Calcitonin gene-related peptide (CGRP) receptor antagonists: Novel aspartates and succinates

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 8, 2012, Pages 2912-2916

  Luo, Guanglin ^a   Chen, Ling ^a   Pin, Sokhom S ^a   Xu, Cen ^a   Conway, Charles M ^a   MacOr, John E ^a   Dubowchik, Gene M ^a  

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

CGRP antagonist; Migraine

Indexed keywords

ASPARTIC ACID DERIVATIVE; BMS 694153; CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONIST; SUCCINIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; ASYMMETRIC SYNTHESIS; DRUG STRUCTURE; MIGRAINE; STRUCTURE ACTIVITY RELATION;

ASPARTIC ACID; HUMANS; INDAZOLES; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; PROTEIN BINDING; QUINAZOLINONES; RECEPTORS, CALCITONIN GENE-RELATED PEPTIDE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; SUCCINATES;

EID: 84862789720     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.02.066     Document Type: Article

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