Design, synthesis and molecular simulation studies of dihydrostilbene derivatives as potent tyrosinase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 17, 2012, Pages 5523-5526

  Vontzalidou, Argyro ^a   Zoidis, Grigoris ^a   Chaita, Eliza ^a   Makropoulou, Maria ^a   Aligiannis, Nektarios ^a   Lambrinidis, George ^a   Mikros, Emmanuel ^a   Skaltsounis, Alexios Leandros ^a  

^a UNIVERSITY OF ATHENS   (Greece)

Author keywords

Deoxybenzoins; Dihydrostilbenes; Gallic acid; Kojic acid; Molecular simulations; Tyrosinase inhibitors

Indexed keywords

BENZENE DERIVATIVE; DIHYDROSTILBENE DERIVATIVE; GALLIC ACID; KOJIC ACID; MONOPHENOL MONOOXYGENASE; UNCLASSIFIED DRUG;

ARTICLE; DRUG DESIGN; DRUG SYNTHESIS; HETERONUCLEAR MULTIPLE BOND CORRELATION; HETERONUCLEAR MULTIPLE QUANTUM COHERENCE; HYDROGEN BOND; IC 50; PROTON NUCLEAR MAGNETIC RESONANCE; STRUCTURE ACTIVITY RELATION;

BACTERIA; BENZOIN; DRUG DESIGN; ENZYME INHIBITORS; FUNGI; MOLECULAR DOCKING SIMULATION; MONOPHENOL MONOOXYGENASE; PYRONES; STILBENES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84865123076     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.07.029     Document Type: Article

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