First enantioselective synthesis of aptazepine

Synthesis

Volumn 2012, Issue 2, 2012, Pages 241-246

  Roszkowski, Piotr ^a   Maurin, Jan K ^b,c   Czarnocki, Zbigniew ^a  

^a UNIVERSITY OF WARSAW   (Poland)

^b NATIONAL MEDICINES INSTITUTE   (Poland)

^c NATIONAL CENTRE FOR NUCLEAR RESEARCH   (Poland)

Author keywords

asymmetric catalysis; asymmetric synthesis; heterocycles; reductions; total synthesis

Indexed keywords

ABSOLUTE CONFIGURATION; ASYMMETRIC CATALYSIS; ASYMMETRIC SYNTHESIS; ASYMMETRIC TRANSFER HYDROGENATION; ENANTIOMERIC PURITY; ENANTIOPURE; ENANTIOSELECTIVE SYNTHESIS; HETEROCYCLES; TOTAL SYNTHESIS;

CHEMISTRY; REDUCTION; SPEECH SYNTHESIS;

X RAY CRYSTALLOGRAPHY;

APTAZAPINE;

ARTICLE; CHIRALITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOSELECTIVITY; HYDROGENATION; REDUCTION; STEREOCHEMISTRY; STEREOISOMERISM; X RAY CRYSTALLOGRAPHY;

EID: 84855716294     PISSN: 00397881     EISSN: 1437210X     Source Type: Journal    
DOI: 10.1055/s-0031-1289646     Document Type: Article

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