SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 2, 2012, Pages 1014-1018

The discovery of potent antagonists of NPBWR1 (GPR7)

(13) Anthony Romero, F a Hastings, Nicholas B a Moningka, Remond a Guo, Zhiqiang a Wang, Ming a Di Salvo, Jerry a Lei, Ying a Trusca, Dorina a Deng, Qiaolin a Tong, Vincent a Terebetski, Jenna L a Ball, Richard G a Ujjainwalla, Feroze a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

Antagonist; Anti obesity; G protein coupled receptor; GPR7; NPBWR1

Indexed keywords

[4 (5 CHLOROPYRIDIN 2 YL)PIPERAZIN 1 YL][4 [[(1 (4 METHOXYPHENYL)ETHYL]AMINO] 2 (THIOPHEN 3 YL)CYCLOHEXYL]METHANONE; ANTIOBESITY AGENT; G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR 7; PROTEIN INHIBITOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING ASSAY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; HIGH THROUGHPUT SCREENING; MOUSE; NONHUMAN; SUBSTITUTION REACTION;

ANIMALS; BENZYLAMINES; CRYSTALLOGRAPHY, X-RAY; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; MICE; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PIPERAZINES; RECEPTORS, G-PROTEIN-COUPLED; RECEPTORS, NEUROPEPTIDE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84855652046 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.11.126 Document Type: Article

Times cited : (6)

References (11)

1
- 0037428459
- S. Brezillon, V. Lannoy, J.D. Franssen, E. Le Poul, V. Dupriez, J. Lucchetti, M. Detheux, and M. Parmentier J. Biol. Chem. 278 2003 776
- (2003) J. Biol. Chem. , vol.278 , pp. 776
- Brezillon, S.¹ Lannoy, V.² Franssen, J.D.³ Le Poul, E.⁴ Dupriez, V.⁵ Lucchetti, J.⁶ Detheux, M.⁷ Parmentier, M.⁸

2
- 0037072769
- R. Fujii, H. Yoshida, S. Fukusumi, Y. Habata, M. Hosoya, Y. Kawamata, T. Yano, S. Hinuma, C. Kitada, T. Asami, M. Mori, Y. Fujisawa, and M. Fujino J. Biol. Chem. 277 2002 34010
- (2002) J. Biol. Chem. , vol.277 , pp. 34010
- Fujii, R.¹ Yoshida, H.² Fukusumi, S.³ Habata, Y.⁴ Hosoya, M.⁵ Kawamata, Y.⁶ Yano, T.⁷ Hinuma, S.⁸ Kitada, C.⁹ Asami, T.¹⁰ Mori, M.¹¹ Fujisawa, Y.¹² Fujino, M.¹³

3
- 0037184091
- Y. Shimomura, M. Harada, M. Goto, T. Sugo, Y. Matsumoto, M. Abe, T. Watanabe, T. Asami, C. Kitada, M. Mori, H. Onda, and M. Fujino J. Biol. Chem. 277 2002 35826
- (2002) J. Biol. Chem. , vol.277 , pp. 35826
- Shimomura, Y.¹ Harada, M.² Goto, M.³ Sugo, T.⁴ Matsumoto, Y.⁵ Abe, M.⁶ Watanabe, T.⁷ Asami, T.⁸ Kitada, C.⁹ Mori, M.¹⁰ Onda, H.¹¹ Fujino, M.¹²

4
- 0038284653
- H. Tanaka, T. Yoshida, N. Miyamoto, T. Motoike, H. Kuroso, K. Shibata, A. Yamanaka, S.C. Williams, S.J. Richardson, N. Tsujino, M.G. Garry, M.R. Lerner, D.S. King, B.F. O'Dowd, T. Sakurai, and M. Yanagisawa Proc. Natl. Acad. Sci. U.S.A. 100 2003 6251
- (2003) Proc. Natl. Acad. Sci. U.S.A. , vol.100 , pp. 6251
- Tanaka, H.¹ Yoshida, T.² Miyamoto, N.³ Motoike, T.⁴ Kuroso, H.⁵ Shibata, K.⁶ Yamanaka, A.⁷ Williams, S.C.⁸ Richardson, S.J.⁹ Tsujino, N.¹⁰ Garry, M.G.¹¹ Lerner, M.R.¹² King, D.S.¹³ O'Dowd, B.F.¹⁴ Sakurai, T.¹⁵ Yanagisawa, M.¹⁶

5
- 43849109597
- M. Hondo, M. Ishii, and T. Sakurai Results Probl. Cell. Differ. 46 2008 239
- (2008) Results Probl. Cell. Differ. , vol.46 , pp. 239
- Hondo, M.¹ Ishii, M.² Sakurai, T.³

6
- 33745002975
- V.R. Jackson, S.H. Lin, Z. Wang, H.P. Nothacker, and O. Civelli J. Comp. Neurol. 497 2006 367
- (2006) J. Comp. Neurol. , vol.497 , pp. 367
- Jackson, V.R.¹ Lin, S.H.² Wang, Z.³ Nothacker, H.P.⁴ Civelli, O.⁵

7
- 33745397752
- Y. Kitamura, H. Tanaka, T. Motoike, M. Ishii, S.C. Williams, M. Yanagisawa, and T. Sakurai Brain Res. 1093 2006 123
- (2006) Brain Res. , vol.1093 , pp. 123
- Kitamura, Y.¹ Tanaka, H.² Motoike, T.³ Ishii, M.⁴ Williams, S.C.⁵ Yanagisawa, M.⁶ Sakurai, T.⁷

8
- 84855713001
- S. Schulz, R. Stumm, and V. Hollt Neurosci. Lett. 16 2007 842
- (2007) Neurosci. Lett. , vol.16 , pp. 842
- Schulz, S.¹ Stumm, R.² Hollt, V.³

9
- 3142718859
- G. Singh, J.J. Maguire, R.E. Kuc, M. Fidock, and A.P. Davenport Brain Res. 1017 2004 222
- (2004) Brain Res. , vol.1017 , pp. 222
- Singh, G.¹ Maguire, J.J.² Kuc, R.E.³ Fidock, M.⁴ Davenport, A.P.⁵

10
- 37349009036
- F. Takenoya, S. Kitamura, H. Kageyama, N. Nonaka, M. Seki, K. Itabashi, Y. Date, M. Nakazato, and S. Shioda Regul. Pept. 145 2008 116
- (2008) Regul. Pept. , vol.145 , pp. 116
- Takenoya, F.¹ Kitamura, S.² Kageyama, H.³ Nonaka, N.⁴ Seki, M.⁵ Itabashi, K.⁶ Date, Y.⁷ Nakazato, M.⁸ Shioda, S.⁹

11
- 19344362055
- A. Levine, R. Winsky-Sommerer, S. Huitron-Resendiz, M. Grace, and L. de Lecea Am. J. Physiol. Regul. Integr. Comp. Physiol. 288 2005 R1727
- (2005) Am. J. Physiol. Regul. Integr. Comp. Physiol. , vol.288 , pp. 1727
- Levine, A.¹ Winsky-Sommerer, R.² Huitron-Resendiz, S.³ Grace, M.⁴ De Lecea, L.⁵

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.