Practical asymmetric synthesis of (+)-erythro mefloquine hydrochloride

Organic Process Research and Development

Volumn 16, Issue 3, 2012, Pages 461-463

  Hems, William P ^a   Jackson, William P ^a   Nightingale, Peter ^b   Bryant, Rob ^c  

^a BRUNEL UNIVERSITY   (United Kingdom)

^b Development Chemicals Limited   (United Kingdom)

^c NONE

Author keywords

[No Author keywords available]

Indexed keywords

ENANTIOSELECTIVITY; KETONES;

ASYMMETRIC SYNTHESIS; COST-EFFICIENT; EFFICIENT PROCESS; ENANTIOSELECTIVE; ENANTIOSELECTIVE REDUCTION; ERYTHRO; HYDROGEN SOURCES; PYRIDYL; TRANSFER HYDROGENATIONS;

FORMIC ACID;

EID: 84858633617     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op200354f     Document Type: Article

References (10)

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9. Adam, S. Tetrahedron 1991, 47, 7609
10. Bomches, H.; Hardegger, B. (Hoffmann-La Roche). Purification of Mefloquine Hydrochloride, US Patent 4,507,482, 1985.