Design and in vitro evaluation of multiparticulate floating drug delivery system of zolpidem tartarate

Colloids and Surfaces B: Biointerfaces

Volumn 89, Issue 1, 2012, Pages 182-187

  Amrutkar, P P ^a   Chaudhari, P D ^b   Patil, S B ^a  

^a Shri Neminath Jain Brahmacharyashram's   (India)

^b Affiliated to Savitribai Phule Pune University   (India)

Author keywords

Floating drug delivery system; Modified release; Pellets; Zolpidem tartarate

Indexed keywords

BIPHASIC; DELIVERY SYSTEMS; DOSAGE FORMS; DRUG DELIVERY SYSTEM; DRUG RELEASE; EUDRAGIT; GAS GENERATION; IN-VITRO; IN-VITRO EVALUATION; MODIFIED RELEASE; RESIDENCE TIME; SECOND PHASE; SODIUM BICARBONATES; TIME-PERIODS; ZOLPIDEM TARTARATE;

BIOCHEMISTRY; DISSOLUTION; PELLETIZING; POLYMERIC MEMBRANES; POLYMERS; SODIUM;

DRUG DELIVERY;

ZOLPIDEM TARTRATE;

ARTICLE; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG COATING; DRUG DELIVERY SYSTEM; DRUG DOSAGE FORM COMPARISON; DRUG PELLET; DRUG RELEASE; DRUG SOLUBILITY; DRUG STABILITY; IN VITRO STUDY; MEAN RESIDENCE TIME; MULTIPARTICULATE FLOATING DRUG DELIVERY SYSTEM; PRIORITY JOURNAL; PROCESS DESIGN; REPRODUCIBILITY;

DRUG DELIVERY SYSTEMS; DRUG DESIGN; MICROSCOPY, ELECTRON, SCANNING; PYRIDINES; SEROTONIN UPTAKE INHIBITORS; SOLUBILITY;

EID: 80054989178     PISSN: 09277765     EISSN: 18734367     Source Type: Journal    
DOI: 10.1016/j.colsurfb.2011.09.011     Document Type: Article

References (30)

1. Whitehead L., Fell J.T., Collett J.H., Sharma H.L., Smith A.M. Floating dosage forms: an in vivo study demonstrating prolonged gastric retention. J. Controlled Release 1998, 55:3-12.
2. Singh B.N., Kim K.H. Floating drug delivery systems: an approach to oral controlled drug delivery via gastric retention. J. Controlled Release 2000, 63:235-259.
3. Arora S., Ali J., Ahuja A., Khar R.K., Baboota S. Floating drug delivery systems: a review. AAPS PharmSciTech 2005, 6. article 47.
4. Bardonnet P.L., Faivre V., Pugh W.J., Piffaretti J.C., Falson F. Gastroretentive dosage forms: overview and special case of Helicobacter pylori. J. Controlled Release 2006, 111:1-18.
5. Sato Y., Kawashima Y., Takeuchi H., Yamamoto H. In vitro and in vivo evaluation of riboflavin-containing microballoons for a floating controlled drug delivery system in healthy humans. Int. J. Pharm. 2004, 275:97-107.
6. Moes A.J. Gastroretentive dosage forms. Crit. Rev. Ther. Drug Carrier Syst. 1993, 10:143-195.
7. Klausner E.A., Lavy E., Friedman M., Hoffman A. Expandable gastroretentive dosage forms. J. Controlled Release 2003, 90:143-162.
8. Umamaheshwari R.B., Jain S., Bhadra D., Jain N.K. Floating microspheres bearing acetohydroxamic acid for the treatment of Helicobacter pylori. J. Pharm. Pharmacol. 2003, 55:1607-1613.
9. Streubel A., Siepmann J., Bodmeier R. Floating microparticles based on low density foam powder. Int. J. Pharm. 2002, 241:279-292.
10. Talukder R., Fassihi R. Gastroretentive delivery systems: hollow beads. Drug Dev. Ind. Pharm. 2004, 30:405-412.
11. Jain S.K., Awasthi A.M., Jain N.K., Agrawal G. Calcium silicate based microspheres of repaglinide for gastroretentive floating drug delivery: preparation and in vitro characterization. J. Controlled Release 2005, 107:300-309.
12. Hamdani J., Moes A.J., Amighi K. Development and in vitro evaluation of a novel floating multiple unit dosage form obtained by melt pelletization. Int. J. Pharm. 2006, 322:96-103.
13. Roy P., Shahiwala A. Multiparticulate formulation approach to pulsatile drug delivery: current perspectives. J. Controlled Release 2009, 134:74-80.
14. N. Talwar, H. Sen, J.N. Staniforth, Orally administered controlled drug delivery system providing temporal and special control, US patent 6,261,601 (2001).
15. Dey N.S., Majumdar S., Rao M.E.B. Multiparticulate drug delivery systems for controlled release. Trop. J. Pharm. Res. 2008, 7(3):1067-1075.
16. Ghebre-Sellassie I. Pellets: a general overview. Pharmaceutical Pelletization Technology 1989, Marcel Dekker Inc., New York. I. Ghebre-Sellassie (Ed.).
17. Melia C., Washington N., Wilson G.C. Multiparticulate Controlled Release Oral Dosage Forms 1994, Scottish Academic Press Ltd, Edinburgh.
18. Kim S.M., Kim J.S., Hwang S.J. The effect of sodium alginate on physical and dissolution properties of Surelease matrix pellets prepared by a novel pelletizer. Chem. Pharm. Bull. 2007, 55(11):1631-1634.
19. Rajinikanth P.S., Karunagaran L.N., Balasubramaniam J., Mishra B. Formulation and evaluation of clarithromycin microspheres for eradication of Helicobacter pylori. Chem. Pharm. Bull. 2008, 56(12):1658-1664.
20. Wiwattanapatapeea R., Pengnoob A., Kanjanamaneesathianc M., Matchavanicha W., Nilratanad L., Jantharangsrie A. Floating pellets containing bacterial antagonist for control sheath blight of rice: formulations, viability and bacterial release studies. J. Controlled Release 2004, 95:455-462.
21. Costa P., Lobo M.S. Modeling and comparison of dissolution profiles. Eur. J. Pharm. Sci. 2001, 13:123-133.
22. Ritger P.L., Peppas N.A. A simple equation for description of solute release. II. Fickian and anomalous release from swellable devices. J. Controlled Release 1987, 5:37-42.
23. Lopes C.M., Lobo J.M.S., Pinto J.F., Costa P. Compressed mini-tablets as a biphasic delivery system. Int. J. Pharm. 2006, 323:93-100.
24. Lee A.J., King J.R., Hibberd S. Mathematical modeling of the release of drug from porous, non-swelling transdermal drug delivery devices. Math. Med. Biol. 1998, 15(2):135-163.
25. Korsmeyer R.W., Gurny R., Doelkar E., Buri P., Peppas N.A. Mechanism of solute release from porous hydrophilic polymers. Int. J. Pharm. 1983, 15:25-35.
26. Peppas N.A. Analysis of Fickian and non-Fickian drug release from polymers. Pharm. Acta Helv. 1985, 60:110-121.
27. ®SR or hydroxy propyl methyl cellulose. AAPS PharmSciTech 2008, 9(2):577-582.
28. Krogel I., Bodmeier R. Floating or pulsatile drug delivery systems based on coated effervescent cores. Int. J. Pharm. 1999, 187:175-184.
29. Iannuccelli V., Coppi G., Bernabei M.T., Cameroni R. Air compartment multiple-unit system for prolonged gastric residence. Part I. Formulation study. Int. J. Pharm. 1998, 174:47-54.
30. Ichigawa M., Watanabe S., Miyake Y. A new multiple-unit oral floating dosage system. I. Preparation and in vitro evaluation of floating and sustained-release characteristics. J. Pharm. Sci. 1991, 80:1062-1066.