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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 9, 2012, Pages 3109-3114

Discovery of small molecule HIV-1 integrase dimerization inhibitors

(7) Tintori, Cristina a Demeulemeester, Jonas b Franchi, Luigi a Massa, Silvio a Debyser, Zeger b Christ, Frauke b Botta, Maurizio a,c

a UNIVERSITY OF SIENA (Italy)

b UNIVERSITY OF LEUVEN (Belgium)

c Temple University (United States)

Author keywords

AlphaScreen; Dimerization; HIV 1 integrase; Protein protein interactions

Indexed keywords

INTEGRASE; INTEGRASE DIMERIZATION INHIBITOR; INTEGRASE INHIBITOR; SMALL MOLECULE TRANSPORT AGENT; UNCLASSIFIED DRUG;

ARTICLE; BIOLOGY; CATALYSIS; DIMERIZATION; DRUG ACTIVITY; DRUG STRUCTURE; HUMAN IMMUNODEFICIENCY VIRUS 1; MOLECULE; NONHUMAN; STRUCTURE ACTIVITY RELATION;

COMPUTER SIMULATION; DRUG DISCOVERY; DRUG EVALUATION, PRECLINICAL; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; PROTEIN MULTIMERIZATION;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 84859812848 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.03.064 Document Type: Article

Times cited : (28)

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