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Volumn 19, Issue 11, 2011, Pages 3384-3393

CXCR3 antagonists: Quaternary ammonium salts equipped with biphenyl- and polycycloaliphatic-anchors

(8) Wijtmans, Maikel a Verzijl, Dennis a Bergmans, Serge a Lai, Michael a Bosch, Leontien a Smit, Martine J a De Esch, Iwan J P a Leurs, Rob a

a VU UNIVERSITY AMSTERDAM (Netherlands)

Author keywords

Ammonium salt; Antagonist; CXCR3; Myrtenyl; Suzuki coupling

Indexed keywords

1 (4 IODOPHENYL) 3 (2 ADAMANTYL)GUANIDINE; ALIPHATIC COMPOUND; AMANTADINE; AMG 487; BIPHENYL; CHEMOKINE RECEPTOR ANTAGONIST; CHEMOKINE RECEPTOR CXCR3 ANTAGONIST; GUANIDINE; QUATERNARY AMMONIUM DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG ACTIVITY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; LIPOPHILICITY; METHYLATION; PROTON TRANSPORT; STRUCTURE ACTIVITY RELATION; SUZUKI REACTION;

BIPHENYL COMPOUNDS; CELL LINE; GUANIDINE; HUMANS; POLYCYCLIC COMPOUNDS; PROTEIN BINDING; QUATERNARY AMMONIUM COMPOUNDS; RECEPTORS, CXCR3; SALTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 79957493207 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2011.04.035 Document Type: Article

Times cited : (19)

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