-
1
-
-
22944457221
-
International Union of Pharmacology. XLVI. G protein-coupled receptor list
-
DOI 10.1124/pr.57.2.5
-
Foord S.M., Bonner T.I., Neubig R.R., Rosser E.M., Pin J.P., and Davenport A.P. International Union of Pharmacology. XLVI. G protein-coupled receptor list Pharmacol. Rev. 57 2005 279 288 (Pubitemid 41043887)
-
(2005)
Pharmacological Reviews
, vol.57
, Issue.2
, pp. 279-288
-
-
Foord, S.M.1
Bonner, T.I.2
Neubig, R.R.3
Rosser, E.M.4
Pin, J.-P.5
Davenport, A.P.6
Spedding, M.7
Harmar, A.J.8
-
2
-
-
77949370572
-
The impact of GPCR structures on pharmacology and structure-based drug design
-
Congreve M., and Marshall F. The impact of GPCR structures on pharmacology and structure-based drug design Br. J. Pharmacol. 159 2010 986 996
-
(2010)
Br. J. Pharmacol.
, vol.159
, pp. 986-996
-
-
Congreve, M.1
Marshall, F.2
-
4
-
-
34447633368
-
Conformational complexity of G-protein-coupled receptors
-
DOI 10.1016/j.tips.2007.06.003, PII S0165614707001459, Allosterism and Collateral Efficacy
-
Kobilka B.K., and Deupi X. Conformational complexity of G-protein-coupled receptors Trends Pharmacol. Sci. 28 2007 397 406 (Pubitemid 47087966)
-
(2007)
Trends in Pharmacological Sciences
, vol.28
, Issue.8
, pp. 397-406
-
-
Kobilka, B.K.1
Deupi, X.2
-
5
-
-
13444261019
-
G protein-coupled receptors: A count of 1001 conformations
-
DOI 10.1111/j.1472-8206.2005.00319.x
-
Vauquelin G., and Van Liefde I. G protein-coupled receptors: a count of 1001 conformations Fundam. Clin. Pharmacol. 19 2005 45 56 (Pubitemid 40204346)
-
(2005)
Fundamental and Clinical Pharmacology
, vol.19
, Issue.1
, pp. 45-56
-
-
Vauquelin, G.1
Van Liefde, I.2
-
6
-
-
79953900818
-
Overcoming barriers to membrane protein structure determination
-
Bill R.M., Henderson P.J., Iwata S., Kunji E.R., Michel H., and Neutze R. Overcoming barriers to membrane protein structure determination Nat. Biotechnol. 29 2011 335 340
-
(2011)
Nat. Biotechnol.
, vol.29
, pp. 335-340
-
-
Bill, R.M.1
Henderson, P.J.2
Iwata, S.3
Kunji, E.R.4
Michel, H.5
Neutze, R.6
-
7
-
-
78651247312
-
Benchmarking membrane protein detergent stability for improving throughput of high-resolution X-ray structures
-
Sonoda Y., Newstead S., Hu N.J., Alguel Y., Nji E., and Beis K. Benchmarking membrane protein detergent stability for improving throughput of high-resolution X-ray structures Structure 19 2011 17 25
-
(2011)
Structure
, vol.19
, pp. 17-25
-
-
Sonoda, Y.1
Newstead, S.2
Hu, N.J.3
Alguel, Y.4
Nji, E.5
Beis, K.6
-
8
-
-
33646011258
-
Fluorescence-detection size-exclusion chromatography for precrystallization screening of integral membrane proteins
-
Kawate T., and Gouaux E. Fluorescence-detection size-exclusion chromatography for precrystallization screening of integral membrane proteins Structure 14 2006 673 681
-
(2006)
Structure
, vol.14
, pp. 673-681
-
-
Kawate, T.1
Gouaux, E.2
-
9
-
-
34250833480
-
A high-throughput method for membrane protein solubility screening: The ultracentrifugation dispersity sedimentation assay
-
DOI 10.1110/ps.072759907
-
Gutmann D.A.P., Mizohata E., Newstead S., Ferrandon S., Henderson P.J.F., van Veen H.W., and Byrne B. A high-throughput method for membrane protein solubility screening: the ultracentrifugation dispersity sedimentation assay Protein Sci. 16 2007 1422 1428 (Pubitemid 46984876)
-
(2007)
Protein Science
, vol.16
, Issue.7
, pp. 1422-1428
-
-
Gutmann, D.A.P.1
Mizohata, E.2
Newstead, S.3
Ferrandon, S.4
Henderson, P.J.F.5
Van Veen, H.W.6
Byrne, B.7
-
10
-
-
57049083012
-
A high-throughput assay for membrane protein stability
-
Postis V.L.G., Deacon S.E., Roach P.C.J., Wright G.S.A., Xia X., and Ingram J.C. A high-throughput assay for membrane protein stability Mol. Membr. Biol. 25 2008 617 624
-
(2008)
Mol. Membr. Biol.
, vol.25
, pp. 617-624
-
-
Postis, V.L.G.1
Deacon, S.E.2
Roach, P.C.J.3
Wright, G.S.A.4
Xia, X.5
Ingram, J.C.6
-
12
-
-
40049099087
-
Microscale Fluorescent Thermal Stability Assay for Membrane Proteins
-
DOI 10.1016/j.str.2008.02.004, PII S0969212608000609
-
Alexandrov A.I., Mileni M., Chien E.Y., Hanson M.A., and Stevens R.C. Microscale fluorescent thermal stability assay for membrane proteins Structure 16 2008 351 359 (Pubitemid 351324124)
-
(2008)
Structure
, vol.16
, Issue.3
, pp. 351-359
-
-
Alexandrov, A.I.1
Mileni, M.2
Chien, E.Y.T.3
Hanson, M.A.4
Stevens, R.C.5
-
13
-
-
36448978229
-
2-adrenergic receptor function
-
DOI 10.1126/science.1150609
-
2-adrenergic receptor function Science 318 2007 1266 1273 (Pubitemid 350172885)
-
(2007)
Science
, vol.318
, Issue.5854
, pp. 1266-1273
-
-
Rosenbaum, D.M.1
Cherezov, V.2
Hanson, M.A.3
Rasmussen, S.G.F.4
Foon, S.T.5
Kobilka, T.S.6
Choi, H.-J.7
Yao, X.-J.8
Weis, W.I.9
Stevens, R.C.10
Kobilka, B.K.11
-
14
-
-
36448995359
-
2-adrenergic G protein-coupled receptor
-
DOI 10.1126/science.1150577
-
2-adrenergic G protein-coupled receptor Science 318 2007 1258 1265 (Pubitemid 350172884)
-
(2007)
Science
, vol.318
, Issue.5854
, pp. 1258-1265
-
-
Cherezov, V.1
Rosenbaum, D.M.2
Hanson, M.A.3
Rasmussen, S.G.F.4
Foon, S.T.5
Kobilka, T.S.6
Choi, H.-J.7
Kuhn, P.8
Weis, W.I.9
Kobilka, B.K.10
Stevens, R.C.11
-
15
-
-
78449305788
-
Structure of the human dopamine D3 receptor in complex with a D2/D3 selective antagonist
-
Chien E.Y., Liu W., Zhao Q., Katritch V., Han G.W., and Hanson M.A. Structure of the human dopamine D3 receptor in complex with a D2/D3 selective antagonist Science 330 2010 1091 1095
-
(2010)
Science
, vol.330
, pp. 1091-1095
-
-
Chien, E.Y.1
Liu, W.2
Zhao, Q.3
Katritch, V.4
Han, G.W.5
Hanson, M.A.6
-
20
-
-
85027927015
-
Structures of the CXCR4 chemokine GPCR with small-molecule and cyclic peptide antagonists
-
Wu B., Chien E.Y., Mol C.D., Fenalti G., Liu W., and Katritch V. Structures of the CXCR4 chemokine GPCR with small-molecule and cyclic peptide antagonists Science 330 2010 1066 1071
-
(2010)
Science
, vol.330
, pp. 1066-1071
-
-
Wu, B.1
Chien, E.Y.2
Mol, C.D.3
Fenalti, G.4
Liu, W.5
Katritch, V.6
-
21
-
-
79960070651
-
Structure of the human histamine H1 receptor complex with doxepin
-
Shimamura T., Shiroishi M., Weyand S., Tsujimoto H., Winter G., and Katritch V. Structure of the human histamine H1 receptor complex with doxepin Nature 475 2011 65 70
-
(2011)
Nature
, vol.475
, pp. 65-70
-
-
Shimamura, T.1
Shiroishi, M.2
Weyand, S.3
Tsujimoto, H.4
Winter, G.5
Katritch, V.6
-
24
-
-
67349173167
-
Thermostabilization of the neurotensin receptor NTS1
-
Shibata Y., White J.F., Serrano-Vega M.J., Magnani F., Aloia A.L., Grisshammer R., and Tate C.G. Thermostabilization of the neurotensin receptor NTS1 J. Mol. Biol. 390 2009 262 277
-
(2009)
J. Mol. Biol.
, vol.390
, pp. 262-277
-
-
Shibata, Y.1
White, J.F.2
Serrano-Vega, M.J.3
Magnani, F.4
Aloia, A.L.5
Grisshammer, R.6
Tate, C.G.7
-
25
-
-
78149501282
-
The properties of thermostabilised G protein-coupled receptors (StaRs) and their use in drug discovery
-
Robertson N., Jazayeri A., Errey J., Baig A., Hurrell E., and Zhukov A. The properties of thermostabilised G protein-coupled receptors (StaRs) and their use in drug discovery Neuropharmacology 60 2010 36 44
-
(2010)
Neuropharmacology
, vol.60
, pp. 36-44
-
-
Robertson, N.1
Jazayeri, A.2
Errey, J.3
Baig, A.4
Hurrell, E.5
Zhukov, A.6
-
26
-
-
70350749580
-
Transferability of thermostabilizing mutations between β-adrenergic receptors
-
Serrano-Vega M.J., and Tate C.G. Transferability of thermostabilizing mutations between β-adrenergic receptors Mol. Membr. Biol. 26 2009 385 396
-
(2009)
Mol. Membr. Biol.
, vol.26
, pp. 385-396
-
-
Serrano-Vega, M.J.1
Tate, C.G.2
-
33
-
-
0037450576
-
Expression and purification of truncated, non-glycosylated turkey beta-adrenergic receptors for crystallization
-
DOI 10.1016/S0005-2736(02)00716-2
-
Warne T., Chirnside J., and Schertler G.F. Expression and purification of truncated, non-glycosylated turkey β-adrenergic receptors for crystallization Biochim. Biophys. Acta 1610 2003 133 140 (Pubitemid 36174004)
-
(2003)
Biochimica et Biophysica Acta - Biomembranes
, vol.1610
, Issue.1
, pp. 133-140
-
-
Warne, T.1
Chirnside, J.2
Schertler, G.F.X.3
-
34
-
-
61849145185
-
Development and crystallization of a minimal thermostabilized G protein-coupled receptor
-
Warne T., Serrano-Vega M.J., Tate C.G., and Schertler G.F. Development and crystallization of a minimal thermostabilized G protein-coupled receptor Protein Expression Purif. 65 2009 204 213
-
(2009)
Protein Expression Purif.
, vol.65
, pp. 204-213
-
-
Warne, T.1
Serrano-Vega, M.J.2
Tate, C.G.3
Schertler, G.F.4
-
35
-
-
3242886780
-
GDAP: A web tool for genome-wide protein disulfide bond prediction
-
O'connor B.D., and Yeates T.O. GDAP: a web tool for genome-wide protein disulfide bond prediction Nucleic Acids Res. 32 2004 W360 W364
-
(2004)
Nucleic Acids Res.
, vol.32
-
-
O'Connor, B.D.1
Yeates, T.O.2
-
36
-
-
0027236794
-
Structural basis of amino acid α helix propensity
-
Blaber M., Zhang X.J., and Matthews B.W. Structural basis of amino acid alpha helix propensity Science 260 1993 1637 1640 (Pubitemid 23247144)
-
(1993)
Science
, vol.260
, Issue.5114
, pp. 1637-1640
-
-
Blaber, M.1
Zhang, X.-J.2
Matthews, B.W.3
-
37
-
-
0031808074
-
A helix propensity scale based on experimental studies of peptides and proteins
-
Pace C.N., and Scholtz J.M. A helix propensity scale based on experimental studies of peptides and proteins Biophys. J. 75 1998 422 427 (Pubitemid 28311831)
-
(1998)
Biophysical Journal
, vol.75
, Issue.1
, pp. 422-427
-
-
Pace, C.N.1
Scholtz, J.M.2
-
38
-
-
63449123226
-
Engineering a G protein-coupled receptor for structural studies: Stabilization of the BLT1 receptor ground state
-
Martin A., Damian M., Laguerre M., Parello J., Pucci B., and Serre L. Engineering a G protein-coupled receptor for structural studies: stabilization of the BLT1 receptor ground state Protein Sci. 18 2009 727 734
-
(2009)
Protein Sci.
, vol.18
, pp. 727-734
-
-
Martin, A.1
Damian, M.2
Laguerre, M.3
Parello, J.4
Pucci, B.5
Serre, L.6
-
39
-
-
0029778268
-
Rhodopsin activation blocked by metal-ion-binding sites linking transmembrane helices C and F
-
DOI 10.1038/383347a0
-
Sheikh S.P., Zvyaga T.A., Lichtarge O., Sakmar T.P., and Bourne H.R. Rhodopsin activation blocked by metal-ion-binding sites linking transmembrane helices C and F Nature 383 1996 347 350 (Pubitemid 26321766)
-
(1996)
Nature
, vol.383
, Issue.6598
, pp. 347-350
-
-
Sheikh, S.P.1
Zvyaga, T.A.2
Lichtarge, O.3
Sakmar, T.P.4
Bourne, H.R.5
-
41
-
-
0031018485
-
Structural instability of a constitutively active G protein-coupled receptor. Agonist-independent activation due to conformational flexibility
-
DOI 10.1074/jbc.272.5.2587
-
Gether U., Ballesteros J.A., Seifert R., Sanders-Bush E., Weinstein H., and Kobilka B.K. Structural instability of a constitutively active G protein-coupled receptor. Agonist-independent activation due to conformational flexibility J. Biol. Chem. 272 1997 2587 2590 (Pubitemid 27053295)
-
(1997)
Journal of Biological Chemistry
, vol.272
, Issue.5
, pp. 2587-2590
-
-
Gether, U.1
Ballesteros, J.A.2
Seifert, R.3
Sanders-Bush, E.4
Weinstein, H.5
Kobilka, B.K.6
-
42
-
-
36248970132
-
2 adrenergic G-protein-coupled receptor
-
DOI 10.1038/nature06325, PII NATURE06325
-
2 adrenergic G-protein-coupled receptor Nature 450 2007 383 387 (Pubitemid 350126755)
-
(2007)
Nature
, vol.450
, Issue.7168
, pp. 383-387
-
-
Rasmussen, S.G.F.1
Choi, H.-J.2
Rosenbaum, D.M.3
Kobilka, T.S.4
Thian, F.S.5
Edwards, P.C.6
Burghammer, M.7
Ratnala, V.R.P.8
Sanishvili, R.9
Fischetti, R.F.10
Schertler, G.F.X.11
Weis, W.I.12
Kobilka, B.K.13
-
44
-
-
69249146075
-
Engineering G protein-coupled receptors to facilitate their structure determination
-
Tate C.G., and Schertler G.F. Engineering G protein-coupled receptors to facilitate their structure determination Curr. Opin. Struct. Biol. 19 2009 386 395
-
(2009)
Curr. Opin. Struct. Biol.
, vol.19
, pp. 386-395
-
-
Tate, C.G.1
Schertler, G.F.2
-
45
-
-
34548529916
-
Crystal Structure of a Thermally Stable Rhodopsin Mutant
-
DOI 10.1016/j.jmb.2007.03.007, PII S0022283607003361
-
Standfuss J., Xie G., Edwards P.C., Burghammer M., Oprian D.D., and Schertler G.F. Crystal structure of a thermally stable rhodopsin mutant J. Mol. Biol. 372 2007 1179 1188 (Pubitemid 47381449)
-
(2007)
Journal of Molecular Biology
, vol.372
, Issue.5
, pp. 1179-1188
-
-
Standfuss, J.1
Xie, G.2
Edwards, P.C.3
Burghammer, M.4
Oprian, D.D.5
Schertler, G.F.X.6
-
46
-
-
0029838532
-
Purification of a rat neurotensin receptor expressed in Escherichia coli
-
Tucker J., and Grisshammer R. Purification of a rat neurotensin receptor expressed in Escherichia coli Biochem. J. 317 1996 891 899 (Pubitemid 26308267)
-
(1996)
Biochemical Journal
, vol.317
, Issue.3
, pp. 891-899
-
-
Tucker, J.1
Grisshammer, R.2
|