Synthesis of N-(1-methyl-1H-indol-3-yl)methyleneamines and 3,3-diaryl-4-(1-methyl-1H-indol-3-yl)azetidin-2-ones as potential antileishmanial agents

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 17, 2012, Pages 5704-5706

  Singh, Girija S ^a   Al Kahraman, Yasser M S A ^b   Mpadi, Disah ^a   Yasinzai, Masoom ^c  

^a UNIVERSITY OF BOTSWANA   (Botswana)

^b UNIVERSITY OF BALOCHISTAN   (Pakistan)

^c QUAID I AZAM UNIVERSITY   (Pakistan)

Author keywords

1 Methyl 1H indole; Antileishmanial; Azetidin 2 ones; Azomethines

Indexed keywords

(1 METHYL 1H INDOL 3 YL)METHYLENEAMINE DERIVATIVE; 3,3 DIARYL 4 (1 METHYL 1H-INDOL 3 YL)AZETIDIN 2 ONE DERIVATIVE; AMPHOTERICIN B; ANTILEISHMANIAL AGENT; AZETIDINONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; CYCLOADDITION; DRUG SCREENING; DRUG SYNTHESIS; LEISHMANIA MAJOR; NONHUMAN; STAUDINGER REACTION;

ANTIPROTOZOAL AGENTS; AZETIDINES; HUMANS; INDOLES; LEISHMANIA MAJOR; LEISHMANIASIS, CUTANEOUS; STRUCTURE-ACTIVITY RELATIONSHIP;

LEISHMANIA MAJOR;

EID: 84865122422     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.06.081     Document Type: Article

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