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Volumn 6, Issue 7, 2011, Pages 1249-1257

Structural Investigation of the Naphthyridone Scaffold: Identification of a 1,6-Naphthyridone Derivative with Potent and Selective Anti-HIV Activity

(8) Tabarrini, Oriana a Massari, Serena a Sancineto, Luca a Daelemans, Dirk b Sabatini, Stefano a Manfroni, Giuseppe a Cecchetti, Violetta a Pannecouque, Christophe b

a UNIVERSITY OF PERUGIA (Italy)

b REGA INSTITUTE FOR MEDICAL RESEARCH (Belgium)

Author keywords

1,6 naphthyridones; Anti HIV quinolones; Antiviral agents; Medicinal chemistry; Transcription inhibitors

Indexed keywords

1,5 NAPHTHYRIDONE; 1,6 NAPHTHYRIDONE; 1,7 NAPHTHYRIDONE; 1,8 NAPHTHYRIDINE DERIVATIVE; AMINO ACID DERIVATIVE; NAPHTHYRIDINE DERIVATIVE; UNCLASSIFIED DRUG; VINYL DERIVATIVE;

ARTICLE; CATALYSIS; CYTOTOXICITY; DRUG ACTIVITY; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS; PRIORITY JOURNAL;

ANTI-HIV AGENTS; CELL LINE; HIV-1; HIV-2; HUMANS; NAPHTHYRIDINES; QUINOLONES; STRUCTURE-ACTIVITY RELATIONSHIP; VIRUS REPLICATION;

EID: 79959707629 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100073 Document Type: Article

Times cited : (31)

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