Sulfonamides as selective oestrogen receptor β agonists

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 19, 2011, Pages 5680-5683

  Roberts, Lee R ^a   Armor, Duncan ^a   Barker, Carolyn ^a   Bent, Andrew ^a   Bess, Kirstin ^a   Brown, Alan ^a   Favor, David A ^a   Ellis, David ^a   Irving, Stephen L ^a   MacKenny, Malcolm ^a   Phillips, Chris ^a   Pullen, Nick ^a   Stennett, Adam ^a   Strand, Linda ^a   Styles, Michelle ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

Author keywords

ER agonist; Nuclear hormone receptor; Oestrogen receptor; Sulfonamides

Indexed keywords

ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; ESTROGEN RECEPTOR BETA AGONIST; HORMONE RECEPTOR STIMULATING AGENT; SULFONAMIDE; UNCLASSIFIED DRUG;

AGONIST; ARTICLE; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS; STRUCTURE ANALYSIS; X RAY ANALYSIS;

DRUG DISCOVERY; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; FEMALE; HUMANS; LIGANDS; MODELS, CHEMICAL; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 80052587585     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.08.041     Document Type: Article

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