Acidic triazoles as soluble guanylate cyclase stimulators

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 21, 2011, Pages 6515-6518

  Roberts, R Lee ^a   Bradley, A Paul ^a   Bunnage, E Mark ^a   England, S Katherine ^a   Fobian, M Yvette ^b   Fox, N A David ^a   Gymer, Geoff E ^a   Heasley, Steven E ^b   Molette, Jerome ^a   Smith, Graham L ^a   Fairman, David ^a   Schmidt, Michelle A ^b   Tones, Michael A ^b   Dack, Kevin N ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

^b PFIZER INC   (United States)

Author keywords

Enzyme; Soluble guanylate cyclase; Stimulator; Triazoles

Indexed keywords

2 [1 (2 FLUOROBENZYL) 1H PYRAZOLO[3,4 B]PYRIDIN 3 YL] 5 MORPHOLINO 4,6 PYRIMIDINEDIAMINE; GUANYLATE CYCLASE ACTIVATOR; LIFICIGUAT; RIOCIGUAT; TRIAZOLE DERIVATIVE;

ARTICLE; DRUG POTENCY; DRUG SOLUBILITY; DRUG SYNTHESIS; PHYSICAL CHEMISTRY;

EID: 80054776720     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.08.071     Document Type: Article

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10. This will be published on in the near future.