Imidazo[1,2-a]pyridines that directly interact with hepatitis C NS4B: Initial preclinical characterization

ACS Medicinal Chemistry Letters

Volumn 3, Issue 7, 2012, Pages 565-569

  Shotwell, J Brad ^a   Baskaran, Subramanian ^a   Chong, Pek ^a   Creech, Katrina L ^a   Crosby, Renae M ^a   Dickson, Hamilton ^a   Fang, Jing ^a   Garrido, Dulce ^a   Mathis, Amanda ^a   Maung, Jack ^b   Parks, Derek J ^a   Pouliot, Jeffrey J ^a   Price, Daniel J ^a   Rai, Roopa ^c   Seal, John W ^a   Schmitz, Uli ^d   Tai, Vincent W F ^a   Thomson, Michael ^a   Xie, Mi ^a   Xiong, Zhiping Z ^a   Peat, Andrew J ^a   more..

^a GLAXOSMITHKLINE   (United States)

^b Kanion USA Inc   (United States)

^c AliosBiopharma   (United States)

^d GILEAD SCIENCES   (United States)

Author keywords

hepatitis C virus; imidazo 1,2 a pyridines; NS4B; replicon

Indexed keywords

ANTIVIRUS AGENT; IMIDAZO[1,2 A]PYRIDINE; NONSTRUCTURAL PROTEIN 4B; PROTEINASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG PROTEIN BINDING; HEPATITIS C VIRUS; HUMAN; HUMAN CELL; NONHUMAN; PRIORITY JOURNAL; RAT; VIRUS REPLICATION;

HEPATITIS C VIRUS;

EID: 84863856281     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml300090x     Document Type: Article

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