-
1
-
-
0002425795
-
Theory and origin of polymorphism
-
Brittain HG, Ed. New York: Marcel Dekker
-
Grant DJW. 1999. Theory and origin of polymorphism. In Polymorphism in pharmaceutical solids; Brittain HG, Ed. New York: Marcel Dekker, pp 1-31.
-
(1999)
Polymorphism in pharmaceutical solids;
, pp. 1-31
-
-
Grant, D.J.W.1
-
2
-
-
0014559313
-
Pharmaceutical applications of polymorphism
-
Haleblian JK, McCrone W. 1969. Pharmaceutical applications of polymorphism. J Pharm Sci 58:911-929.
-
(1969)
J Pharm Sci
, vol.58
, pp. 911-929
-
-
Haleblian, J.K.1
McCrone, W.2
-
3
-
-
0035157406
-
Polymorph screening: Influence of solvents on the rate of solvent-mediated polymorphic transformation
-
Gu CH, Young V Jr, Grant DJW. 2001. Polymorph screening: Influence of solvents on the rate of solvent-mediated polymorphic transformation. J Pharm Sci 90:1878-1890.
-
(2001)
J Pharm Sci
, vol.90
, pp. 1878-1890
-
-
Gu, C.H.1
Young Jr., V.2
Grant, D.J.W.3
-
4
-
-
18744373010
-
Identifying the stable polymorph early in the drug discovery-development process
-
Miller JM, Collman BM, Greene LR, Grant DJW, Blackburn AC. 2005. Identifying the stable polymorph early in the drug discovery-development process. Pharm Dev Technol 10:291-297.
-
(2005)
Pharm Dev Technol
, vol.10
, pp. 291-297
-
-
Miller, J.M.1
Collman, B.M.2
Greene, L.R.3
Grant, D.J.W.4
Blackburn, A.C.5
-
5
-
-
34248994636
-
Identification of phase boundaries in anhydrate/hydrate systems
-
Krzyzaniak JF, Williams GR, Ni N. 2007. Identification of phase boundaries in anhydrate/hydrate systems. J Pharm Sci 96:1270-1281.
-
(2007)
J Pharm Sci
, vol.96
, pp. 1270-1281
-
-
Krzyzaniak, J.F.1
Williams, G.R.2
Ni, N.3
-
6
-
-
0037168237
-
Application of slurry bridging experiments at controlled water activities to predict the solid-state conversion between anhydrous and hydrated forms using theophylline as a model drug
-
Ticehurst MD, Storey RA, Watt C. 2002. Application of slurry bridging experiments at controlled water activities to predict the solid-state conversion between anhydrous and hydrated forms using theophylline as a model drug. Int J Pharm 247:1-10.
-
(2002)
Int J Pharm
, vol.247
, pp. 1-10
-
-
Ticehurst, M.D.1
Storey, R.A.2
Watt, C.3
-
7
-
-
0029074760
-
Inferring thermodynamic stability relationship of polymorphs from melting data
-
Yu L. 1995. Inferring thermodynamic stability relationship of polymorphs from melting data. J Pharm Sci 84:966-974.
-
(1995)
J Pharm Sci
, vol.84
, pp. 966-974
-
-
Yu, L.1
-
8
-
-
27744509918
-
Measuring free-energy difference between crystal polymorphs through eutectic melting
-
Yu L, Huang J, Jones KJ. 2005. Measuring free-energy difference between crystal polymorphs through eutectic melting. J Phys Chem B 109:19915-19922.
-
(2005)
J Phys Chem B
, vol.109
, pp. 19915-19922
-
-
Yu, L.1
Huang, J.2
Jones, K.J.3
-
9
-
-
77951619640
-
Varenicline l-tartrate crystal forms: Characterization through crystallography, spectroscopy and thermodynamics
-
Murphy BJ, Huang J, Casteel MJ, Cobani A, Krzyzaniak JF. 2010. Varenicline l-tartrate crystal forms: Characterization through crystallography, spectroscopy and thermodynamics. J Pharm Sci 99:2766-2776.
-
(2010)
J Pharm Sci
, vol.99
, pp. 2766-2776
-
-
Murphy, B.J.1
Huang, J.2
Casteel, M.J.3
Cobani, A.4
Krzyzaniak, J.F.5
-
11
-
-
0031958398
-
Formation of isomorphic desolvates: Creating a molecular vacuum
-
Stephenson GA, Groleau EG, Kleemann RL, Xu W, Rigsbee DR. 1998. Formation of isomorphic desolvates: Creating a molecular vacuum. J Pharm Sci 87:536-542.
-
(1998)
J Pharm Sci
, vol.87
, pp. 536-542
-
-
Stephenson, G.A.1
Groleau, E.G.2
Kleemann, R.L.3
Xu, W.4
Rigsbee, D.R.5
-
12
-
-
33646759962
-
Establishment of correlation between in vitro enzyme binding potency and in vivo pharmacological activity: Application to liver glycogen phosphorylase a inhibitors
-
Yu LJ, Chen Y, Treadway JL, McPherson RK, McCoid SC, Gibbs EM, Hoover DJ. 2006. Establishment of correlation between in vitro enzyme binding potency and in vivo pharmacological activity: Application to liver glycogen phosphorylase a inhibitors. J Pharmacol Exp Ther 317:1230-1237.
-
(2006)
J Pharmacol Exp Ther
, vol.317
, pp. 1230-1237
-
-
Yu, L.J.1
Chen, Y.2
Treadway, J.L.3
McPherson, R.K.4
McCoid, S.C.5
Gibbs, E.M.6
Hoover, D.J.7
-
13
-
-
0017437920
-
Humidity fixed points of binary saturated aqueous solutions
-
Greenspan L. 1977. Humidity fixed points of binary saturated aqueous solutions. J Res Nat Bur Stand 81A:89-96.
-
(1977)
J Res Nat Bur Stand
, vol.81 A
, pp. 89-96
-
-
Greenspan, L.1
-
15
-
-
16444369059
-
Nuclear magnetic resonance investigation of the interaction of water vapor with sildenafil citrate in the solid state
-
Apperley DC, Basford PA, Dallman CI, Harris RK, Kinns M, Marshall PV, Swanson AG. 2005. Nuclear magnetic resonance investigation of the interaction of water vapor with sildenafil citrate in the solid state. J Pharm Sci 94:516-523.
-
(2005)
J Pharm Sci
, vol.94
, pp. 516-523
-
-
Apperley, D.C.1
Basford, P.A.2
Dallman, C.I.3
Harris, R.K.4
Kinns, M.5
Marshall, P.V.6
Swanson, A.G.7
-
17
-
-
32644460308
-
A study of variable hydration states in topotecan hydrochloride
-
Vogt FG, Dell'Orco PC, Diederich AM, Su Q, Wood JL, Zuber GE, Katrincic LM, Mueller RL, Busby DJ, DeBrosse CW. 2006. A study of variable hydration states in topotecan hydrochloride. J Pharm Biomed Anal 40:1080-1088.
-
(2006)
J Pharm Biomed Anal
, vol.40
, pp. 1080-1088
-
-
Vogt, F.G.1
Dell'Orco, P.C.2
Diederich, A.M.3
Su, Q.4
Wood, J.L.5
Zuber, G.E.6
Katrincic, L.M.7
Mueller, R.L.8
Busby, D.J.9
DeBrosse, C.W.10
-
18
-
-
0030722151
-
Solid-state investigation of erythromycin a dihydrate: Structure, NMR spectroscopy, and hygroscopicity
-
Stephenson GA, Stowell JG, Toma PH, Pfeiffer RR, Byrn SR. 1997. Solid-state investigation of erythromycin a dihydrate: Structure, NMR spectroscopy, and hygroscopicity. J Pharm Sci 86:1239-1244.
-
(1997)
J Pharm Sci
, vol.86
, pp. 1239-1244
-
-
Stephenson, G.A.1
Stowell, J.G.2
Toma, P.H.3
Pfeiffer, R.R.4
Byrn, S.R.5
-
19
-
-
34247275857
-
Water activity-mediated control of crystalline phases of an active pharmaceutical ingredient
-
Variankaval N, Lee C, Xu J, Calabria R, Tsou N, Ball R. 2007. Water activity-mediated control of crystalline phases of an active pharmaceutical ingredient. Org Process Res Dev 11:229-236.
-
(2007)
Org Process Res Dev
, vol.11
, pp. 229-236
-
-
Variankaval, N.1
Lee, C.2
Xu, J.3
Calabria, R.4
Tsou, N.5
Ball, R.6
-
20
-
-
0018625999
-
On the polymorphism of pharmaceuticals and other molecular crystals. I. Theory of thermodynamic rules. II. Applicability of thermodynamic rules
-
Burger A, Ramberger R. 1979. On the polymorphism of pharmaceuticals and other molecular crystals. I. Theory of thermodynamic rules. II. Applicability of thermodynamic rules. Mikrochim Acta 2:259-271, 273-316.
-
(1979)
Mikrochim Acta
, vol.2
, pp. 259-271
-
-
Burger, A.1
Ramberger, R.2
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