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Volumn 38, Issue 9, 2011, Pages 1732-1741

One-step radiosynthesis of 18F-AlF-NOTA-RGD2 for tumor angiogenesis PET imaging

Author keywords

18F; Aluminum fluoride; Integrin v 3; Molecular imaging; NOTA; PET; RGD dimer

Indexed keywords

ALUMINUM FLUORIDE 1,4,7 TRIAZACYCLONONANE 1,4,7 TRIACETIC ACID ARGININE GLYCINE ASPARTIC ACID F 18; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG; 1,4,7 TRIAZACYCLONONANE 1,4,7 TRIACETIC ACID; 1,4,7-TRIAZACYCLONONANE-N,N',N''-TRIACETIC ACID; ARGINYL-GLYCYL-ASPARTIC ACID; ARGINYLGLYCYLASPARTIC ACID; DIAGNOSTIC AGENT; HETEROCYCLIC COMPOUND; INTEGRIN; OLIGOPEPTIDE;

EID: 80955178858     PISSN: 16197070     EISSN: 16197089     Source Type: Journal    
DOI: 10.1007/s00259-011-1847-4     Document Type: Article
Times cited : (86)

References (31)
  • 1
    • 0028670833 scopus 로고
    • Integrin αvβ3 antagonists promote tumor regression by inducing apoptosis of angiogenic blood vessels
    • Brooks PC, Montgomery AM, Rosenfeld M, Reisfeld RA, Hu T, Klier G, et al. Integrin αvβ3 antagonists promote tumor regression by inducing apoptosis of angiogenic blood vessels. Cell 1994;79:1157-64.
    • (1994) Cell , vol.79 , pp. 1157-1164
    • Brooks, P.C.1    Montgomery, A.M.2    Rosenfeld, M.3    Reisfeld, R.A.4    Hu, T.5    Klier, G.6
  • 2
    • 58149102321 scopus 로고    scopus 로고
    • Molecular basis of metastasis
    • Chiang AC, Massagué J. Molecular basis of metastasis. N Engl J Med 2008;359:2814-23.
    • (2008) N Engl J Med , vol.359 , pp. 2814-2823
    • Chiang, A.C.1    Massagué, J.2
  • 3
    • 52949124048 scopus 로고    scopus 로고
    • Cancer. The metastasis cascade
    • Klein CA. Cancer. The metastasis cascade. Science 2008;321:1785-7.
    • (2008) Science , vol.321 , pp. 1785-1787
    • Klein, C.A.1
  • 5
    • 0037318003 scopus 로고    scopus 로고
    • Integrin 3 as a therapeutic target for blocking tumor-induced angiogenesis
    • DOI 10.2174/1389450033346830
    • Kumar CC. Integrin αvβ3 as a therapeutic target for blocking tumor-induced angiogenesis. Curr Drug Targets 2003;4:123-31. (Pubitemid 36553584)
    • (2003) Current Drug Targets , vol.4 , Issue.2 , pp. 123-131
    • Kumar, C.C.1
  • 6
    • 84872219330 scopus 로고    scopus 로고
    • MicroPET imaging of integrin α (v) β (3) expressing tumors using (89) Zr-RGD peptides
    • Jacobson O, Zhu L, Niu G, Weiss ID, Szajek LP, Ma Y, et al. MicroPET imaging of integrin α (v) β (3) expressing tumors using (89) Zr-RGD peptides. Mol Imaging Biol 2010.
    • (2010) Mol Imaging Biol
    • Jacobson, O.1    Zhu, L.2    Niu, G.3    Weiss, I.D.4    Szajek, L.P.5    Ma, Y.6
  • 7
    • 77956267966 scopus 로고    scopus 로고
    • Positron emission tomography tracers for imaging angiogenesis
    • Haubner R, Beer AJ, Wang H, Chen X. Positron emission tomography tracers for imaging angiogenesis. Eur J Nucl Med Mol Imaging 2010;37 Suppl 1:S86-103.
    • (2010) Eur J Nucl Med Mol Imaging , vol.37 , Issue.1 SUPPL.
    • Haubner, R.1    Beer, A.J.2    Wang, H.3    Chen, X.4
  • 11
    • 18244376347 scopus 로고    scopus 로고
    • Noninvasive visualization of the activated αvβ3 integrin in cancer patients by positron emission tomography and [18F]Galacto-RGD
    • Haubner R, Weber WA, Beer AJ, Vabuliene E, Reim D, Sarbia M, et al. Noninvasive visualization of the activated αvβ3 integrin in cancer patients by positron emission tomography and [18F]Galacto-RGD. PLoS Med 2005;2:e70.
    • (2005) PLoS Med , vol.2
    • Haubner, R.1    Weber, W.A.2    Beer, A.J.3    Vabuliene, E.4    Reim, D.5    Sarbia, M.6
  • 12
    • 58249127731 scopus 로고    scopus 로고
    • Use of a novel Arg-Gly-Asp radioligand, 18F-AH111585, to determine changes in tumor vascularity after antitumor therapy
    • Morrison MS, Ricketts SA, Barnett J, Cuthbertson A, Tessier J, Wedge SR. Use of a novel Arg-Gly-Asp radioligand, 18F-AH111585, to determine changes in tumor vascularity after antitumor therapy. J Nucl Med 2009;50:116-22.
    • (2009) J Nucl Med , vol.50 , pp. 116-122
    • Morrison, M.S.1    Ricketts, S.A.2    Barnett, J.3    Cuthbertson, A.4    Tessier, J.5    Wedge, S.R.6
  • 13
    • 53749107069 scopus 로고    scopus 로고
    • The biodistribution and radiation dosimetry of the Arg-Gly-Asp peptide 18F-AH111585 in healthy volunteers
    • McParland BJ, Miller MP, Spinks TJ, Kenny LM, Osman S, Khela MK, et al. The biodistribution and radiation dosimetry of the Arg-Gly-Asp peptide 18F-AH111585 in healthy volunteers. J Nucl Med 2008;49:1664-7.
    • (2008) J Nucl Med , vol.49 , pp. 1664-1667
    • McParland, B.J.1    Miller, M.P.2    Spinks, T.J.3    Kenny, L.M.4    Osman, S.5    Khela, M.K.6
  • 17
    • 33747150885 scopus 로고    scopus 로고
    • v3 integrin expression
    • Cai W, Zhang X, Wu Y, Chen X. A thiol-reactive 18F-labeling agent, N-[2-(4-18F-fluorobenzamido) ethyl]maleimide, and synthesis of RGD peptide-based tracer for PET imaging of αvβ3 integrin expression. J Nucl Med 2006;47:1172-80. (Pubitemid 47544912)
    • (2006) Journal of Nuclear Medicine , vol.47 , Issue.7 , pp. 1172-1180
    • Cai, W.1    Zhang, X.2    Wu, Y.3    Chen, X.4
  • 18
    • 52249113335 scopus 로고    scopus 로고
    • Synthesis, 18F-labeling, and in vitro and in vivo studies of bombesin peptides modified with silicon-based building blocks
    • Höhne A, Mu L, Honer M, Schubiger PA, Ametamey SM, Graham K, et al. Synthesis, 18F-labeling, and in vitro and in vivo studies of bombesin peptides modified with silicon-based building blocks. Bioconjug Chem 2008;19:1871-9.
    • (2008) Bioconjug Chem , vol.19 , pp. 1871-1879
    • Höhne, A.1    Mu, L.2    Honer, M.3    Schubiger, P.A.4    Ametamey, S.M.5    Graham, K.6
  • 19
    • 63849316541 scopus 로고    scopus 로고
    • Organofluorosilanes as model compounds for 18F-labeled siliconbased PET tracers and their hydrolytic stability: Experimental data and theoretical calculations (PET=positron emission tomography)
    • Höhne A, Yu L, Mu L, Reiher M, Voigtmann U, Klar U, et al. Organofluorosilanes as model compounds for 18F-labeled siliconbased PET tracers and their hydrolytic stability: experimental data and theoretical calculations (PET=positron emission tomography). Chemistry 2009;15:3736-43.
    • (2009) Chemistry , vol.15 , pp. 3736-3743
    • Höhne, A.1    Yu, L.2    Mu, L.3    Reiher, M.4    Voigtmann, U.5    Klar, U.6
  • 20
    • 51749104170 scopus 로고    scopus 로고
    • Toward [18F]-labeled aryltrifluoroborate radiotracers: In vivo positron emission tomography imaging of stable aryltrifluoroborate clearance in mice
    • Ting R, Harwig C, auf dem Keller U, McCormick S, Austin P, Overall CM, et al. Toward [18F]-labeled aryltrifluoroborate radiotracers: in vivo positron emission tomography imaging of stable aryltrifluoroborate clearance in mice. J Am Chem Soc 2008;130:12045-55.
    • (2008) J Am Chem Soc , vol.130 , pp. 12045-12055
    • Ting, R.1    Harwig, C.2    Auf Dem Keller, U.3    McCormick, S.4    Austin, P.5    Overall, C.M.6
  • 25
    • 77956264376 scopus 로고    scopus 로고
    • 18F-labeled galacto and PEGylated RGD dimers for PET imaging of αvβ3 integrin expression
    • Liu S, Liu Z, Chen K, Yan Y, Watzlowik P, Wester HJ, et al. 18F-labeled galacto and PEGylated RGD dimers for PET imaging of αvβ3 integrin expression. Mol Imaging Biol 2010;12:530-8.
    • (2010) Mol Imaging Biol , vol.12 , pp. 530-538
    • Liu, S.1    Liu, Z.2    Chen, K.3    Yan, Y.4    Watzlowik, P.5    Wester, H.J.6
  • 26
    • 27944452698 scopus 로고    scopus 로고
    • v3 expression in living mice
    • DOI 10.1021/bc0501698
    • Cheng Z, Wu Y, Xiong Z, Gambhir SS, Chen X. Near-infrared fluorescent RGD peptides for optical imaging of integrin αvβ3 expression in living mice. Bioconjug Chem 2005;16:1433-41. (Pubitemid 41681509)
    • (2005) Bioconjugate Chemistry , vol.16 , Issue.6 , pp. 1433-1441
    • Cheng, Z.1    Wu, Y.2    Xiong, Z.3    Gambhir, S.S.4    Chen, X.5
  • 27
    • 79959567221 scopus 로고    scopus 로고
    • Pilot pharmacokinetic and dosimetric studies of [18F] FPPRGD2: A PET radiopharmaceutical agent for imaging αvβ3 integrin levels
    • In press
    • Mittra E, Goris ML, Lagaru AH, Kardan A, Burton L, Berganos R, et al. Pilot pharmacokinetic and dosimetric studies of [18F] FPPRGD2: A PET radiopharmaceutical agent for imaging αvβ3 integrin levels. Radiology. In press 2011.
    • (2011) Radiology
    • Mittra, E.1    Goris, M.L.2    Lagaru, A.H.3    Kardan, A.4    Burton, L.5    Berganos, R.6
  • 29
    • 75749091879 scopus 로고    scopus 로고
    • Evaluation of a (64) Cu-labeled cystine-knot peptide based on agouti-related protein for PET of tumors expressing αvβ3 integrin
    • Jiang L, Kimura RH, Miao Z, Silverman AP, Ren G, Liu H, et al. Evaluation of a (64) Cu-labeled cystine-knot peptide based on agouti-related protein for PET of tumors expressing αvβ3 integrin. J Nucl Med 2010;51:251-8.
    • (2010) J Nucl Med , vol.51 , pp. 251-258
    • Jiang, L.1    Kimura, R.H.2    Miao, Z.3    Silverman, A.P.4    Ren, G.5    Liu, H.6
  • 31
    • 34447336118 scopus 로고    scopus 로고
    • v3 integrin expression
    • DOI 10.2967/jnumed.107.039859
    • Li ZB, Cai W, Cao Q, Chen K, Wu Z, He L, et al. (64) Cu-labeled tetrameric and octameric RGD peptides for small-animal PET of tumor αvβ3 integrin expression. J Nucl Med 2007;48:1162-71. (Pubitemid 47052657)
    • (2007) Journal of Nuclear Medicine , vol.48 , Issue.7 , pp. 1162-1171
    • Li, Z.-B.1    Cai, W.2    Cao, Q.3    Chen, K.4    Wu, Z.5    He, L.6    Chen, X.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.