Overview of P-glycoprotein inhibitors: A rational outlook

Brazilian Journal of Pharmaceutical Sciences

Volumn 48, Issue 3, 2012, Pages 353-367

  Raghava, Kale Mohana ^a   Lakshmi, P K ^a  

^a OSMANIA UNIVERSITY   (India)

Author keywords

Cluster of differentiation 243; Competitive inhibitors; Multidrug resistence; P glycoprotein inhibitors; Sphingolipids

Indexed keywords

CLARITHROMYCIN; COLCHICINE; CYCLOSPORIN; DILTIAZEM; DOXORUBICIN; ERYTHROMYCIN; ESOMEPRAZOLE; FELODIPINE; FENOFIBRATE; GALLOPAMIL; GLYCOPROTEIN P INHIBITOR; LANSOPRAZOLE; MULTIDRUG RESISTANCE PROTEIN; NIFEDIPINE; OMEPRAZOLE; PANTOPRAZOLE; PAROXETINE; PROPAFENONE; QUINIDINE; RESERPINE; RITONAVIR; SERTRALINE; TAMOXIFEN; TOREMIFENE; TRIFLUOPERAZINE; UNINDEXED DRUG; VALSPODAR; VERAPAMIL; VINBLASTINE; YOHIMBINE;

ALLOSTERISM; CHIRALITY; DRUG FORMULATION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SENSITIVITY; DRUG STRUCTURE; HIGH THROUGHPUT SCREENING; HYDROLYSIS; MICHAELIS MENTEN KINETICS; MOLECULAR MODEL; PROTEIN BINDING; PROTEIN TARGETING; PROTEIN TRANSPORT; QUANTITATIVE STRUCTURE ACTIVITY RELATION; REVIEW;

EID: 84868287895     PISSN: 19848250     EISSN: 21759790     Source Type: Journal    
DOI: 10.1590/S1984-82502012000300002     Document Type: Review

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