메뉴 건너뛰기




Volumn 16, Issue 6, 2011, Pages 637-644

Formulation, characterization and in vitro evaluation of theophylline-loaded Eudragit RS 100 microspheres prepared by an emulsion-solvent diffusion/evaporation technique

Author keywords

Aluminum tristearate; Dispersing agent; Drug release; Eudragit RS 100; Microspheres; Theophylline anhydrous

Indexed keywords

ACETONE; ALUMINUM DERIVATIVE; ALUMINUM TRISTEARATE; EUDRAGIT RS; METHANOL; MICROSPHERE; PARAFFIN; THEOPHYLLINE; UNCLASSIFIED DRUG;

EID: 80755168159     PISSN: 10837450     EISSN: 10979867     Source Type: Journal    
DOI: 10.3109/10837450.2010.508075     Document Type: Article
Times cited : (30)

References (30)
  • 1
    • 0036875661 scopus 로고    scopus 로고
    • Preparation and characterization of drug-loaded polymethacrylate microspheres by an emulsion solvent evaporation method
    • DOI 10.1080/0265204021000022770
    • Kim BK, Hwang SJ, Park JB, Park HJ. Preparation and characterization of drug-loaded polymethacrylate microspheres by an emulsion solvent evaporation method. J Microencapsul 2002;19:811-822. (Pubitemid 36149841)
    • (2002) Journal of Microencapsulation , vol.19 , Issue.6 , pp. 811-822
    • Kim, B.K.1    Hwang, S.J.2    Park, J.B.3    Park, H.J.4
  • 2
    • 51649129933 scopus 로고    scopus 로고
    • Microencapsulation by solvent evaporation: State of the art for process engineering approaches
    • Li M, Rouad O, Poncelet D. Microencapsulation by solvent evaporation: State of the art for process engineering approaches. Int J Pharm 2008;363:26-39.
    • (2008) Int J Pharm , vol.363 , pp. 26-39
    • Li, M.1    Rouad, O.2    Poncelet, D.3
  • 3
    • 0022650603 scopus 로고    scopus 로고
    • Te current status of solid dispersions
    • Ford JL. Te current status of solid dispersions. Pharm Acta Helv 86;61:69-88.
    • Pharm Acta Helv , vol.86 , Issue.61 , pp. 69-88
    • Ford, J.L.1
  • 4
    • 0022531912 scopus 로고
    • Application of solid dispersions with enteric coating agents to overcome some pharmaceutical problems
    • Hasegawa A, Kawamura R, Nakagawa H, Sugimoto I. Application of solid dispersions with enteric coating agents to overcome some pharmaceutical problems. Chem Pharm Bull 1986;4:2183-2190. (Pubitemid 16087549)
    • (1986) Chemical and Pharmaceutical Bulletin , vol.34 , Issue.5 , pp. 2183-2190
    • Hasegawa, A.1    Kawamura, R.2    Nakagawa, H.3    Sugimoto, I.4
  • 5
    • 0000853493 scopus 로고
    • Chemistry and application properties of polymethacrylate coating systems
    • McGinity JW editor New York: Marcel Dekker
    • Lehmann K. Chemistry and application properties of polymethacrylate coating systems In: McGinity JW, editor. Aqueous polymeric coating for pharmaceutical dosage forms. New York: Marcel Dekker; 1989:153-245.
    • (1989) Aqueous Polymeric Coating for Pharmaceutical Dosage Forms , pp. 153-245
    • Lehmann, K.1
  • 6
    • 0029076832 scopus 로고
    • Physicochemical evaluation of acetylsalicylic acid-Eudragit RS 100 microspheres prepared using a solvent partition method
    • Vachon MG, Nairn JG. Physicochemical evaluation of acetylsalicylic acid-Eudragit RS 100 microspheres prepared using a solvent partition method. J Microencapsul 1995;12:287-305.
    • (1995) J Microencapsul , vol.12 , pp. 287-305
    • Vachon, M.G.1    Nairn, J.G.2
  • 7
    • 0348048798 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of Eudragit microspheres containing acetazolamide
    • DOI 10.1016/j.ijpharm.2003.09.015
    • Haznedar S, Dortunc B. Preparation and in vitro evaluation of Eudragit microspheres containing acetazolamide. Int J Pharm 2004;269:131-140. (Pubitemid 38032830)
    • (2004) International Journal of Pharmaceutics , vol.269 , Issue.1 , pp. 131-140
    • Haznedar, S.1    Dortunc, B.2
  • 8
    • 0023268639 scopus 로고
    • Radioprotective activity of ethylcellulose microspheres containing WR 2721, after oral administration
    • Fatome M, Courteille F, Laval JD, Roman V. Radioprotective activity of ethylcellulose microspheres containing WR 272, after oral administration. Int J Pharm 1987;52:21-29. (Pubitemid 17104595)
    • (1987) International Journal of Radiation Biology , vol.52 , Issue.1 , pp. 21-29
    • Fatome, M.1    Courteille, F.2    Laval, J.D.3    Roman, V.4
  • 9
    • 33646683064 scopus 로고    scopus 로고
    • In vitro gentamicin release from commercially available calcium-phosphate bone substitutes infuence of carrier type on duration of the release profle BMC
    • Stallmann HP, Faber C, Bronckers AL, Amerongen AVN, Wuisman PI. In vitro gentamicin release from commercially available calcium-phosphate bone substitutes infuence of carrier type on duration of the release profle BMC. Musculoskelet Disord 2006;7:18.
    • (2006) Musculoskelet Disord , vol.7 , pp. 18
    • Stallmann, H.P.1    Faber, C.2    Bronckers, A.L.3    Avn, A.4    Wuisman, P.I.5
  • 10
    • 0027536260 scopus 로고
    • Preparation and characterization of cisplatin-loaded polymethyl methacrylate microspheres
    • DOI 10.1016/0378-5173(93)90248-E
    • Mestiri M, Puisieux F, Benoit JP. Preparation and characterization of cisplatin-loaded polymethyl methacrylate microspheres. Int J Pharm 1993;89:229-234. (Pubitemid 23067158)
    • (1993) International Journal of Pharmaceutics , vol.89 , Issue.3 , pp. 229-234
    • Mestiri, M.1    Puisieux, F.2    Benoit, J.P.3
  • 11
    • 68649094176 scopus 로고    scopus 로고
    • Particle size design of PLGA microspheres for pulmonary drug delivery: Mathematical modeling and statistical optimization using response surface methodology
    • Hamishekar H, Emami J, Najafabadi AR, Gilani K, Minaiyan M, Mahdavai H, Nokhodchi A. Particle size design of PLGA microspheres for pulmonary drug delivery: Mathematical modeling and statistical optimization using response surface methodology. J Microencapsul 2009;26:1-8.
    • (2009) J Microencapsul , vol.26 , pp. 1-8
    • Hamishekar, H.1    Emami, J.2    Najafabadi, A.R.3    Gilani, K.4    Minaiyan, M.5    Mahdavai, H.6    Nokhodchi, A.7
  • 12
    • 0042848556 scopus 로고    scopus 로고
    • Release profiles of theophylline from microspheres consisting of dextran derivatives and cellulose acetate butyrate: Effect of polyion complex formation
    • DOI 10.1081/DDC-120021779
    • Miyazaki Y, Yakou S, Nagai T, Takayama, K. Release profles of theophylline from microspheres consisting of dextran derivatives and cellulose acetate butyrate: Efect of polyion complex formation. Drug Dev Ind Pharm 2003;29:795-804. (Pubitemid 36899886)
    • (2003) Drug Development and Industrial Pharmacy , vol.29 , Issue.7 , pp. 795-804
    • Miyazaki, Y.1    Yakou, S.2    Nagai, T.3    Takayama, K.4
  • 13
    • 34147148609 scopus 로고    scopus 로고
    • Efect of the dispersion of Eudragit S100 powder on the properties of cellulose acetate butyrate microspheres containing theophylline made by the emulsion-solvent evaporation method
    • Obaidat WM, Obaidat IM. Efect of the dispersion of Eudragit S100 powder on the properties of cellulose acetate butyrate microspheres containing theophylline made by the emulsion-solvent evaporation method. J Microencap 2007;24:263-273.
    • (2007) J Microencap , vol.24 , pp. 263-273
    • Obaidat, W.M.1    Obaidat, I.M.2
  • 14
    • 33744902106 scopus 로고    scopus 로고
    • Preparation and evaluation of Eudragit S 100 microspheres as pH-sensitive release preparations for piroxicam and theophylline using the emulsion-solvent evaporation method
    • DOI 10.1080/02652040500435337, PII G1861660616890
    • Obaidat WM, Price JC. Preparation and evaluation of eudragite S100 microspheres as pH-sensitive release preparation for piroxicam and theophylline using the emulsionsolvent evaporation method. J Microencap 2006;23:195-202. (Pubitemid 43840670)
    • (2006) Journal of Microencapsulation , vol.23 , Issue.2 , pp. 195-202
    • Obeidat, W.M.1    Price, J.C.2
  • 15
    • 0028793206 scopus 로고
    • Evaluation of an aliphatic polyurethane as a microsphere matrix for sustained theophylline delivery
    • Subhaga CS, Ravi KG, Sunny MC, Jayakrishnan SA. Evaluation of an aliphatic polyurethane as a microsphere matrix for sustained theophylline delivery. J Microencap 1995;12:617-625.
    • (1995) J Microencap , vol.12 , pp. 617-625
    • Subhaga, C.S.1    Ravi, K.G.2    Sunny, M.C.3    Jayakrishnan, S.A.4
  • 16
    • 79951686969 scopus 로고    scopus 로고
    • Evaluation of drug-polymer interaction in polymeric microspheres containing diltiazem hydrochloride
    • Türk CT, Hasçiçek C, Gönül N. Evaluation of drug-polymer interaction in polymeric microspheres containing diltiazem hydrochloride. J Term Analys Calori 2009;95:865-869.
    • (2009) J Term Analys Calori , vol.95 , pp. 865-869
    • Türk, C.T.1    Hasçiçek, C.2    Gönül, N.3
  • 17
    • 0022826259 scopus 로고
    • Eudragit RS and RL (acrylic resins) microcapsules at pH insensitive and sustained release preparations of ketoprofen
    • Goto S, Kawata M, Nakamura M, Maekauwa K, Ayoam AT. Eudragit RS and RL (acrylic esins) microcapsules as pH insensitive and sustained release preparations of ketoprofen. J Microencapsul 1986;293-304. (Pubitemid 17220750)
    • (1986) Journal of Microencapsulation , vol.3 , Issue.4 , pp. 293-304
    • Goto, S.1    Kawata, M.2    Nakamura, M.3
  • 18
    • 0022839358 scopus 로고
    • Eudragit E, L and S (acrylic resins) microcapsules as pH sensitive release preparations of ketoprofen
    • Goto S, Kawata M, Nakamura M, Maekauwa K, Ayoam AT. Eudragit E, L and S (acrylic resins) microcapsules as pH sensitive release preparations of ketoprofen. J Microencapsul 1986;3: 305-316. (Pubitemid 17220751)
    • (1986) Journal of Microencapsulation , vol.3 , Issue.4 , pp. 305-316
    • Goto, S.1    Kawata, M.2    Nakamura, M.3
  • 19
    • 0022445026 scopus 로고
    • Preparation and dissolution pattern of Eudragit RS microcapsules containing ketoprofen
    • Kawata M, Nakamura M, Goto S, Aoyama, T. Preparation and dissolution pattern of Eudragit RS microcapsules containing ketoprofen. Chem Pharm Bull 1986;34:2618-2623. (Pubitemid 16056469)
    • (1986) Chemical and Pharmaceutical Bulletin , vol.34 , Issue.6 , pp. 2618-2623
    • Kawata, M.1    Nakamura, M.2    Goto, S.3    Aoyama, T.4
  • 20
    • 0030729177 scopus 로고    scopus 로고
    • Preparation of polymeric microspheres by the solvent evaporation method using sucrose stearate as a droplet stabilizer
    • Yuksel N, Kanik AE, Baykara T. Preparation of polymeric microspheres by the solvent evaporation method using sucrose stearate as droplet stabilizer. J Microencapsul 1997;4:725-733. (Pubitemid 27483090)
    • (1997) Journal of Microencapsulation , vol.14 , Issue.6 , pp. 725-733
    • Yuksel, N.1    Baykara, T.2
  • 21
    • 0025813293 scopus 로고
    • Eudragit e microspheres containing bacampicillin: Preparation by solvent removal methods
    • Bogataj M, Mrhar A, Kristl A, Kozjek F. Eudragit E microspheres containing bacampicillin: Preparation by solvent removal methods. J Microencapsul 1991;8:401-406.
    • (1991) J Microencapsul , vol.8 , pp. 401-406
    • Bogataj, M.1    Mrhar, A.2    Kristl, A.3    Kozjek, F.4
  • 22
    • 0002725227 scopus 로고
    • Formation of degradable drug-loaded microparticles by in-liquid drying processes
    • Donbrow M editor London: CRC Press
    • Ties C. Formation of degradable drug-loaded microparticles by in-liquid drying processes In: Donbrow M, editor. Microcapsules and nanoparticles in medicine and pharmacy. London: CRC Press; 1992:47-71.
    • (1992) Microcapsules and Nanoparticles in Medicine and Pharmacy , pp. 47-71
    • Ties, C.1
  • 23
    • 0028329379 scopus 로고
    • Preparation and evaluation of sustained release microspheres of terbutaline sulfate
    • Kim CK, Kim MJ, Oh KH. Preparation and evaluation of sustained release microspheres of terbutaline sulfate. Int J Pharm 1994;106:213-219.
    • (1994) Int J Pharm , vol.106 , pp. 213-219
    • Kim, C.K.1    Kim, M.J.2    Oh, K.H.3
  • 24
    • 0028960948 scopus 로고
    • Efect of varying drug loading on particle size distribution and drug release kinetics of verapamil hydrochloride microspheres prepared with cellulose esters
    • Bhardwaj SB, Shukla AJ, Collins CC. Efect of varying drug loading on particle size distribution and drug release kinetics of verapamil hydrochloride microspheres prepared with cellulose esters. J Microcapsul 1995;12:71-81.
    • (1995) J Microcapsul , vol.12 , pp. 71-81
    • Bhardwaj, S.B.1    Shukla, A.J.2    Collins, C.C.3
  • 25
    • 0035806261 scopus 로고    scopus 로고
    • An alternative method to the evaluation of similarity factor in dissolution testing
    • DOI 10.1016/S0378-5173(01)00651-2, PII S0378517301006512
    • Costa P. An alternative method to the evaluation of similarity factor in dissolution testing. Int J Pharm 2001;220:77-83. (Pubitemid 32476843)
    • (2001) International Journal of Pharmaceutics , vol.220 , Issue.1-2 , pp. 77-83
    • Costa, P.1
  • 26
    • 0030954517 scopus 로고    scopus 로고
    • Use of enteric polymers for production of microspheres by extrusion-spheronization
    • DOI 10.1016/S0031-6865(97)00005-8, PII S0031686597000058
    • Varshosaz J, Kennedy RA, Gipps EM. Use of enteric polymers for production of microspheres by extrusion-spheronization. Pharm Acta Helv 1997;72:145-152. (Pubitemid 27246712)
    • (1997) Pharmaceutica Acta Helvetiae , vol.72 , Issue.3 , pp. 145-152
    • Varshosaz, J.1    Kennedy, R.A.2    Gipps, E.M.3
  • 27
    • 58149321881 scopus 로고
    • Study of a theophylline-Eudragit L mixture using a combined system of microscopic fourier-transform infrared spectroscopy and diferential scanning calorimetry
    • Lin SY, Liao CM, Hsiue GH, Liang RC. Study of a theophylline-Eudragit L mixture using a combined system of microscopic fourier-transform infrared spectroscopy and diferential scanning calorimetry. Termochmica Acta 1995;245:153-166.
    • (1995) Termochmica Acta , vol.245 , pp. 153-166
    • Lin, S.Y.1    Liao, C.M.2    Hsiue, G.H.3    Liang, R.C.4
  • 29
    • 2342652446 scopus 로고    scopus 로고
    • Mathematical comparison of dissolution profles
    • Moore, JW, Flanner HH. Mathematical comparison of dissolution profles. Pharm Technol 1996;20:64-74.
    • (1996) Pharm Technol , vol.20 , pp. 64-74
    • Moore, J.W.1    Flanner, H.H.2
  • 30
    • 0034687583 scopus 로고    scopus 로고
    • Comparison of in vitro dissolution profles by ANOVA-based, model dependent and independent methods
    • Yuksel N, Kanik AE, Baykara T. Comparison of in vitro dissolution profles by ANOVA-based, model dependent and independent methods. Int J Pharm 2000;209:57-67.
    • (2000) Int J Pharm , vol.209 , pp. 57-67
    • Yuksel, N.1    Kanik, A.E.2    Baykara, T.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.