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Volumn 7, Issue 12, 2012, Pages 2077-2081

Discovery of Depsides and Depsidones from Lichen as Potent Inhibitors of Microsomal Prostaglandin E2 Synthase-1 Using Pharmacophore Models

(9) Bauer, Julia a Waltenberger, Birgit b Noha, Stefan M b Schuster, Daniela b Rollinger, Judith M b Boustie, Joel c Chollet, Marylene c Stuppner, Hermann b Werz, Oliver d

a UNIVERSITY OF TÜBINGEN (Germany)

b UNIVERSITY OF INNSBRUCK (Austria)

c UNIVERSITÉ DE RENNES 1 (France)

d FRIEDRICH SCHILLER UNIVERSITY JENA (Germany)

Author keywords

Depsides; Depsidones; Lichens; Pharmacophore models; Prostaglandin E2 synthase 1

Indexed keywords

3 [3 TERT BUTYLTHIO 1 (4 CHLOROBENZYL) 5 ISOPROPYL 2 INDOLYL] 2,2 DIMETHYLPROPIONIC ACID; ATRANORIN; CELECOXIB; DEPSIDE; DEPSIDONE; EVERNIC ACID; FUMARPROTOCETRARIC ACID; INDOMETACIN; METHYLBETAORCINOL CARBOXYLATE; OLIVETORIC ACID; PERLATOLIC ACID; PHYSODIC ACID; PROSTAGLANDIN E SYNTHASE 1; PROSTAGLANDIN SYNTHASE INHIBITOR; SALAZINIC ACID; SCENSIDIN; UNCLASSIFIED DRUG; VARIOLARIC ACID;

ARTICLE; CHINESE MEDICINE; COMPETITIVE INHIBITION; DRUG STRUCTURE; HYDROPHOBICITY; HYPERICUM PERFORATUM; LICHEN (ORGANISM); MYRTLE; NONHUMAN; PHARMACOPHORE; PRIORITY JOURNAL; SITE DIRECTED MUTAGENESIS; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS; TEA;

ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; CELL LINE; COMPUTER SIMULATION; DEPSIDES; DRUG DISCOVERY; HUMANS; INTRAMOLECULAR OXIDOREDUCTASES; LACTONES; LICHENS; MICROSOMES; MODELS, MOLECULAR;

EID: 84870265989 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201200345 Document Type: Article

Times cited : (55)

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