Formulation and evaluation of biodegradable polyphenolic microspheres for cancer

International Journal of Pharmacy and Technology

Volumn 4, Issue 2, 2012, Pages 4493-4505

  Sivabalan, M ^a   Gayathri, V ^a   Kiruthika, C ^a   Madhan, B ^b  

^a Mother Theresa Post Graduate and Research Institute of Health Sciences   (India)

^b CENTRAL LEATHER RESEARCH INSTITUTE   (India)

Author keywords

Catechin; Gallic acid; o w solvent evaporation; Polyphenol; Tannic acid

Indexed keywords

CATECHIN; GALLIC ACID; MICROSPHERE; POLYCAPROLACTONE; POLYVINYL ALCOHOL; TANNIN;

ANTINEOPLASTIC ACTIVITY; ARTICLE; BIODEGRADABILITY; CANCER CELL CULTURE; CELL VIABILITY; DRUG CYTOTOXICITY; DRUG FORMULATION; EVAPORATION; HUMAN; HUMAN CELL; IN VITRO STUDY; MICROENCAPSULATION; PARTICLE SIZE; SQUAMOUS CELL CARCINOMA; SURFACE PROPERTY; SUSTAINED DRUG RELEASE;

EID: 84864751510     PISSN: None     EISSN: 0975766X     Source Type: Journal    
DOI: None     Document Type: Article

References (20)

1. Afef Abdelwahwed, Lines bouhlel, Ines skandrani, Kita valenti, Malika kadri, Pascal Guiraud, et al. Study of antimutagenic and antioxidant activities of Gallic acid and 1, 2, 3, 4, 6-pentagalloylglucose from Pistacia lentiscus confimation by microarray expression profiling Chemico-biological Interactions,165 (2007).
2. Alexander Schlachterman, Felix Valle, Kristin M. Wall, Nicolas G. Azios, Linette Castillo, Lymer Morell, A, et al. Cubano and Surangani F Dharmawardhane. Combined reveratrol, quercetin and catechin treatment reduces breast tumour growth in a nude mouse model. Translational Oncology 2008; 1: 19-27.
3. Arts, I.C. and P.C. Hollman. Polyphenols and disease risk in epidemilogic studies. American Journal Clinical Nutrition 2005; 81:317S-325S.
4. rded. Bombay (India): Varghese publication company 1987:453-455.
5. Berchane NS, Carson KH, Rice-ficht AC, Andrews MJ. Effect of mean diameter and polydispersity of PLG microspheres on drug release: experiment and theory. Nt J pharm 2007;337(1-2): 118-12
6. Bin-Chaun ji, Wu-Huei Hsu, Jai-Sing Yang, Te-Chun Hsia and Chi-Cheng Lu. Gallic acid induces Apoptosis via Caspase-3 and Mitochondrion-Dependent pathways invitro and suppresses Lung Xenograft Tumour Growth in-vivo. J. Agric. Food Chem. 2009; 57:7596-7604
7. Chin-Lin Hsu, Wen-Hsieh Lo, and Gow-chin Yen. Gallic Acid induces Apoptosis in 3T3-L1 Pre-dipocytes via a Fas-and Mitochondrial-Mediated Pathways. J. Agric. Food Chem. 2007;55:7359-7365.
8. thed. USA: Merck & Co inc;1989.
9. Ching-Hsein Chen, Tsan-zon liu, Chin-Hui Chen, Chung Hang Wong, Chi-Hung Chen Fung-Jou Luand Ssu Ching Chen. The efficiency of protective effects of tannic acid and gallic acid against hydrogen peroxideinduced oxidative stress and DNA damages in IMR-90 cells. Mol. Nutr. Food Res.2007; 51: 962-968.
10. Dasaratha Dhanaraju. Preparation and characterisation of injectable microsphers of contraceptive hormones. Int.J. Pharm 2003; 268 (1-2): 23-29.
11. Faried A, D. kurnia, L.S. Faried, N. Usman, T. Miyazaki, H. kato and H. Kuwano. The protective effect of ellagic acid and propyl gallate against hydrogen peroxide-induced oxidative stress and DNA damages in IMR-90 cells. International journal of oncology 2007;30:605-613.
12. H. Huatan. Preparation and characterisation of poly (€ caprolactone) polymer blends for the delivery of protiens. Biomaterials 1995;16:1297-1303.
13. James s. Injectable dispersed systems. Formulation, processing and performance. Florida (USA): Janet taylor & francis group, LLC, 2005.
14. Janet Taylor, John r.N. Tayor, Peter S, Belton and Amanda minnar kafirin. Microparticle encapsulation of Catechin and Sorghum Condensed Tannins. J. Agri. Food Chem. 2009; 57:7523-7528.
15. Jayvadan K. Patel, Rakesh P. Patel, Avani F Amin, and Madhabhai M. Patel. Formulation and Evaluation of Mucoadhesive Glipizide Microspheres. AAPS PharmSciTech 2005;6:12-34 (http://www.aapspharmscitech.org).
16. Jayaprakash, S. Mohamed Firthouse, K. Kulaturanpillai, Abhijit and M. Nagarajan. Preparation and evaluation of biodegradable microspheres of Methotrexate. Asian Journal Of Pharmaceutics. 2009;1:32-43.
17. Jeong JC and Lee J. Cho K. Effects of crystalline microstucture on drug release behaviour of Poly €-caprolactone microsphere. J. Control release 2003; 92(3):249-258.
18. DR. Soniya Ramos Biochemistry, Cancer Research, Molecular Biology, 2009. http://www.scitopics.com/Polyphenols_and_cancer.html
19. Kosaraju SL, Dath L and Lawrence A. Preparation and characterisation of chitosan microspheres for antioxidant delivery. Polymer 2006; 64(11):163-167.
20. Eun Young Hwanga, Jae-Wan Huha, Myung-min choia and Soo Young Choi Inhibitory effectts of gallic acid and quercetin on UDP-glucose dehydrogenase activity.2008;582:3793-3797.