An efficient and large scale synthesis of Clopidogrel: Antiplatelet drug

Der Pharma Chemica

Volumn 4, Issue 1, 2012, Pages 479-488

  Madivada, Lokeswara Rao ^a   Anumala, Raghupathi Reddy ^a   Gilla, Goverdhan ^a   Kagga, Mukkanti ^b   Bandichhor, Rakeshwar ^a  

^a DR REDDY'S LABORATORIES LTD   (India)

^b JAWAHARLAL NEHRU TECHNOLOGICAL UNIVERSITY   (India)

Author keywords

Clopidogrel; Electrophilic cyclization; Large scale synthesis; Strecker synthesis

Indexed keywords

2 CHLOROBENZALDEHYDE; 2 PROPANOL; 4,5,6,7 TETRAHYDROTHIENO[2,3 C]PYRIDINE; ACETIC ACID ETHYL ESTER; ACETONE; ACETONITRILE; BENZALDEHYDE DERIVATIVE; CAMPHOR DERIVATIVE; CAMPHOR SULFONIC ACID; CLOPIDOGREL; DICHLOROMETHANE; DIMETHYL SULFATE; DIPOTASSIUM HYDROGEN PHOSPHATE; FORMALDEHYDE; HYDROCHLORIC ACID; METHANOL; METHYL ACETATE; PYRIDINE DERIVATIVE; SOLVENT; SULFONIC ACID DERIVATIVE; SULFURIC ACID; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; CHEMICAL REACTION; CHIRALITY; CONTROLLED STUDY; CYCLIZATION; DRUG PURIFICATION; DRUG PURITY; DRUG STRUCTURE; DRUG SYNTHESIS; ELECTROPHILIC CYCLISATION; LARGE SCALE PRODUCTION; METHODOLOGY; RACEMIC MIXTURE; SOLVENT EFFECT; STRECKER SYNTHESIS; TEMPERATURE; TOSYLATION;

EID: 84860850460     PISSN: None     EISSN: 0975413X     Source Type: Journal    
DOI: None     Document Type: Article

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