Synthesis of some 7-arylidene-3-(4-(methylthio)bezyl)-7Hthiazolo[ 2,3-c][1,2,4]triazine-4,6-diones and their anticonvulsant and antimicrobial activity

Journal of Chemical and Pharmaceutical Research

Volumn 4, Issue 5, 2012, Pages 2522-2531

  Lobo, Prajwal L ^a,b   Poojary, Boja ^a   Manjunatha, K ^a,c   Kumar, Vasantha ^a   Chullikana, Anoop ^e   SuchethaKumari, N ^d  

^a MANGALORE UNIVERSITY   (India)

^b Maharani's Science College for Women   (India)

^c NAGARJUNA COLLEGE OF ENGINEERING AND TECHNOLOGY   (India)

^d NITTE DEEMED TO BE UNIVERSITY   (India)

^e Clinigene Intl Ltd   (India)

Author keywords

4 Methylthiobenzyl; Anticonvulsant; Antimicrobial; Thiazole

Indexed keywords

4-METHYLTHIOBENZYL; ACETIC ANHYDRIDES; ANIMAL MODEL; ANTI-MICROBIAL ACTIVITY; ANTICONVULSANT; ANTIMICROBIAL; CHLOROACETIC ACIDS; MULTI-COMPONENT REACTIONS; SODIUM ACETATE; SPECTRAL STUDIES; THIAZOLE;

ACETIC ACID; ALDEHYDES; SPECTROSCOPIC ANALYSIS;

ANIMALS;

1,2,4 TRIAZINE DERIVATIVE; 3 [4 (METHYLSULFANYL)BENZYL] 7 [[5 (2,4,5 TRICHLOROPHENYL)FURAN 2 YL]METHYLIDENE] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 3 [4 (METHYLTHIO)BENZYL] 7 [[5 (2 METHYL 4 NITROPHENYL)FURAN 2 YL]METHYLIDENE] 7H THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6 DIONE; 3 [4 (METHYLTHIO)BENZYL] 7 [[5 (4 METHOXY 2 NITROPHENYL)FURAN 2 YL]METHYLENE] 7H THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6 DIONE; 3 [4 (METHYLTHIO)BENZYL] 7 [[5 (4 NITROPHENYL)FURAN 2 YL]METHYLENE] 7H THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6 DIONE; 7 (2,4 DICHLOROBENZYLIDENE) 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 (3,4 DIMETHOXYBENZYLIDENE) 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 (4 BROMO 2 HYDROXYBENZYLIDENE) 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 (4 HYDROXYBENZYLIDENE) 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 (4 METHOXYBENZYLIDENE) 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 [4 (DIMETHYLAMINO)BENZYLIDENE] 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 [[5 (3 CHLORO 4 FLUOROPHENYL)FURAN 2 YL]METHYLIDENE] 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 [[5 (4 CHLOROPHENYL)FURAN 2 YL]METHYLIDENE] 3 [4 (METHYLSULFANYL)BENZYL] 4H[1,3]THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6(7H)DIONE; 7 ARYLIDENE 3 [4 (METHYLTHIO)BENZYL] 7H THIAZOLO[2,3 C][1,2,4]TRIAZINE 4,6 DIONE DERIVATIVE; ACETIC ACID; ACETIC ANHYDRIDE; ALDEHYDE; CHLOROACETIC ACID; CICLOPIROXOLAMINE; CIPROFLOXACIN; DIAZEPAM; FURFURAL; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBACTERIAL ACTIVITY; ANTICONVULSANT ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS FLAVUS; ASPERGILLUS FUMIGATUS; CONTROLLED STUDY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; FEMALE; IN VITRO STUDY; KLEBSIELLA PNEUMONIAE; MALE; MINIMUM INHIBITORY CONCENTRATION; MOUSE; NONHUMAN; PENICILLIUM MARNEFFEI; PROTECTION; PSEUDOMONAS AERUGINOSA; SEIZURE; STAPHYLOCOCCUS AUREUS; TRICHOPHYTON MENTAGROPHYTES;

EID: 84863114174     PISSN: None     EISSN: 09757384     Source Type: Journal    
DOI: None     Document Type: Article

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