imaging of glioma integrin αvβ3 expression using 64Cu-labeled tetrameric RGD peptide
    • Wu Y, Zhang X, Xiong Z et al (2005) microPET imaging of glioma integrin αvβ3 expression using 64Cu-labeled tetrameric RGD peptide. J Nucl Med 46:1707-1718
    • (2005) J Nucl Med , vol.46 , pp. 1707-1718
    • Wu, Y.1    Zhang, X.2    Xiong, Z.3
  • 17
    • 79851504879 scopus 로고    scopus 로고
    • 18F-FPPRGD2 and 18F-FDG PET of response to Abraxane therapy
    • Sun X, Yan Y, Liu S et al (2011) 18F-FPPRGD2 and 18F-FDG PET of response to Abraxane therapy. J Nucl Med 52:140-146
    • (2011) J Nucl Med , vol.52 , pp. 140-146
    • Sun, X.1    Yan, Y.2    Liu, S.3
  • 18
    • 77956264376 scopus 로고    scopus 로고
    • 18F-labeled galacto and PEGylated RGD dimers for PET imaging of αvβ3 integrin expression
    • Liu S, Liu Z, Chen K et al (2010) 18F-labeled galacto and PEGylated RGD dimers for PET imaging of αvβ3 integrin expression. Mol Imaging Biol 12:530-538
    • (2010) Mol Imaging Biol , vol.12 , pp. 530-538
    • Liu, S.1    Liu, Z.2    Chen, K.3
  • 19
    • 33646415036 scopus 로고    scopus 로고
    • Quantitative PET imaging of tumor integrin alphavbeta3 expression with 18F-FRGD2
    • Zhang X, Xiong Z, Wu Y et al (2006) Quantitative PET imaging of tumor integrin alphavbeta3 expression with 18F-FRGD2. J NuclMed 47:113-121
    • (2006) J NuclMed , vol.47 , pp. 113-121
    • Zhang, X.1    Xiong, Z.2    Wu, Y.3
  • 20
    • 70349263634 scopus 로고    scopus 로고
    • Noninvasive imaging of tumor integrin expression using 18F-labeled RGD dimer peptide with PEG4 linkers
    • Liu Z, Liu S, Wang F et al (2009) Noninvasive imaging of tumor integrin expression using 18F-labeled RGD dimer peptide with PEG4 linkers. Eur J Nucl Med Mol Imaging 36:1296-1307
    • (2009) Eur J Nucl Med Mol Imaging , vol.36 , pp. 1296-1307
    • Liu, Z.1    Liu, S.2    Wang, F.3
  • 21
    • 74949085524 scopus 로고    scopus 로고
    • Quantitative small animal PET
    • Shoghi KI (2009) Quantitative small animal PET. Q J Nucl Med Mol Imaging 53:365-373
    • (2009) Q J Nucl Med Mol Imaging , vol.53 , pp. 365-373
    • Shoghi, K.I.1
  • 22
    • 79551620355 scopus 로고    scopus 로고
    • Parametric mapping of [18F] fluoromisonidazole positron emission tomography using basis functions
    • Hong YT, Beech JS, Smith R et al (2011) Parametric mapping of [18F] fluoromisonidazole positron emission tomography using basis functions. J Cereb Blood Flow Metab 31:648-657
    • (2011) J Cereb Blood Flow Metab , vol.31 , pp. 648-657
    • Hong, Y.T.1    Beech, J.S.2    Smith, R.3
  • 23
    • 25444503494 scopus 로고    scopus 로고
    • Biodistribution and pharmacokinetics of the alphavbeta3-selective tracer 18F-galacto-RGD in cancer patients
    • Beer AJ, Haubner R, Goebel M et al (2005) Biodistribution and pharmacokinetics of the alphavbeta3-selective tracer 18F-galacto-RGD in cancer patients. J Nucl Med 46:1333-1341
    • (2005) J Nucl Med , vol.46 , pp. 1333-1341
    • Beer, A.J.1    Haubner, R.2    Goebel, M.3
  • 24
    • 59249086628 scopus 로고    scopus 로고
    • Derivation of a compartmental model for quantifying 64Cu-DOTA-RGD kinetics in tumor-bearing mice
    • Ferl GZ, Dumont RA, Hildebrandt IJ et al (2009) Derivation of a compartmental model for quantifying 64Cu-DOTA-RGD kinetics in tumor-bearing mice. J Nucl Med 50:250-258
    • (2009) J Nucl Med , vol.50 , pp. 250-258
    • Ferl, G.Z.1    Dumont, R.A.2    Hildebrandt, I.J.3
  • 25
    • 80455124484 scopus 로고    scopus 로고
    • 18F-labeled GRPR agonists and antagonists: A comparative study in prostate cancer imaging
    • Yang M, Gao H, Zhou Y et al (2011) 18F-labeled GRPR agonists and antagonists: a comparative study in prostate cancer imaging. Theranostics 1:220-229
    • (2011) Theranostics , vol.1 , pp. 220-229
    • Yang, M.1    Gao, H.2    Zhou, Y.3
  • 26
    • 80455155057 scopus 로고    scopus 로고
    • Imaging tumor endothelial marker 8 using an 18F-labeled peptide
    • Quan Q, Yang M, Gao H et al (2011) Imaging tumor endothelial marker 8 using an 18F-labeled peptide. Eur J Nucl Med Mol Imaging 38:1806-1815
    • (2011) Eur J Nucl Med Mol Imaging , vol.38 , pp. 1806-1815
    • Quan, Q.1    Yang, M.2    Gao, H.3
  • 27
    • 0018582265 scopus 로고
    • Tomographic measurement of local cerebral glucose metabolic rate in humans with 18F-2-fluoro-2-deoxy-D-glucose: Validation of method
    • Phelps ME, Huang SC, Hoffman EJ et al (1979) Tomographic measurement of local cerebral glucose metabolic rate in humans with 18F-2-fluoro-2-deoxy-D- glucose: validation of method. Ann Neurol 6:371-388
    • (1979) Ann Neurol , vol.6 , pp. 371-388
    • Phelps, M.E.1    Huang, S.C.2    Hoffman, E.J.3
  • 28
    • 0016355478 scopus 로고
    • A new look at the statistical model identification
    • Akaike H (1974) A new look at the statistical model identification. IEEE Trans Automat Contr AC:716-723
    • (1974) IEEE Trans Automat Contr AC , pp. 716-723
    • Akaike, H.1
  • 29
    • 33845647144 scopus 로고    scopus 로고
    • PET kinetic analysis -compartmental model
    • Watabe H, Ikoma Y, Kimura Y et al (2006) PET kinetic analysis -compartmental model. Ann Nucl Med 20:583-588
    • (2006) Ann Nucl Med , vol.20 , pp. 583-588
    • Watabe, H.1    Ikoma, Y.2    Kimura, Y.3
  • 30
    • 34547846251 scopus 로고    scopus 로고
    • Consensus nomenclature for in vivo imaging of reversibly binding radioligands
    • Innis RB, Cunningham VJ, Delforge J et al (2007) Consensus nomenclature for in vivo imaging of reversibly binding radioligands. J Cereb Blood Flow Metab 27:1533-1539
    • (2007) J Cereb Blood Flow Metab , vol.27 , pp. 1533-1539
    • Innis, R.B.1    Cunningham, V.J.2    Delforge, J.3
  • 31
    • 43749105336 scopus 로고    scopus 로고
    • 68Ga-labeled multimeric RGD peptides for microPET imaging of integrin αvβ3 expression
    • Li ZB, Chen K, Chen X (2008) 68Ga-labeled multimeric RGD peptides for microPET imaging of integrin αvβ3 expression. Eur J Nucl Med Mol Imaging 35:1100-1108
    • (2008) Eur J Nucl Med Mol Imaging , vol.35 , pp. 1100-1108
    • Li, Z.B.1    Chen, K.2    Chen, X.3
  • 32
    • 84861482301 scopus 로고    scopus 로고
    • Importance of quantification for the analysis of PET data in oncology: Review of current methods and trends for the future
    • doi:10.1007/s11307-011-0514-2
    • Tomasi G, Turkheimer F, Aboagye E (2011) Importance of quantification for the analysis of PET data in oncology: review of current methods and trends for the future. Mol Imaging Biol. doi:10.1007/s11307-011-0514-2
    • (2011) Mol Imaging Biol.
    • Tomasi, G.1    Turkheimer, F.2    Aboagye, E.3
  • 33
    • 34447336118 scopus 로고    scopus 로고
    • 64Cu-labeled tetrameric and octameric RGD peptides for small-animal PET of tumor αvβ3 integrin expression
    • Li ZB, Cai W, Cao Q et al (2007) 64Cu-labeled tetrameric and octameric RGD peptides for small-animal PET of tumor αvβ3 integrin expression. J Nucl Med 48:1162-1171
    • (2007) J Nucl Med , vol.48 , pp. 1162-1171
    • Li, Z.B.1    Cai, W.2    Cao, Q.3
  • 34
    • 4644327177 scopus 로고    scopus 로고
    • Micro-PET imaging of αvβ3-integrin expression with 18F-labeled dimeric RGD peptide
    • Chen X, Tohme M, Park R et al (2004) Micro-PET imaging of αvβ3-integrin expression with 18F-labeled dimeric RGD peptide. Mol Imaging 3:96-104
    • (2004) Mol Imaging , vol.3 , pp. 96-104
    • Chen, X.1    Tohme, M.2    Park, R.3
  • 35
    • 84856235199 scopus 로고    scopus 로고
    • Quantification of receptorligand binding with [18F]fluciclatide in metastatic breast cancer patients
    • Tomasi G, Kenny L, Mauri F et al (2011) Quantification of receptorligand binding with [18F]fluciclatide in metastatic breast cancer patients. Eur J Nucl Med Mol Imaging 38:2186-2197
    • (2011) Eur J Nucl Med Mol Imaging , vol.38 , pp. 2186-2197
    • Tomasi, G.1    Kenny, L.2    Mauri, F.3


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