Measurement and correlation of the solubility of febuxostat in four organic solvents at various temperatures

Journal of Chemical and Engineering Data

Volumn 57, Issue 11, 2012, Pages 3149-3152

  Zhang, Lei ^a   Huang, Zhiping ^a   Wan, Xiaoran ^a   Li, Jing ^a   Liu, Jing ^a  

^a SOUTH CHINA UNIVERSITY OF TECHNOLOGY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

CORRELATION EQUATION; ETHYL ACETATES; GRAVIMETRIC METHODS; SOLUBILITY DATA; SOLVENT SELECTION; VAN'T HOFF EQUATION;

ACETONE; ATMOSPHERIC PRESSURE; ETHANOL; METHANOL; ORGANIC SOLVENTS;

SOLUBILITY;

EID: 84868695221     PISSN: 00219568     EISSN: 15205134     Source Type: Journal    
DOI: 10.1021/je300647k     Document Type: Article

References (11)

1. Becker, M. A.; Schumacher, H. R., Jr.; Wortmann, R. L.; Macdonald, P. A.; Eustace, D.; Palo, W. A.; Streit, J.; Joseph-Ridge, N. Febuxostat compared with allopurinol in patients with hyperuricemia and gout N. Engl. J. Med. 2005, 353, 2450-2461
2. Schumacher, H. R., Jr.; Becker, M. A.; Wortmann, R. L.; Macdonald, P. A.; Hunt, B.; Streit, J.; Lademacher, C.; Joseph-Ridge, N. Effects of febuxostat versus allopurinol and placebo in reducing serum urate in subjects with hyperuricemia and gout: A 28-week, phase III, randomized, double-blind, parallel-group trial Arthritis Rheum. 2008, 59 (11) 1540-1548
3. Kitamura, M. Controlling factors and mechanism of polymorphic crystallization Cryst. Growth Des. 2004, 4 (6) 1153-1159
4. Kitamura, M.; Hironaka, S. Effect of temperature on antisolvent crystallization and transformation behaviors of thiazole-derivative polymorphs Cryst. Growth Des. 2006, 6 (5) 1214-1218
5. Kitamura, M.; Sugimoto, M. Anti-solvent crystallization and transformation of thiazole-derivative polymorphs-I: effect of addition rate and initial concentrations J. Cryst. Growth 2003, 257 (1-2) 177-184
6. Kitamura, M. Strategy for control of crystallization of polymorphs CrystEngComm 2009, 11 (6) 949-964
7. Baluja, S.; Bhalodia, R.; Bhatt, M.; Vekariya, N.; Gajera, R. Solubility of enrofloxacin sodium in various solvents at various temperatures J. Chem. Eng. Data 2008, 53 (12) 2897-2899
8. Sun, H.; Wang, J. Solubility of lovastatin in acetone + water solvent mixtures J. Chem. Eng. Data 2008, 53 (6) 1335-1337
9. Wang, S.; Li, Q. S.; Su, M. G. Solubility of 1 H -1,2,4-triazole in ethanol, 1-propanol, 2-propanol, 1,2-propanediol, ethyl formate, methyl acetate, ethyl acetate, and butyl acetate at (283 to 363) K J. Chem. Eng. Data 2007, 52 (3) 856-858
10. Yang, X.; Wang, X.; Ching, C. B. Solubility of form α and form γ of glycine in aqueous solutions J. Chem. Eng. Data 2008, 53, 1133-1137
11. Song, L.; Gao, Y.; Gong, J. Measurement and correlation of solubility of clopidogrel hydrogen sulfate (metastable form) in lower alcohols J. Chem. Eng. Data 2011, 56, 2553-2556