Investigation of the impact of insoluble diluents on the compression and release properties of matrix based sustained release tablets

Powder Technology

Volumn 214, Issue 3, 2011, Pages 375-381

  Vaidya, M P ^a   Avachat, A M ^a  

^a SINHGAD COLLEGE OF PHARMACY   (India)

Author keywords

Compression force; Dibasic calcium phosphate; Heckel's equation; Kawakita equation; Microcrystalline cellulose; Sustained release

Indexed keywords

COMPRESSION FORCE; DIBASIC CALCIUM PHOSPHATE; HECKEL'S EQUATION; KAWAKITA EQUATION; MICROCRYSTALLINE CELLULOSE; SUSTAINED RELEASE;

CALCIUM PHOSPHATE; CELLULOSE; DRUG PRODUCTS; GRANULATION; INVESTMENTS; PHOSPHATES; SODIUM;

DATA COMPRESSION;

CALCIUM PHOSPHATE DIBASIC; DICLOFENAC; DILUENT; HYDROXYPROPYLMETHYLCELLULOSE; MICROCRYSTALLINE CELLULOSE;

ARTICLE; COMPRESSION FORCE; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DENSIFICATION; DRUG DOSAGE FORM COMPARISON; DRUG SOLUBILITY; GRANULE FRAGMENTATION; HECKEL EQUATION; KAWAKITA EQUATION; MATHEMATICAL ANALYSIS; PHYSICAL PARAMETERS; PLASTIC DEFORMATION; SUSTAINED RELEASE PREPARATION; TABLET COMPRESSION; TABLET FRIABILITY; TABLET HARDNESS; TABLET PROPERTY; TABLET THICKNESS; TENSILE STRENGTH;

EID: 80054847800     PISSN: 00325910     EISSN: 1873328X     Source Type: Journal    
DOI: 10.1016/j.powtec.2011.08.035     Document Type: Article

References (20)

1. Bankar G.S., Anderson N.R. Tablets. The Theory and Practice of Industrial Pharmacy 1990, 325. Varghese publishing house, Mumbai. Third ed. L. Lachman, H.A. Lieberman, J.L. Kanig (Eds.).
2. Levina M., Rajabi-Siahboomi A.R. The influence of excipients on drug release from hydroxypropyl methylcellulose matrices. Journal of Pharmaceutical Sciences 2004, 93(11):2746-2754.
3. Thapa P., Ghimire M., Mullen A.B., Stevens H.N.E. Controlled release oral delivery system containing water insoluble drug. Kathmandu University Journal of Science, Engineering Technology 2005, I(1):1-10.
4. Bravo S.A., Lamas M.C., Salomon C.J. In-vitro studies of diclofenac sodium controlled-release from biopolymeric hydrophilic matrices. Journal of Pharmacy and Pharmaceutical Science 2002, 5(3):213-219.
5. Khan G.M., Jiabi Z. Formulation and in vitro evaluation of ibuprofen-carbopol 974PNF controlled release matrix tablets III: influence of co-excipients on release rate of the drug. Journal of Controlled Release 1998, 54:185-190.
6. Ohwoavworhua F.O., Adelakun T.A., Kunle O.O. A comparative evaluation of the flow and compaction characteristics of α-cellulose obtained from waste paper. Tropical Journal of Pharmaceutical Research 2007, 6(1):645-651.
7. Newton J.M., Alderborn G., Nystrom C., Stanley P. The compressive to tensile strength ratio of pharmaceutical compacts. International Journal of Pharmaceutics 1993, 93(1-3):249-251.
8. Haware R.V., Tho I., Bauer-Brand A. Multivariate analysis of relationships between material properties, process parameters and tablet tensile strength for α-lactose monohydrates. European Journal of Pharmaceutics and Biopharmaceutics 2009, 73(3):424-431.
9. Odeku O.A., Itiola O.A. Compaction properties of three types of starch, Iran. Journal of Pharmaceutics Research 2007, 6(1):17-23.
10. Mitrevej A., Faroongsarng D., Sinchaipanid N. Compression behavior of spray dried rice starch. International Journal of Pharmaceutics 1996, 140:61-68.
11. Banker G.S., Anderson N.R. Tablets. The Theory and Practice of Industrial Pharmacy 1987, 293. Varghese Publishing House, Bombay. third ed. L. Lachman, H.A. Liberman, J.L. Kanig (Eds.).
12. Indian Pharmacopoeia, Government of India. Ministry of Health and Family Welfare 1996, I:522-523. Published by the controller of Publications, Delhi.
13. USP 28-NF 23 2005, 626. The United States Pharmacopoeial Convention, Rockville, MD. Asian Edition.
14. Sunada H., Bi Y. Preparation, evaluation and optimization of rapidly disintegrating tablets. Powder Technology 2002, 122:188-198.
15. USP 30-NF 25 2005, 643. The United States Pharmacopoeial Convention, Rockville, MD. Asian Edition.
16. Odeku O.A., Awe O.O., Popoola B., Odeniyi M.A., Itiola O.A. Compression and mechanical properties of tablet formulations containing corn, sweet potato, and cocoyam starches as binders. Pharmaceutical Technology 2005, 82-90.
17. Roberts R.J., Rowe R.C. The effect of the relationship between punch velocity and particle size on the compaction behaviour of materials with varying deformation mechanisms. The Journal of Pharmacy and Pharmacology 1986, 38:566-571.
18. Chowhan C.T., Chow Y.P. Compression behaviour of granulations made with different binders. International Journal of Pharmaceutical Technology and Product Manufacture 1981, 2(1):29-34.
19. Humbert-Droz P., Gurny R., Mordier D., Doelker E. Densification behaviour of drugs presenting availabilty problems. International Journal of Pharmaceutical Technology and Product Manufacture 1983, 4:29-35.
20. Roberts R.J., Rowe R.C. The effect of punch velocity on the compaction of a variety of materials. The Journal of Pharmacy and Pharmacology 1985, 37:377-384.