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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 19, 2011, Pages 5961-5963

Preparation and antibacterial evaluation of decarboxylated fluoroquinolones

(6) Nguyen, Son T a Ding, Xiaoyuan a Butler, Michelle M a Tashjian, Tommy F a Peet, Norton P a Bowlin, Terry L a

a MICROBIOTIX INC (United States)

Author keywords

Antibacterial; Ciprofloxacin; Decarboxylated; Enrofloxacin; Fluoroquinolone; Norfloxacin

Indexed keywords

CARBOXYLIC ACID DERIVATIVE; CIPROFLOXACIN; ENROFLOXACIN; NORFLOXACIN; QUINOLINE DERIVED ANTIINFECTIVE AGENT;

AGAR DILUTION; ANTIBACTERIAL ACTIVITY; ARTICLE; BACILLUS SUBTILIS; BROTH DILUTION; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; ENTEROBACTER CLOACAE; ENTEROCOCCUS FAECALIS; ESCHERICHIA COLI; NONHUMAN; SERRATIA MARCESCENS; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; CARBOXYLIC ACIDS; DRUG DESIGN; FLUOROQUINOLONES; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; MICROBIAL SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP;

BACILLUS SUBTILIS; ENTEROBACTER CLOACAE; ENTEROCOCCUS FAECALIS; ESCHERICHIA COLI; SERRATIA MARCESCENS; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS;

EID: 80052586743 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.07.060 Document Type: Article

Times cited : (16)

References (16)

1
- 14844356060
- Birkhauser Verlag Basel
- A.R. Ronald, and D.E. Low Fluoroquinolone Antibiotics 2003 Birkhauser Verlag Basel
- (2003) Fluoroquinolone Antibiotics
- Ronald, A.R.¹ Low, D.E.²

2
- 0022633174
- J.M. Domagala, L.D. Hanna, C.L. Heifetz, M.P. Huff, T.F. Mich, P. Sanchez, and M. Solomon J. Med. Chem. 29 1986 394
- (1986) J. Med. Chem. , vol.29 , pp. 394
- Domagala, J.M.¹ Hanna, L.D.² Heifetz, C.L.³ Huff, M.P.⁴ Mich, T.F.⁵ Sanchez, P.⁶ Solomon, M.⁷

3
- 0023838559
- H. Kondo, F. Sakamoto, K. Kawakami, and G. Tsukamoto J. Med. Chem. 31 1998 221
- (1998) J. Med. Chem. , vol.31 , pp. 221
- Kondo, H.¹ Sakamoto, F.² Kawakami, K.³ Tsukamoto, G.⁴

4
- 0024555842
- D.T.W. Chu, and P.B. Fernandes Antimicrob. Agents Chemother. 33 1989 131
- (1989) Antimicrob. Agents Chemother. , vol.33 , pp. 131
- Chu, D.T.W.¹ Fernandes, P.B.²

5
- 34548120538
- C.H. Park, J. Lee, H.Y. Jung, M.J. Kim, S.H. Lim, H.T. Yeo, E.C. Choi, E.J. Yoon, K.W. Kim, J.H. Cha, S.-H. Kim, D.-J. Chang, D.-Y. Kwon, F. Li, and Y.-G. Suh Bioorg. Med. Chem. 15 2007 6517
- (2007) Bioorg. Med. Chem. , vol.15 , pp. 6517
- Park, C.H.¹ Lee, J.² Jung, H.Y.³ Kim, M.J.⁴ Lim, S.H.⁵ Yeo, H.T.⁶ Choi, E.C.⁷ Yoon, E.J.⁸ Kim, K.W.⁹ Cha, J.H.¹⁰ Kim, S.-H.¹¹ Chang, D.-J.¹² Kwon, D.-Y.¹³ Li, F.¹⁴ Suh, Y.-G.¹⁵

6
- 80052598216
- EP1245566 A1
- Al-Hajjar, F. H.; Jabal Al-Hussain, A. EP1245566 A1, 2002.
- (2002)
- Al-Hajjar, F.H.¹ Jabal Al-Hussain, A.²

7
- 80052566647
- Boston (MA) MEDI-325
- Marks, K. R.; Kerns, R. J. 240th ACS Meeting & Exposition, Boston (MA), 2010, MEDI-325.
- (2010) 240th ACS Meeting & Exposition
- Marks, K.R.¹ Kerns, R.J.²

8
- 0037534121
- R.J. Kerns, M.J. Rybak, G.W. Kaatz, F. Vaka, R. Cha, R.G. Grucz, and V.U. Diwadkar Bioorg. Med. Chem. Lett. 13 2003 2109
- (2003) Bioorg. Med. Chem. Lett. , vol.13 , pp. 2109
- Kerns, R.J.¹ Rybak, M.J.² Kaatz, G.W.³ Vaka, F.⁴ Cha, R.⁵ Grucz, R.G.⁶ Diwadkar, V.U.⁷

9
- 84860221495
- 4d reported MIC > 16 μg/mL.
- 4d Reported MIC > 16 μg/mL
- Against, S.¹

10
- 80052587918
- US 6320051 B1
- Berge, J. M.; Brown, P.; Elder, J. S.; Forrest, A. K.; Hamprecht, D. W.; Jarvest, R. L.; McNair, D. J.; Sheppard, R. J. US 6320051 B1, 2001.
- (2001)
- Berge, J.M.¹ Brown, P.² Elder, J.S.³ Forrest, A.K.⁴ Hamprecht, D.W.⁵ Jarvest, R.L.⁶ McNair, D.J.⁷ Sheppard, R.J.⁸

11
- 0019252702
- H. Koga, A. Itoh, S. Murayama, S. Suzue, and T. Irikura J. Med. Chem. 23 1980 1358
- (1980) J. Med. Chem. , vol.23 , pp. 1358
- Koga, H.¹ Itoh, A.² Murayama, S.³ Suzue, S.⁴ Irikura, T.⁵

12
- 0025906086
- For preparation and MIC values of 10 see: J.M. Domagala, A.J. Bridges, T.P. Culbertson, L. Gambino, S.E. Hagen, G. Karrick, K. Porter, J.P. Sanchez, J.A. Sesnie, G. Spense, D. Szotek, and J. Wemple J. Med. Chem. 34 1991 1142
- (1991) J. Med. Chem. , vol.34 , pp. 1142
- Domagala, J.M.¹ Bridges, A.J.² Culbertson, T.P.³ Gambino, L.⁴ Hagen, S.E.⁵ Karrick, G.⁶ Porter, K.⁷ Sanchez, J.P.⁸ Sesnie, J.A.⁹ Spense, G.¹⁰ Szotek, D.¹¹ Wemple, J.¹²

13
- 0027423686
- T. Uno, T. Okuno, K. Kawakami, F. Sakamoto, and G. Tsukamoto J. Med. Chem. 36 1993 2711
- (1993) J. Med. Chem. , vol.36 , pp. 2711
- Uno, T.¹ Okuno, T.² Kawakami, K.³ Sakamoto, F.⁴ Tsukamoto, G.⁵

14
- 14844283708
- B. Liu, C.-H. Yang, G.-Y. Xu, Y.-H. Zhu, J.-R. Cui, X.-H. Wu, and Y.-Y. Xie Bioorg. Med. Chem. 13 2005 2451
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 2451
- Liu, B.¹ Yang, C.-H.² Xu, G.-Y.³ Zhu, Y.-H.⁴ Cui, J.-R.⁵ Wu, X.-H.⁶ Xie, Y.-Y.⁷

15
- 0028113629
- M. Reuman, M.A. Eissenstat, and J.D. Weaver III Tetrahedron Lett. 35 1994 8303
- (1994) Tetrahedron Lett. , vol.35 , pp. 8303
- Reuman, M.¹ Eissenstat, M.A.² Weaver Iii, J.D.³

16
- 0022450259
- For a different method to prepare 4 see: W. Gau, J. Kurz, U. Petersen, H.J. Ploschke, and C. Wuensche Arzneimittel Forschung 36 1986 1545
- (1986) Arzneimittel Forschung , vol.36 , pp. 1545
- Gau, W.¹ Kurz, J.² Petersen, U.³ Ploschke, H.J.⁴ Wuensche, C.⁵

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