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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 19, 2011, Pages 5808-5811

Synthesis of β-functionalized Temoporfin derivatives for an application in photodynamic therapy

(4) Aicher, Daniel a,b Gräfe, Susanna c Stark, Christian B W a Wiehe, Arno c

a UNIVERSITY OF LEIPZIG (Germany)

b FREIE UNIVERSITÄT BERLIN (Germany)

c Biolitec AG (Germany)

Author keywords

Chlorins; Photocytotoxicity; Photodynamic therapy (PDT); Photosensitizer; Temoporfin

Indexed keywords

7,8 DIHYDROXY 5,10,15,20 TETRAKIS(3 HYDROXYPHENYL) 7,8 BIS(TRIFLUOROMETHYL) 7,8 CHLORIN; RADIOSENSITIZING AGENT; SINGLET OXYGEN; TEMOPORFIN; TEMOPORFIN DERIVATIVE; UNCLASSIFIED DRUG;

ADDITION REACTION; ARTICLE; CELL STRAIN HT29; CONTROLLED STUDY; DRUG EFFECT; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; PHOTODYNAMIC THERAPY; PHOTOTOXICITY; REACTION ANALYSIS; STRUCTURE ANALYSIS;

ANTINEOPLASTIC AGENTS; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; HT29 CELLS; HUMANS; HYDROXYLATION; MESOPORPHYRINS; MOLECULAR STRUCTURE; OSMIUM; PHOTOCHEMOTHERAPY; PHOTOSENSITIZING AGENTS; PORPHYRINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 80052602954 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.07.113 Document Type: Article

Times cited : (21)

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