Biodynamic parameters of micellar diminazene in sheep erythrocytes and blood plasma

Journal of Veterinary Science

Volumn 12, Issue 4, 2011, Pages 303-307

  Staroverov, Sergey A ^a,b   Sidorkin, Vladimir A ^a   Fomin, Alexander S ^a   Shchyogolev, Sergey Yu ^b   Dykman, Lev A ^b  

^a SARATOV STATE VAVILOV AGRARIAN UNIVERSITY   (Russian Federation)

^b INSTITUTE OF BIOCHEMISTRY AND PHYSIOLOGY OF PLANTS AND MICROORGANISMS   (Russian Federation)

Author keywords

Babesia; Biodynamic; Diminazene; Kinetic; Micelles

Indexed keywords

ANTITRYPANOSOMAL AGENT; DIMINAZENE; POLYSORBATE;

ANIMAL; ANIMAL DISEASE; ARTICLE; BABESIOSIS; BLOOD; CLINICAL TRIAL; CYTOLOGY; DOSE RESPONSE; FEMALE; MALE; METABOLISM; MICELLE; PERITONEUM MACROPHAGE; RAT; SHEEP; SHEEP DISEASE;

ANIMALS; BABESIOSIS; DIMINAZENE; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; MACROPHAGES, PERITONEAL; MALE; MICELLES; POLYSORBATES; RATS; SHEEP; SHEEP DISEASES; TRYPANOCIDAL AGENTS;

ANIMALIA; BABESIA; CYTAUXZOON; MASTIGOPHORA (FLAGELLATES); OVIS ARIES; PIROPLASMIDA; PROTOZOA; THEILERIA; TRYPANOSOMA;

EID: 84860725596     PISSN: 1229845X     EISSN: None     Source Type: Journal    
DOI: 10.4142/jvs.2011.12.4.303     Document Type: Article

References (21)

1. Aboofazeli R, Lawrence MJ. Investigations into the formation and characterization of phospholipid microemul-sions. I. Pseudo-ternary phase diagrams of systems containing water-lecithin-alcohol-isopropyl myristate. Int J Pharm 1993, 93, 161-175.
2. Campbell M, Prankerd RJ, Davie AS, Charman WN. Degradation of berenil a (diminazene aceturate) in acidic aqueous solution. Int J Pharm 2004, 56, 1327-1332.
3. Çomoǧlu T, Gönül N. Microemulsions. J Fac Pharm Ankara 1997, 26, 95-108.
4. Davenas E, Poitevin B, Benveniste J. Effect on mouse peritoneal macrophages of orally administered very high dilutions of silica. Eur J Pharmacol 1987, 135, 313-319.
5. Fubini B, Gasco MR, Gallarate M. Microcalorimetric study of microemulsions as potential drug delivery systems. II. Evaluation of enthalpy in the presence of drugs. Int J Pharm 1989, 50, 213-217.
6. Homer MJ, Aguilar-Delfin I, Telford SR III, Krause PJ, Persing DH. Babesiosis. Clin Microbiol Rev 2000, 13, 451-469.
7. Karvonen E, Kauppinen L, Partanen T, Pösö H. Irrever-sible inhibition of putrescine-stimulated S-adenosyl-L-methionine decarboxylase by Berenil and Pentamidine. Biochem J 1985, 231, 165-169.
8. Klatt P, Hajdu P. Pharmacokinetic investigations on diminazene and rolitetracycline in comparison to a com-bination of both. Vet Res 1976, 99, 372-374.
9. Kwon GS. Polymeric micelles for delivery of poorly water-soluble compounds. Crit Rev Ther Drug Carrier Syst 2003, 20, 357-403.
10. Langer R, Tirrell DA. Designing materials for biology and medicine. Nature 2004, 428, 487-492.
11. Loginova NV, Polozov GI. An Introduction to Pharma-ceutical Chemistry. pp. 70-72, BGU Publishing House, Minsk, 2003. [in Russian].
12. Men'shikov VV. Clinical Laboratory Analytics. Vol. II. Special Analytical Technologies in Clinical Laboratory. pp. 17, Labinform-RAMLD Publishing House, Moscow, 1999. [in Russian].
13. Munshi N, Rapoport N, Pitt WG. Ultrasonic activated drug delivery from pluronic P-105 micelles. Cancer Lett 1997, 118, 13-19.
14. Osborne DU, Ward AJ, O'neill KJ. Microemulsions as topical drug delivery vehicles. I. Characterization of a model system. Drug Dev Ind Pharm 1988, 14, 1203-1219.
15. Pattarino F, Carlotti ME, Gasco MR. Topical delivery systems for azelaic acid: effect of the suspended drug in microemulsion. Pharmazie 1994, 49, 72-73.
16. Penzhorn BL, Lewis BD, de Waal DT, López Rebollar LM. Sterilisation of Babesia canis infections by imidocarb alone or in combination with diminazene. J S Afr Vet Assoc 1995, 66, 157-159.
17. Seddon JM, Templer RH. Polymorphism of lipid-water systems. In: Hoff AJ, Lipowsky R, Sackmann E (eds.). Handbook of Biological Physics. Vol. 1. Chap. 3, pp. 97-160, Elsevier, Amsterdam, 1995.
18. Staroverov SA, Pristensky DV, Yermilov DN, Gabalov KP, Zhemerichkin DA, Sidorkin VA, Shcherbakov AA, Shcyogolev SY, Dykman LA. The effectivity analysis of accumulation of liposomal, micellar, and water-soluble forms of diminazene in cells and in organs. Drug Deliv 2006, 13, 351-355.
19. Staroverov SA, Sidorkin VA, Yermilov DN, Vasilenko OA, Ulizko MA. Pharmacodynamics of a new diminazene drug form. Veterinary 2005, 5, 49-51. [in Russian].
20. Storz H. Immunofluorescene. In: Friemel H (ed.). Immunologische Methods. pp. 128-131, Meditsina Publishing House, Moscow, 1987. [in Russian].
21. Woodburn K, Kessel D. The alteration of plasma lipoproteins by cremophor EL. J Photochem Photobiol B 1994, 22, 197-201.