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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 15, 2012, Pages 5104-5107

Synthesis and in vitro evaluation of [18F](R)-FEPAQ: A potential PET ligand for VEGFR2

(11) Prabhakaran, Jaya a Arango, Victoria a,b Majo, Vattoly J a Simpson, Norman R a,b Kassir, Suham A b Underwood, Mark D a,b Polavarapu, Hanish a Bruce, Jeffrey N c Canoll, Peter c John Mann, J a,b Dileep Kumar, J S a,b

a New York Presbyterian Columbia University Medical Center (United States)

b NEW YORK STATE PSYCHIATRIC INSTITUTE (United States)

c Columbia University ^* (United States)

Author keywords

Bioimaging; Glioma; PET; Radiotracer; VEGFR2

Indexed keywords

DIMETHYL SULFOXIDE; FLUORINE 18; N (4 BROMO 2 FLUOROPHENYL) 7 ((1 (2 FLUOROETHYL)PIPERIDIN 3 YL)METHOXY 6 METHOXYQUINAZOLIN 4 AMINE F 18; TERT BUTYL 3 (HYDROXYMETHYL)PIPERIDINE 1 CARBOXYLATE; UNCLASSIFIED DRUG; VASCULOTROPIN RECEPTOR 2;

ARTICLE; AUTORADIOGRAPHY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; GLIOBLASTOMA; HUMAN; HUMAN CELL; HUMAN TISSUE; NEUROIMAGING; POSITRON EMISSION TOMOGRAPHY; RADIOCHEMISTRY;

BRAIN; DRUG EVALUATION, PRECLINICAL; FLUORINE RADIOISOTOPES; GLIOMA; HUMANS; LIGANDS; POSITRON-EMISSION TOMOGRAPHY; QUINAZOLINES; RADIOPHARMACEUTICALS; STEREOISOMERISM; VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR-2;

EID: 84863986268 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.05.099 Document Type: Article

Times cited : (7)

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- KDR in Vitro Enzymatic Binding Assay Was Performed by Calipers Life Sciences Discovery and Alliance Services

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