Selective non-lipid modulator of LPA5 activity in human platelets

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 16, 2012, Pages 5239-5243

  Kozian, Detlef H ^a   Evers, Andreas ^a   Florian, Peter ^a   Wonerow, Peter ^a   Joho, Sabrina ^a   Nazare, Marc ^a  

^a SANOFI AVENTIS DEUTSCHLAND GMBH   (Germany)

Author keywords

Atherosclerosis; G protein coupled receptor; LPA5 antagonist; LPA5 GPR92; Platelet aggregation

Indexed keywords

LPA5 INHIBITOR; PROTEIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG RECEPTOR BINDING; DRUG SPECIFICITY; HIGH THROUGHPUT SCREENING; THROMBOCYTE; THROMBOCYTE ACTIVATION;

BINDING SITES; BLOOD PLATELETS; COMPUTER SIMULATION; HUMANS; LYSOPHOSPHOLIPIDS; PLATELET ACTIVATION; PROTEIN ISOFORMS; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, LYSOPHOSPHATIDIC ACID;

EID: 84864417552     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.06.057     Document Type: Article

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