Clinical pharmacokinetic and pharmacodynamic evaluation of transdermal drug delivery systems of salbutamol sulfate

International Journal of Pharmaceutics

Volumn 287, Issue 1-2, 2004, Pages 47-53

  Murthy, S Narasimha ^a   Hiremath, Shobharani R ^b  

^a ROSWELL PARK CANCER INSTITUTE   (United States)

^b AL AMEEN COLLEGE OF PHARMACY   (India)

Author keywords

Bronchodilation; FEV1; Salbutamol sulfate; Transdermal delivery

Indexed keywords

ALKENE DERIVATIVE; HYDROXYPROPYLMETHYLCELLULOSE; MACROGOL 400; PLASTICIZER; POLYISOBUTYLENE; SALBUTAMOL SULFATE; UNCLASSIFIED DRUG;

ADULT; AREA UNDER THE CURVE; ARTICLE; ASTHMA; CLINICAL ARTICLE; CORRELATION ANALYSIS; DRUG BLOOD LEVEL; DRUG CLEARANCE; DRUG DIFFUSION; DRUG ELIMINATION; DRUG FORMULATION; DRUG HALF LIFE; FEMALE; FORCED EXPIRATORY VOLUME; HUMAN; MALE; PRIORITY JOURNAL; STEADY STATE; TRANSDERMAL PATCH; TREATMENT OUTCOME;

ADMINISTRATION, CUTANEOUS; ADULT; ALBUTEROL; BRONCHODILATOR AGENTS; DRUG DELIVERY SYSTEMS; FEMALE; FORCED EXPIRATORY VOLUME; HUMANS; MALE;

EID: 8444233183     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2004.08.018     Document Type: Article

References (23)

1. R.C. Ahrens, and G.D. Smith Albuterol: an adrenergic agent for use in the treatment of asthma pharmacology, pharmacokinetics and clinical use Pharmacotherapy 4 1984 105 121
2. N.R. Badcock, and J.A. Leach Albuterol: transdermal absorption and fingerprick blood-sample contamination from nebulizers Clin. Chem. 35 1989 889
3. B. Berner, G.M. Gerard, H.O. John, J.S. Robert, R.H. Juang, and D.R. Charles Ethanol-water: mutually enhanced transdermal therapeutic system II; skin permeation of ethanol and nitroglycerin J. Pharm. Sci. 78 1989 401 405
4. R.A. Biddlecombe, and S. Pleasance Automated protein precipitation by filtration in the 96-well format J. Chro. Biomed. Appl. 734 1999 257 265
5. Y.W. Chien Transdermal Controlled Medications 1987 Marcel Dekker pp. 127-157
6. S. Crescioli, C.A. Dal, and P. Maestrelli Controlled-release theophylline inhibits early morning airway obstruction and hyperresponsiveness in asthmatic subjects Ann. Allergy Asthma Immunol. 77 1996 106 110
7. A.J. Fairfax, W.R. McNabb, H.J. Davies, and S.G. Spiro Slow release oral salbutamol and aminophylline in nocturnal asthma: relation of overnight changes in lung function and serum drug levels Thorax 35 1980 526 530
8. D. Fishwick, L. Bradshaw, C. Macdonald, R. Beasley, D. Gash, T. Bengtsson, E. Bondesson, and L. Borgstrom Cumulative single-dose design to assess the bronchodilator effects of beta2-agonists in individuals with asthma Am. J. Resp. Crit. Med. 163 2001 474 477
9. K.T. Ghosh, M.J. Habib, K. Childs, and M. Alexander Transdermal delivery of metoprolol I: comparison between hairless mouse and human cadaver skin and effect of n-decylmethyl sulfoxide Int. J. Pharm. 88 1992 391 396
10. M. Gibaldi The basic concept: clearance J. Clin. Pharmacol. 26 1986 330 331
11. H.W. Kelly, and S. Murphy Beta-adrenergic agonists for acute, severe asthma Ann. Pharmacother. 26 1992 81 91
12. B.J. Lipworth, and D.J. Clark Comparative lung delivery of salbutamol given via turbuhaler and Discus dry powder inhaler devices Eur. J. Clin. Pharmacol. 53 1997 47 49
13. R.F.V. Lopez, J.H. Collett, and M.V.L.B. Bentley Influence of cyclodextrin complexation on the in vitro permeation and skin metabolism of dexamethasone Int. J. Pharm. 200 2000 127 132
14. M.S. Marion, G.R. Leonardson, E.R. Rhoades, T.K. Welty, and P.L. Enright Spirometry reference values for American-Indian adults Chest 120 2001 489 495
15. D.J. Morgan, J.D. Paull, B.H. Richmond, E.W. Evered, and S.P. Ziccone Pharmacokinetics of intravenous and oral salbutamol and its sulphate conjugate Br. J. Clin. Pharm. 22 1986 587 593
16. S.N. Murthy, and S.R. Hiremath Formulation and evaluation of controlled-release transdermal patches of theophylline-salbutamol sulfate Drug Dev. Ind. Pharm. 27 2001 1057 1062
17. S.N. Murthy, S.R. Hiremath, and K.L.K. Pranjothy Evaluation of carboxymethyl guar films for the formulation of transdermal therapeutic systems Int. J. Pharm. 272 2004 11 18
18. M.L. Powell, M. Weisberger, R. Gural, M. Chung, J.E. Patrick, E. Radwanski, and S.S. Symchowicz Comparative bioavailability and pharmacokinetics of three formulations of albuterol J. Pharm. Sci. 74 1985 217 219
19. G. Rajeev, S. Cynthia, A. Lisa, S. James, S. Grant, F. Bahram, and N. Thomas Transdermal drug delivery systems of albuterol; in vitro and in vivo studies J. Pharm. Sci. 81 1982 996 1000
20. V.V. Ranade Drug delivery systems 6: transdermal drug delivery J. Clin. Pharmacol. 31 1991 401 418
21. S.D. Roy, S.Y.E. Hou, S.L. Witham, and G.L. Flynn Transdermal delivery of narcotic analgesics: comparative metabolism and permeability of human cadaver skin and hairless mouse skin J. Pharm. Sci. 83 1994 1723 1728
22. K.G. Shah, D.J. Kellerman, S. DeGraw, and P. Koch Pharmacokinetics and pharmacodynamics of cumulative single dose of inhaled salbutamol enantiomers in asthmatic subjects Pulm. Pharmcol. Therap. 12 1999 353 362
23. S.S. Verma, Y.K. Sharma, and S. Arora A multivariate study of some lung function tests at different age groups in healthy Indian males Indian J. Chest Dis. Allied Sci. 2002 44