Compatibility study between ibuprofen and excipients in their physical mixtures

Journal of Thermal Analysis and Calorimetry

Volumn 105, Issue 2, 2011, Pages 517-527

  Tiţa, Bogdan ^a   Fuliaş, Adriana ^a   Szabadai, Zoltan ^a   Rusu, Gerlinde ^b   Bandur, Geza ^b   Tiţa, Dumitru ^a  

^a VICTOR BABES UNIVERSITY OF MEDICINE AND PHARMACY   (Romania)

^b POLITEHNICA UNIVERSITY OF TIMISOARA   (Romania)

Author keywords

Drug excipient compatibility; Ibuprofen; TG DSC; Thermal behaviour

Indexed keywords

ANALYTES; DRUG-EXCIPIENT COMPATIBILITY; DRUG-EXCIPIENT INTERACTIONS; ENDOTHERMIC PEAKS; FTIR SPECTROSCOPY; GENERAL METHOD; IBUPROFEN; LONG TERM STABILITY; MAGNESIUM STEARATE; MASS LOSS; MICROCRYSTALLINE CELLULOSE; PHARMACEUTICAL PRODUCTS; PHYSICAL MIXTURES; POLY VINYL PYRROLIDONE; SINGLE STAGE; SYSTEMATIC STUDY; TG/DSC; THERMAL BEHAVIOURS; THERMAL TECHNIQUES;

DIFFERENTIAL SCANNING CALORIMETRY; DRUG INTERACTIONS; DRUG PRODUCTS; MAGNESIUM; SILICA; SUGARS; THERMODYNAMIC PROPERTIES; THERMOGRAVIMETRIC ANALYSIS; X RAY POWDER DIFFRACTION;

BINARY MIXTURES;

EID: 79960065595     PISSN: 13886150     EISSN: None     Source Type: Journal    
DOI: 10.1007/s10973-010-1188-8     Document Type: Conference Paper

References (41)

1. D Kovala-Demertzi 2006 Recent advances on non-steroidal anti-inflammatory drugs, NSAIDs: Organotin complexes of NSAIDs J Organomet Chem. 691 1767 1774 10.1016/j.jorganchem.2005.11.058 1:CAS:528:DC%2BD28XislCns70%3D
2. K Kafarska D Czakis-Sulikowska WM Wolf 2009 Novel Co(II) and Cd(II) complexes with non-steroidal anti-inflammatory drugs. Synthesis, properties and thermal investigation J Therm Anal Calorim. 96 617 621 10.1007/s10973-008-9456-6 1:CAS:528:DC%2BD1MXmsVOrt78%3D
3. OI Teslyuk SV Beltyukova AV Yegorova BN Yagodkin 2007 Complex compounds of terbium(III) with some nonsteroidal anti-inflammatory drugs and their analytical applications J Anal Chem. 62 330 335 10.1134/S1061934807040065 1:CAS:528:DC%2BD2sXktVehur4%3D (Pubitemid 46572094)
4. YC Ying L Yi ZJ Cheng Z Dan 2008 Inhibitory effect of copper complex of indomethacin on bacteria studied by microcalorimetry Biol Trace Elem Res 122 82 88 10.1007/s12011-007-8063-x
5. A Fini G Fasio L Benetti V Ghedini 2007 Thermal analysis of some diclofenac salts with alkyl and alkylhydroxy amines Thermochim Acta. 464 65 74 10.1016/j.tca.2007.08.006 1:CAS:528:DC%2BD2sXhtFKiu7zP (Pubitemid 47532174)
6. P Mora Corvi M Cirri P Mura 2006 Differential scanning calorimetry as a screening technique in compatibility studies of DHEA extended release formulations J Pharm Biomed Anal. 42 3 10 10.1016/j.jpba.2006.02.038 1:STN:280:DC%2BD28rht1Sltw%3D%3D (Pubitemid 44403899)
7. Neto HS, Barros FAP, de Sousa Carvalho FM, Matos JR, Thermal analysis of prednicarbate and characterization of thermal decomposition product, J Therm Anal Calorim. 2010. doi: 10.1007/s10973-009-0419-3.
8. RO Macêdo CFS Aragão TG do Nascimento AMC Macêdo 1999 Application of thermogravimetry in the quality control of chloramphenicol tablets J Therm Anal Calorim. 56 1323 1327 10.1023/A:1010102422381
9. Moura EA, Correia LP, Pinto MF, Procopio JVV, de Sousa FS, Macedo RO. Thermal characterization of the solid state and raw material fluconazole by thermal analysis and pyrolysis coupled to GC/MS. J Therm Anal Calorim. 2010. doi: 10.1007/s10973-009-0473-X.
10. F Giordano A Rossi I Pasquali R Bettini E Frigo A Gazzaniga ME Sangalli V Miles S Catinella 2003 Thermal degradation and melting point determination of diclofenac J Therm Anal Calorim. 73 509 518 10.1023/A:1025421911670 1:CAS:528:DC%2BD3sXnslGisbw%3D
11. R Picciochi HP Diogo MEM da Piedade 2010 Thermochemistry of paracetamol J Therm Anal Calorim. 99 391 401 10.1007/s10973-009-0634-y
12. B Tiţa E Marian D Tiţa G Vlase N Doca T Vlase 2008 Comparative kinetic study of decomposition of some diazepine derivatives under isothermal and non-isothermal conditions J Therm Anal Calorim. 94 447 452 10.1007/s10973-008-9146-4
13. B Tiţa A Fuliaş E Marian D Tiţa 2009 Thermal behaviour of acetylsalicylic acid-active substance and tablets. Kinetic study under non-isothermal conditions Rev Chim (Bucureşti) 60 419 423
14. B Tiţa A Fuliaş E Marian D Tiţa 2009 Thermal stability and decomposition kinetics under non-isothermal conditions of sodium diclofenac Rev Chim (Bucureşti) 60 524 528
15. A Fuliaş B Tiţa G Bandur D Tiţa 2009 Thermal decomposition of some benzodiazepines under non-isothermal conditions. Kinetic study Rev Chim (Bucureşti) 60 1079 1083
16. B Tiţa A Fuliaş G Rusu D Tiţa 2009 Thermal behaviour of indomethacin-active substance and tablets kinetic study under non-isothermal conditions Rev Chim (Bucureşti) 60 1210 1215
17. LS Bernardi PR Oliveira FS Murakami MAS Silva SHM Borgmann SG Cardoso 2009 Characterization of venlafoxine with pharmaceutical excipients J Therm Anal Calorim. 97 729 733 10.1007/s10973-009-0282-2 1:CAS:528:DC%2BD1MXhtlWns73M
18. Moyano MA, Broussalis AM, Segall AI. Thermal analysis of lipoic acid and evaluation of the compatibility with excipients. J Therm Anal Calorim. 2010. doi: 10.1007/s10973-009-0351-6.
19. PR Oliveira LS Bernardi FS Murakami C Mendes MAS Silva 2009 Thermal characterization and compatibility studies of norfloxacin for development of extended release tablets J Therm Anal Calorim. 97 741 745 10.1007/s10973-009- 0347-2 1:CAS:528:DC%2BD1MXhtlWns7%2FE
20. AM Lira AAS Araújo IDJ Basílio BLL Santos DP Santana RO Macedo 2007 Compatibility studies of lapachol with pharmaceutical excipients for the development of topical formulations Thermochim Acta. 457 1 6 10.1016/j.tca.2007.02.017 1:CAS:528:DC%2BD2sXkvFGgtL0%3D (Pubitemid 46661953)
21. M Tomassetti A Catalani V Rossi S Vecchio 2005 Thermal analysis study of the interactions between acetaminophen and excipients in solid dosage forms and in some binary mixtures J Pharm Biomed Anal. 37 949 955 10.1016/j.jpba.2004.10. 008 1:CAS:528:DC%2BD2MXjs1Klsrk%3D (Pubitemid 40614824)
22. F Barboza DD Vecchia MP Tagliari MAS Silva HK Stulzer 2009 Differential scanning calorimetry as a screening technique in compatibility studies of acyclovir extended release formulations Pharm Chem J. 43 363 368 10.1007/s11094-009-0304-1 1:CAS:528:DC%2BD1MXhtlShsrzL
23. Bannach G, Cervini P, Cavalheiro ETG, Ionashiro M. Using thermal and spectroscopic data to investigate the thermal behaviour of drugs and excipients by unique calculations. J Therm Anal Calorim. 2010. doi: 10.007/s10973-009-0595- 1.
24. T Iliescu M Baia V Miclǎuş 2004 A Raman spectroscopic study of the diclofenac sodium-β-cyclodextrin interaction Eur J Pharm Sci. 22 487 495 10.1016/j.ejps.2004.05.003 1:CAS:528:DC%2BD2cXlsl2nt74%3D (Pubitemid 38953908)
25. G Bannach P Cervini ETG Cavalheiro M Ionashiro 2010 Using thermal and spectroscopic data to investigate the thermal behaviour of drugs and excipients by unique calculations Thermochim Acta. 499 123 127 10.1016/j.tca.2009.11.012 1:CAS:528:DC%2BC3cXht1yjsbs%3D
26. B Tiţa A Fuliaş G Bandur G Rusu D Tiţa 2010 Thermal stability of ibuprofen. Kinetic study under non-isothermal conditions Rev Roum Chim. 55 553 558
27. CD Bertol AP Cruz HK Stulzer FS Murakami MAS Silva 2010 Thermal decomposition kinetics and compatibility studies of primaquine under isothermal and non-isothermal conditions J Therm Anal Calorim. 102 187 192 10.1007/s10973-009-0540-3 1:CAS:528:DC%2BC3cXhtFartL7J
28. A Marini V Berbenni S Moioli G Bruni P Cofrancesco C Margheritis 2003 Drug-excipient compatibility studies by physico-chemical techniques. The case of indomethacin J Therm Anal Calorim. 73 529 545 10.1023/A:1025426012578 1:CAS:528:DC%2BD3sXnslGisbo%3D
29. A Gombas P Szabo-Revesz M Kata G Regdon Jr I Eros 2002 Quantitative determination of crystallinity of α-lactose monohydrate by DSC J Therm Anal Calorim. 68 503 510 10.1023/A:1016039819247 1:CAS:528:DC%2BD38XkvFegsrc%3D (Pubitemid 34614450)
30. F Balestrieri AD Magri AL Magri D Marini A Sacchini 1996 Application of differential scanning calorimetry to the study of drug-excipient compatibility Thermochim Acta. 285 337 345 10.1016/0040-6031(96)02904-8 1:CAS:528: DyaK28XmtVyrurk%3D (Pubitemid 126316647)
31. SR Desai MM Shaikh SR Dharwadkar 2003 Preformulation compatibility studies of etamsylate and fluconazole drugs with lactose by DSC J Therm Anal Calorim. 71 651 658 10.1023/A:1022832732679 1:CAS:528:DC%2BD3sXitVynsb8%3D
32. LCS Cides AAS Araújo M Santos-Filho JR Matos 2006 Thermal behaviour, compatibility study and decomposition kinetics of glimepiride under isothermal and non-isothermal conditions J Therm Anal Calorim. 84 441 445 10.1007/s10973-005-7131-8 1:CAS:528:DC%2BD28XksFektL8%3D (Pubitemid 43724304)
33. GGG Oliveira HG Ferraz JSR Matos 2005 Thermoanalytical study of glibenclamide and excipients J Therm Anal Calorim. 79 267 270 10.1007/s10973-005-0047-5 1:CAS:528:DC%2BD2MXkt1Ciu70%3D (Pubitemid 40626210)
34. A Marini V Berbenni M Pegoretti G Bruni P Cofrancesco C Sinistri M Villa 2003 Drug-excipient compatibility studies by physico-chemical techniques. The case of atenolol J Therm Anal Calorim. 73 547 561 10.1023/A:1025478129417 1:CAS:528:DC%2BD3sXnslGisbs%3D
35. G Bruni L Amici V Berbenni A Marini A Orlandi 2002 Drug-excipient compatibility studies J Therm Anal Calorim. 68 561 573 10.1023/A:1016052121973 1:CAS:528:DC%2BD38XkvFegsL8%3D (Pubitemid 34614455)
36. RS Nunes FS Semaan AT Riga ÉTG Cavalheiro 2009 Thermal behavior of verapamil hydrochloride and its association with excipients J Therm Anal Calorim. 97 349 353 10.1007/s10973-009-0072-x 1:CAS:528:DC%2BD1MXht1OgurvK
37. HK Stulzer MP Tagliari AP Cruz MAS Silva MCM Laranjeira 2008 Compatibility studies between piroxicam and pharmaceutical excipients used in solid dosage forms Pharm Chem J. 42 215 219 10.1007/s11094-008-0091-0 1:CAS:528:DC%2BD1cXht1aisb3J
38. HK Stulzer PO Rodrigues TM Cardoso JSR Matos MAS Silva 2008 Compatibility studies between captopril and pharmaceutical excipients used in tablets formulations J Therm Anal Calorim. 91 323 328 10.1007/s10973-006-7935-1 1:CAS:528:DC%2BD1cXhsFansrc%3D (Pubitemid 351199257)
39. HS Neto Cs Novák JR Matos 2009 Thermal analysis and compatibility studies of prednicarbate with excipients used in semi solid pharmaceutical form J Therm Anal Calorim. 97 367 374 10.1007/s10973-009-0234-x
40. FD Freire CFS Aragao TFA e Moura FN Raffin 2009 Compatibility study between chlorpropamide and excipients in their physical mixtures J Therm Anal Calorim. 97 355 357 10.1007/s10973-009-0258-2 1:CAS:528:DC%2BD1MXht1OgurzI
41. D Abbas J Kaloustian C Orneto P Piccerelle H Portugal A Nicolay 2008 DSC and physico-chemical properties of a substituted pyridoquinoline and its interaction study with excipients J Therm Anal Calorim. 93 353 360 10.1007/s10973-008-9062-7 1:CAS:528:DC%2BD1cXosl2mtb4%3D