Potent inhibition of Norwalk virus by cyclic sulfamide derivatives

Bioorganic and Medicinal Chemistry

Volumn 19, Issue 20, 2011, Pages 5975-5983

  Dou, Dengfeng ^a   Tiew, Kok Chuan ^a   He, Guijia ^a   Mandadapu, Sivakoteswara Rao ^a   Aravapalli, Sridhar ^a   Alliston, Kevin R ^a   Kim, Yunjeong ^b   Chang, Kyeong Ok ^b   Groutas, William C ^a  

^a WICHITA STATE UNIVERSITY   (United States)

^b KANSAS STATE UNIVERSITY   (United States)

Author keywords

Inhibitor; Norwalk virus

Indexed keywords

2 (3 CHLOROBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (3 METHOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (3 PHENOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 BUTOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 BUTYLBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 CHLOROBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 ETHOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 METHOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 PHENOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 PROPOXYBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 (4 PROPYLBENZYL) 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [(1 BENZYL 1H 1,2,3 TRIAZOL 4 YL)METHYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [3 (4 FLUOROPHENOXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [3 (BENZYLOXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [3 (HYDROXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [3 (TRIFLUOROMETHOXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [4 (2 METHYLPROPYL)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [4 (BENZYLOXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [4 (METHYLSULFANYL)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [4 (PROPAN 2 YLOXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [4 (TRIFLUOROMETHOXY)BENZYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; 2 [[1 (4 METHOXYBENZYL) 1H 1,2,3 TRIAZOL 4 YL]METHYL] 1,2,5 THIADIAZOLIDINE 1,1 DIOXIDE; ANTIVIRUS AGENT; CYCLOSULFAMIDE DERIVATIVE; SULFAMIDE DERIVATIVE; TERT BUTYL 1,2,5 THIADIAZOLIDINE 2 CARBOXYLATE 1,1 DIOXIDE; TERT BUTYL 5(PROP 2 YN 1 YL) 1,2,5 THIADIAZOLIDINE 2 CARBOXYLATE 1,1 DIOXIDE; TERT BUTYL 5[(1 BENZYL 1H 1,2,3 TRIAZOL 4 YL)METHYL] 1,2,5 THIADIAZOLIDINE 2 CARBOXYLATE 1,1 DIOXIDE; TERT BUTYL 5[[1 (4 METHOXYBENZYL) 1H 1,2,3 TRIAZOL 4 YL]METHYL] 1,2,5 THIADIAZOLI DINE 2 CARBOXYLATE 1,1 DIOXIDE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ANTIVIRAL ACTIVITY; ARTICLE; BIODIVERSITY; CONTROLLED STUDY; DRUG INHIBITION; DRUG STRUCTURE; NONHUMAN; NOROVIRUS;

AMIDES; CELL LINE, TUMOR; HUMANS; MOLECULAR STRUCTURE; NORWALK VIRUS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONIC ACIDS;

NOROVIRUS; NORWALK VIRUS;

EID: 80053223749     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2011.08.054     Document Type: Article

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