메뉴 건너뛰기




Volumn 9, Issue 5, 2011, Pages 338-344

Brazilein, a selective 5-HT receptors antagonist in mouse uterus

Author keywords

5 HT receptor; Brazilein; Mouse; Uterus

Indexed keywords

1 [5 (2 THIENYLMETHOXY) 3 INDOLYL] 2 PROPANAMINE; BRAZILEIN; CISAPRIDE; ERGOMETRINE MALEATE; MESSENGER RNA; SEROTONIN; SEROTONIN 1 RECEPTOR; SEROTONIN 2 RECEPTOR; SEROTONIN ANTAGONIST; SUMATRIPTAN; TANDOSPIRONE; UNCLASSIFIED DRUG;

EID: 80053242003     PISSN: 20956975     EISSN: 18755364     Source Type: Journal    
DOI: 10.3724/SP.J.1009.2011.00338     Document Type: Article
Times cited : (3)

References (33)
  • 1
    • 53149111135 scopus 로고    scopus 로고
    • Molecularbiology of 5-HT receptors [J]
    • Hannon J, Hoyer D Molecularbiology of 5-HT receptors [J]. Behav Brain Res 2008, 195(1):198-213.
    • (2008) Behav Brain Res , vol.195 , Issue.1 , pp. 198-213
    • Hannon, J.1    Hoyer, D.2
  • 2
    • 77749328955 scopus 로고    scopus 로고
    • Endogenous activation of spinal 5-hydroxytryptamine (5-HT) receptors contributes to the thermoregulatory activation of brown adipose tissue [J]
    • Madden CJ, Morrison SF Endogenous activation of spinal 5-hydroxytryptamine (5-HT) receptors contributes to the thermoregulatory activation of brown adipose tissue [J]. Am J Physiol Regul Integr Comp Physiol 2010, 298(3):776-783.
    • (2010) Am J Physiol Regul Integr Comp Physiol , vol.298 , Issue.3 , pp. 776-783
    • Madden, C.J.1    Morrison, S.F.2
  • 3
    • 0021894691 scopus 로고
    • 2 receptors in serotonin-induced contractions of nonvascular smooth muscle [J]
    • 2 receptors in serotonin-induced contractions of nonvascular smooth muscle [J]. J Pharmacol Exp Ther 1985, 232(3):770-774.
    • (1985) J Pharmacol Exp Ther , vol.232 , Issue.3 , pp. 770-774
    • Cohen, M.L.1    Schenck, K.W.2    Colbert, W.3
  • 5
    • 0024340545 scopus 로고
    • Effects of histamine and serotonin on the contractility of isolated pregnant and nonpregnant human myometrium [J]
    • Cruz MA, Gonzalez C, Acevedo CG, et al. Effects of histamine and serotonin on the contractility of isolated pregnant and nonpregnant human myometrium [J]. Gynecol Obstet Invest 1989, 28(1):1-4.
    • (1989) Gynecol Obstet Invest , vol.28 , Issue.1 , pp. 1-4
    • Cruz, M.A.1    Gonzalez, C.2    Acevedo, C.G.3
  • 6
    • 33646803502 scopus 로고    scopus 로고
    • Pharmacological evidence for a functional serotonin-2B receptor in a human uterine smooth muscle cell line [J]
    • Kelly CR, Sharif NA Pharmacological evidence for a functional serotonin-2B receptor in a human uterine smooth muscle cell line [J]. J Pharmacol Exp Ther 2006, 317(3):1254-1261.
    • (2006) J Pharmacol Exp Ther , vol.317 , Issue.3 , pp. 1254-1261
    • Kelly, C.R.1    Sharif, N.A.2
  • 7
    • 84990860428 scopus 로고    scopus 로고
    • Quality standard of Caesalpinia sappan L [J]
    • Wang ZX, Ding Y, Du LJ, et al. Quality standard of Caesalpinia sappan L [J]. Cent South Pharm 2008, 6(4):403-405.
    • (2008) Cent South Pharm , vol.6 , Issue.4 , pp. 403-405
    • Wang, Z.X.1    Ding, Y.2    Du, L.J.3
  • 8
    • 0034252043 scopus 로고    scopus 로고
    • Anticonvulsant compounds from the wood of Caesalpinia sappan L. [J]
    • Baek NI, Jeon SG, Ahn EM, et al. Anticonvulsant compounds from the wood of Caesalpinia sappan L. [J]. Arch Pharm Res 2000, 23(4):344-348.
    • (2000) Arch Pharm Res , vol.23 , Issue.4 , pp. 344-348
    • Baek, N.I.1    Jeon, S.G.2    Ahn, E.M.3
  • 9
    • 0034265647 scopus 로고    scopus 로고
    • Vasorelaxing effects of Caesalpinia sappan involvement of endogenous nitric oxide [J]
    • Xie YW, Ming DS, Xu HX, et al. Vasorelaxing effects of Caesalpinia sappan involvement of endogenous nitric oxide [J]. Life Sci 2000, 67(15):1913-1918.
    • (2000) Life Sci , vol.67 , Issue.15 , pp. 1913-1918
    • Xie, Y.W.1    Ming, D.S.2    Xu, H.X.3
  • 10
    • 47649108805 scopus 로고    scopus 로고
    • Antioxidant activity in vitro of three constituents from Caesalpinia sappan L. [J]
    • Hu J, Yan XL, Wang W, et al. Antioxidant activity in vitro of three constituents from Caesalpinia sappan L. [J]. Tsinghua Sci Technol 2008, 13(4):474-479.
    • (2008) Tsinghua Sci Technol , vol.13 , Issue.4 , pp. 474-479
    • Hu, J.1    Yan, X.L.2    Wang, W.3
  • 11
    • 79958119289 scopus 로고    scopus 로고
    • Extract of the dried heartwood of Caesalpinia sappan L. attenuates collagen-induced arthritis [J]
    • Wang YZ, Sun SQ, Zhou YB Extract of the dried heartwood of Caesalpinia sappan L. attenuates collagen-induced arthritis [J]. Eur J Pharmacol 2011, 136(1):271-278.
    • (2011) Eur J Pharmacol , vol.136 , Issue.1 , pp. 271-278
    • Wang, Y.Z.1    Sun, S.Q.2    Zhou, Y.B.3
  • 12
    • 31144439752 scopus 로고    scopus 로고
    • Study on cardioactive effects of brazilein [J]
    • Zhao YN, Pan Y, Tao JL, et al. Study on cardioactive effects of brazilein [J]. Pharmacology 2006, 76(2):76-83.
    • (2006) Pharmacology , vol.76 , Issue.2 , pp. 76-83
    • Zhao, Y.N.1    Pan, Y.2    Tao, J.L.3
  • 13
    • 31044435056 scopus 로고    scopus 로고
    • Brazilein, an important immunosuppressive component from Caesalpinia sappan L. [J]
    • Ye M, Xie WD, Lei F, et al. Brazilein, an important immunosuppressive component from Caesalpinia sappan L. [J]. Int Immunopharmacol 2006, 6(3):426-432.
    • (2006) Int Immunopharmacol , vol.6 , Issue.3 , pp. 426-432
    • Ye, M.1    Xie, W.D.2    Lei, F.3
  • 14
    • 33847301419 scopus 로고    scopus 로고
    • Brazilein protects the brain against focal cerebral ischemia reperfusion injury correlating to inflammatory response suppression [J]
    • Shen J, Zhang HY, Lin H, et al. Brazilein protects the brain against focal cerebral ischemia reperfusion injury correlating to inflammatory response suppression [J]. Eur J Pharmacol 2007, 558(1-3):88-95.
    • (2007) Eur J Pharmacol , vol.558 , Issue.1-3 , pp. 88-95
    • Shen, J.1    Zhang, H.Y.2    Lin, H.3
  • 15
    • 38549134417 scopus 로고    scopus 로고
    • 2+ entry and ROK, ERK pathways [J]
    • 2+ entry and ROK, ERK pathways [J]. Eur J Pharmacol 2008, 580(3):366-371.
    • (2008) Eur J Pharmacol , vol.580 , Issue.3 , pp. 366-371
    • Shen, J.1    Yip, S.2    Wang, Z.X.3
  • 16
    • 65949116574 scopus 로고    scopus 로고
    • Determination of brazilein in rat plasma after intravenous administration by HPLC [J]
    • Lan JQ, Hu J, Li BN, et al. Determination of brazilein in rat plasma after intravenous administration by HPLC [J]. Biomed Chromatogr 2008, 22(11):1201-1205.
    • (2008) Biomed Chromatogr , vol.22 , Issue.11 , pp. 1201-1205
    • Lan, J.Q.1    Hu, J.2    Li, B.N.3
  • 17
    • 0033305565 scopus 로고    scopus 로고
    • Relaxin up-regulates the nitric oxide biosynthetic pathway in the mouse uterus: involvement in the inhibition of myometrial contractility [J]
    • Bani D, Caterina M, Baccari C, et al. Relaxin up-regulates the nitric oxide biosynthetic pathway in the mouse uterus: involvement in the inhibition of myometrial contractility [J]. Endocrinology 1999, 140(10):4434-4441.
    • (1999) Endocrinology , vol.140 , Issue.10 , pp. 4434-4441
    • Bani, D.1    Caterina, M.2    Baccari, C.3
  • 18
    • 77955267304 scopus 로고    scopus 로고
    • 1A receptor binding and expression in conditional brain-derived neurotrophic factor knock-out mice [J]
    • 1A receptor binding and expression in conditional brain-derived neurotrophic factor knock-out mice [J]. Neuroscience 2010, 169(3):1007-1016.
    • (2010) Neuroscience , vol.169 , Issue.3 , pp. 1007-1016
    • Klein, A.B.1    Santini, M.A.2    Aznar, S.3
  • 20
    • 29444439666 scopus 로고    scopus 로고
    • Serotonin (5-HT) receptor subtypes mediate specific modes of 5-HT-induced signaling and regulation of neurosecretion in gonadotropin-releasing hormone neurons [J]
    • Wada K, Hu L, Mores N, et al. Serotonin (5-HT) receptor subtypes mediate specific modes of 5-HT-induced signaling and regulation of neurosecretion in gonadotropin-releasing hormone neurons [J]. Mol Endocrinol 2006, 20(1):125-135.
    • (2006) Mol Endocrinol , vol.20 , Issue.1 , pp. 125-135
    • Wada, K.1    Hu, L.2    Mores, N.3
  • 21
    • 0009644628 scopus 로고
    • Some quantitative uses of drug antogonists [J]
    • Arunlakshana O, Schild HO Some quantitative uses of drug antogonists [J]. Br J Pharmacol Chemother 1959, 14(1):48-58.
    • (1959) Br J Pharmacol Chemother , vol.14 , Issue.1 , pp. 48-58
    • Arunlakshana, O.1    Schild, H.O.2
  • 22
    • 0036119338 scopus 로고    scopus 로고
    • Molecular, pharmacological and functional diversity of 5-HT receptors [J]
    • Hoyer D, Hannon JP, Martin GR. Molecular, pharmacological and functional diversity of 5-HT receptors [J]. Pharmacol Biochem Behav 2002, 71(4):533-554.
    • (2002) Pharmacol Biochem Behav , vol.71 , Issue.4 , pp. 533-554
    • Hoyer, D.1    Hannon, J.P.2    Martin, G.R.3
  • 23
    • 44649101927 scopus 로고    scopus 로고
    • G protein-coupled receptor dimers: Functional consequences, disease states and drug targets [J]
    • Dalrymple MB, Pfleger KDG, Eidne KA G protein-coupled receptor dimers: Functional consequences, disease states and drug targets [J]. Pharmacol Therap 2008, 118(3):359-371.
    • (2008) Pharmacol Therap , vol.118 , Issue.3 , pp. 359-371
    • Dalrymple, M.B.1    Pfleger, K.D.G.2    Eidne, K.A.3
  • 24
    • 85193581142 scopus 로고    scopus 로고
    • Classification and signaling characteristics of 5-HT receptors. Handbook of Behavioral Neuroscience [M].
    • Bockaert J, Claeysena S, Dumuisa A, et al. Classification and signaling characteristics of 5-HT receptors. Handbook of Behavioral Neuroscience [M]. 2010: 103-121.
    • (2010) , pp. 103-121
    • Bockaert, J.1    Claeysena, S.2    Dumuisa, A.3
  • 25
    • 62449243011 scopus 로고    scopus 로고
    • Characterization of serotonin receptors in pregnant human [J]
    • Cordeaux Y, Pasupathy D, Bacon J, et al. Characterization of serotonin receptors in pregnant human [J]. Myometrium J Pharmacol Exp Ther 2009, 328(3):682-691.
    • (2009) Myometrium J Pharmacol Exp Ther , vol.328 , Issue.3 , pp. 682-691
    • Cordeaux, Y.1    Pasupathy, D.2    Bacon, J.3
  • 26
    • 0025964487 scopus 로고
    • Innervation of the human uterine artery and contractile responses to neuropeptides [J]
    • Ekesbo R, Alm P, Ekström P, et al. Innervation of the human uterine artery and contractile responses to neuropeptides [J]. Gynecol Obstet Invest 1991, 31(1):30-36.
    • (1991) Gynecol Obstet Invest , vol.31 , Issue.1 , pp. 30-36
    • Ekesbo, R.1    Alm, P.2    Ekström, P.3
  • 27
    • 0024273543 scopus 로고
    • Ergometrine-A partial agonist at 5-HT receptors in the uterus isolated from the oestrogen-primed rat [J]
    • Hollingsworth M, Edwards D, Miller M Ergometrine-A partial agonist at 5-HT receptors in the uterus isolated from the oestrogen-primed rat [J]. Eur J Pharmacol 1988, 158(1):79-84.
    • (1988) Eur J Pharmacol , vol.158 , Issue.1 , pp. 79-84
    • Hollingsworth, M.1    Edwards, D.2    Miller, M.3
  • 28
    • 55949088459 scopus 로고    scopus 로고
    • Excitatory and inhibitory 5-hydroxytryptamine (5-HT) receptors expressed in the isolated porcine uterine muscles [J]
    • Nakamura T, Kitazawa T, Cao J, et al. Excitatory and inhibitory 5-hydroxytryptamine (5-HT) receptors expressed in the isolated porcine uterine muscles [J]. Eur J Pharmacol 2008, 600(1-3):123-129.
    • (2008) Eur J Pharmacol , vol.600 , Issue.1-3 , pp. 123-129
    • Nakamura, T.1    Kitazawa, T.2    Cao, J.3
  • 29
    • 0034672622 scopus 로고    scopus 로고
    • Diverse signalling by 5-hydroxytryptamine (5-HT) receptors [J]
    • Petrus JP Diverse signalling by 5-hydroxytryptamine (5-HT) receptors [J]. Biochem Pharmacol 2000, 60(12):1743-1750.
    • (2000) Biochem Pharmacol , vol.60 , Issue.12 , pp. 1743-1750
    • Petrus, J.P.1
  • 30
    • 40849139137 scopus 로고    scopus 로고
    • The role of 5-HT receptor subtypes in the ventrolateral orbital cortex of 5-HT-induced antinociception in the rat [J]
    • Qu CL, Huo FQ, Huang FS, et al. The role of 5-HT receptor subtypes in the ventrolateral orbital cortex of 5-HT-induced antinociception in the rat [J]. Orig Neurosc 2008, 152(2):487-494.
    • (2008) Orig Neurosc , vol.152 , Issue.2 , pp. 487-494
    • Qu, C.L.1    Huo, F.Q.2    Huang, F.S.3
  • 31
    • 60149086219 scopus 로고    scopus 로고
    • Elevated 5-HT 2A receptors in postmortem prefrontal cortex in major depression is associated with reduced activity of protein kinase A [J]
    • Shelton RC, Sanders-Bush E, Manier DH, et al. Elevated 5-HT 2A receptors in postmortem prefrontal cortex in major depression is associated with reduced activity of protein kinase A [J]. Neuroscience 2009, 158(4):1406-1415.
    • (2009) Neuroscience , vol.158 , Issue.4 , pp. 1406-1415
    • Shelton, R.C.1    Sanders-Bush, E.2    Manier, D.H.3
  • 32
    • 0036765561 scopus 로고    scopus 로고
    • Differential activation of Gq/11 and Gi3 proteins at 5-hydroxytryptamine 2C receptors revealed by antibody capture assays: influence of receptor reserve and relationship to agonist-directed trafficking [J]
    • Cussac D, Newman-Tancredi A, Duqueyroix D, et al. Differential activation of Gq/11 and Gi3 proteins at 5-hydroxytryptamine 2C receptors revealed by antibody capture assays: influence of receptor reserve and relationship to agonist-directed trafficking [J]. Mol Pharmacol 2002, 62(3):578-589.
    • (2002) Mol Pharmacol , vol.62 , Issue.3 , pp. 578-589
    • Cussac, D.1    Newman-Tancredi, A.2    Duqueyroix, D.3
  • 33
    • 0036892263 scopus 로고    scopus 로고
    • Phospholipase D activation by endogenous 5-hydroxytryptamine 2C receptors is mediated by Galpha13 and pertussis toxin-insensitive Gbetagamma subunits [J]
    • McGrew L, Chang MS, Sanders-Bush E Phospholipase D activation by endogenous 5-hydroxytryptamine 2C receptors is mediated by Galpha13 and pertussis toxin-insensitive Gbetagamma subunits [J]. Mol Pharmacol 2002, 62(6):1339-1343.
    • (2002) Mol Pharmacol , vol.62 , Issue.6 , pp. 1339-1343
    • McGrew, L.1    Chang, M.S.2    Sanders-Bush, E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.