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Bioorganic and Medicinal Chemistry

Volumn 19, Issue 10, 2011, Pages 3274-3279

Design, synthesis and inhibition activity of a novel cyclic enediyne amino acid conjugates against MPtpA

(5) Chandra, Koushik a Dutta, Debajyoti a Mitra, Analava a Das, Amit K a Basak, Amit a

a INDIAN INSTITUTE OF TECHNOLOGY (India)

Author keywords

Amino acid; Conjugate; Enediyne; Inhibition; Knoevenagel; MPtpA

Indexed keywords

CYCLIC ENEDIYNE AMINO ACID CONJUGATE DERIVATIVE; CYCLIC ENEDIYNE MALONAMIC ACID CONJUGATE DERIVATIVE; ENEDIYNE; PROTEIN MPTPA; PROTEIN TYROSINE PHOSPHATASE; UNCLASSIFIED DRUG;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG CONJUGATION; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TARGETING; IC 50; KNOEVENAGEL CONDENSATION; MICHAEL ADDITION; MOLECULAR DOCKING; PHARMACOLOGICAL BLOCKING; SOLVENT EFFECT; TEMPERATURE SENSITIVITY;

AMINO ACIDS, CYCLIC; BACTERIAL PROTEINS; CYCLIZATION; DRUG DESIGN; ENEDIYNES; ENZYME INHIBITORS; HUMANS; MALONATES; MODELS, MOLECULAR; MYCOBACTERIUM TUBERCULOSIS; PROTEIN BINDING; PROTEIN TYROSINE PHOSPHATASES; TUBERCULOSIS;

EID: 79956201657 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2011.03.024 Document Type: Article

Times cited : (6)

References (39)

1
- 84883839798
- N. Ishida, K. Miyazaki, K. Kumagai, and M. Rikimaru J. Antibiot. 18 1965 68
- (1965) J. Antibiot. , vol.18 , pp. 68
- Ishida, N.¹ Miyazaki, K.² Kumagai, K.³ Rikimaru, M.⁴

2
- 0003451102
- Springer Tokyo
- H. Maeda, K. Edo, and N. Ishida Neocarzinostatin: The Past, Present and Future of An Anticancer Drug 1997 Springer Tokyo
- (1997) Neocarzinostatin: The Past, Present and Future of An Anticancer Drug
- Maeda, H.¹ Edo, K.² Ishida, N.³

3
- 0030005845
- J.W. Grissom, G.U. Gunawardena, D. Klingberg, and D. Huang Tetrahedron 52 1996 6453
- (1996) Tetrahedron , vol.52 , pp. 6453
- Grissom, J.W.¹ Gunawardena, G.U.² Klingberg, D.³ Huang, D.⁴

4
- 0001055380
- K.C. Nicolaou, and A.L. Smith Acc. Chem. Res. 25 1992 497
- (1992) Acc. Chem. Res. , vol.25 , pp. 497
- Nicolaou, K.C.¹ Smith, A.L.²

5
- 0023228110
- M.D. Lee, T.S. Dunne, M.M. Siegel, C.C. Chang, G.O. Morton, and D.B. Borders J. Am. Chem. Soc. 109 1987 3464
- (1987) J. Am. Chem. Soc. , vol.109 , pp. 3464
- Lee, M.D.¹ Dunne, T.S.² Siegel, M.M.³ Chang, C.C.⁴ Morton, G.O.⁵ Borders, D.B.⁶

6
- 0026045597
- K.C. Nicolaou, and W.M. Dai Angew. Chem., Int. Ed. Engl. 30 1991 1387
- (1991) Angew. Chem., Int. Ed. Engl. , vol.30 , pp. 1387
- Nicolaou, K.C.¹ Dai, W.M.²

7
- 0035878068
- F.J. Giles, H.M. Kantarjian, S.M. Kornblau, D.A. Thomas, G. Garcia-Manero, T.A. Waddelow, C.L. David, A.T. Phan, D.E. Colburn, A. Rashid, and E.H. Estey Cancer 92 2001 406
- (2001) Cancer , vol.92 , pp. 406
- Giles, F.J.¹ Kantarjian, H.M.² Kornblau, S.M.³ Thomas, D.A.⁴ Garcia-Manero, G.⁵ Waddelow, T.A.⁶ David, C.L.⁷ Phan, A.T.⁸ Colburn, D.E.⁹ Rashid, A.¹⁰ Estey, E.H.¹¹

8
- 0034900174
- P.F. Bross, J. Beitz, G. Chen, X.H. Chen, E. Duffy, L. Kieffer, S. Roy, R. Sridhara, A. Rahman, G. Williams, and R. Pazdur Clin. Cancer Res. 7 2001 1490
- (2001) Clin. Cancer Res. , vol.7 , pp. 1490
- Bross, P.F.¹ Beitz, J.² Chen, G.³ Chen, X.H.⁴ Duffy, E.⁵ Kieffer, L.⁶ Roy, S.⁷ Sridhara, R.⁸ Rahman, A.⁹ Williams, G.¹⁰ Pazdur, R.¹¹

9
- 0042442407
- M. Wadleigh, P.G. Richardson, D. Zahrieh, S.J. Lee, C. Cutler, V. Ho, E.P. Alyea, J.H. Antin, R.M. Stone, R.J. Soiffer, and D.J. DeAngelo Blood 102 2003 1578
- (2003) Blood , vol.102 , pp. 1578
- Wadleigh, M.¹ Richardson, P.G.² Zahrieh, D.³ Lee, S.J.⁴ Cutler, C.⁵ Ho, V.⁶ Alyea, E.P.⁷ Antin, J.H.⁸ Stone, R.M.⁹ Soiffer, R.J.¹⁰ Deangelo, D.J.¹¹

10
- 40949133462
- R.P. Jones, and R.G. Bergman J. Am. Chem. Soc. 94 1972 960
- (1972) J. Am. Chem. Soc. , vol.94 , pp. 960
- Jones, R.P.¹ Bergman, R.G.²

11
- 0002933542
- R.G. Bergman Acc. Chem. Res. 6 1973 25
- (1973) Acc. Chem. Res. , vol.6 , pp. 25
- Bergman, R.G.¹

12
- 33845557780
- T.P. Lockhart, P.B. Comita, and R.G. Bergman J. Am. Chem. Soc. 103 1981 4082
- (1981) J. Am. Chem. Soc. , vol.103 , pp. 4082
- Lockhart, T.P.¹ Comita, P.B.² Bergman, R.G.³

13
- 33845557570
- T.P. Lockhart, P.B. Comita, and R.G. Bergman J. Am. Chem. Soc. 103 1981 4091
- (1981) J. Am. Chem. Soc. , vol.103 , pp. 4091
- Lockhart, T.P.¹ Comita, P.B.² Bergman, R.G.³

14
- 0019167917
- L.S. Kappen, and I.H. Goldberg Biochemistry 19 1980 4786
- (1980) Biochemistry , vol.19 , pp. 4786
- Kappen, L.S.¹ Goldberg, I.H.²

15
- 0021960376
- K. Edo, M. Mizugaki, Y. Koide, H. Seto, K. Furihata, N. Otake, and N. Ishida Tetrahedron Lett. 26 1985 331
- (1985) Tetrahedron Lett. , vol.26 , pp. 331
- Edo, K.¹ Mizugaki, M.² Koide, Y.³ Seto, H.⁴ Furihata, K.⁵ Otake, N.⁶ Ishida, N.⁷

16
- 0028793511
- M.P. Hay, W.R. Wilson, and W.A. Denny Bioorg. Med. Chem. Lett. 5 1995 2829
- (1995) Bioorg. Med. Chem. Lett. , vol.5 , pp. 2829
- Hay, M.P.¹ Wilson, W.R.² Denny, W.A.³

17
- 34250851878
- J.R. Baker, D.N. Woolfson, F.W. Muskett, R.G. Stoneman, M.D. Urbaniak, and S. Caddick ChemBioChem 8 2007 704
- (2007) ChemBioChem , vol.8 , pp. 704
- Baker, J.R.¹ Woolfson, D.N.² Muskett, F.W.³ Stoneman, R.G.⁴ Urbaniak, M.D.⁵ Caddick, S.⁶

18
- 0034704611
- G.B. Jones, G.W. Plourde II, and J.M. Wright Org. Lett. 2 2000 811
- (2000) Org. Lett. , vol.2 , pp. 811
- Jones, G.B.¹ Plourde, G.W.I.I.² Wright, J.M.³

19
- 0025100205
- M. Konishi, H. Ohkuma, T. Tsuno, T. Oki, G.D. Vanduyne, and J. Clardy J. Am. Chem. Soc. 112 1990 3715
- (1990) J. Am. Chem. Soc. , vol.112 , pp. 3715
- Konishi, M.¹ Ohkuma, H.² Tsuno, T.³ Oki, T.⁴ Vanduyne, G.D.⁵ Clardy, J.⁶

20
- 0026512210
- M.D. Lee, T.S. Dunne, C.C. Chang, M.M. Siegel, G.O. Morton, G.A. Ellestad, W.J. McGahren, and D.B. Borders J. Am. Chem. Soc. 114 1992 985
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 985
- Lee, M.D.¹ Dunne, T.S.² Chang, C.C.³ Siegel, M.M.⁴ Morton, G.O.⁵ Ellestad, G.A.⁶ McGahren, W.J.⁷ Borders, D.B.⁸

21
- 0031465920
- S. Kawata, S. Ashizawa, and M. Hirama J. Am. Chem. Soc. 119 1997 12012
- (1997) J. Am. Chem. Soc. , vol.119 , pp. 12012
- Kawata, S.¹ Ashizawa, S.² Hirama, M.³

22
- 14644438366
- C. Madhurantakam, E. Rajakumara, P.A. Mazumdar, B. Saha, D. Mitra, H.G. Wiker, R. Sankaranarayanan, and A.K. Das J. Bactoriol. 187 2005 2175
- (2005) J. Bactoriol. , vol.187 , pp. 2175
- Madhurantakam, C.¹ Rajakumara, E.² Mazumdar, P.A.³ Saha, B.⁴ Mitra, D.⁵ Wiker, H.G.⁶ Sankaranarayanan, R.⁷ Das, A.K.⁸

23
- 0032508046
- S.T. Cole, R. Brosch, J. Parkhill, T. Garnier, C. Churcher, D. Harris, S.V. Gordon, K. Eiglmeier, S. Gas, C.E. Barry, F. Tekaia, K. Badcock, D. Basham, D. Brown, T. Chillingworth, R. Connor, R. Davies, K. Devlin, T. Feltwell, S. Gentles, N. Hamlin, S. Holroyd, T. Hornsby, K. Jagels, A. Krogh, J. McLean, S. Moule, I. Murphy, K. Oliver, J. Osborne, M.A. Quail, M.A. Rajandream, J. Roger, S. Rutter, K. Seeger, J. Skelton, R. Squares, S. Squares, J.E. Sulston, K. Taylor, S. Whitehead, and B.G. Barell Nature 393 1998 537
- (1998) Nature , vol.393 , pp. 537
- Cole, S.T.¹ Brosch, R.² Parkhill, J.³ Garnier, T.⁴ Churcher, C.⁵ Harris, D.⁶ Gordon, S.V.⁷ Eiglmeier, K.⁸ Gas, S.⁹ Barry, C.E.¹⁰ Tekaia, F.¹¹ Badcock, K.¹² Basham, D.¹³ Brown, D.¹⁴ Chillingworth, T.¹⁵ Connor, R.¹⁶ Davies, R.¹⁷ Devlin, K.¹⁸ Feltwell, T.¹⁹ Gentles, S.²⁰ more..

24
- 34547842536
- N. Beresford, S. Patel, J. Armstrong, B. Szöor, A.P. Fordham-Skelton, and L. Tabernero Biochem. J. 406 2007 13
- (2007) Biochem. J. , vol.406 , pp. 13
- Beresford, N.¹ Patel, S.² Armstrong, J.³ Szöor, B.⁴ Fordham-Skelton, A.P.⁵ Tabernero, L.⁶

25
- 0036218194
- S.C. Cowley, R. Babakaiff, and Y. Av-Gay Res. Microbiol. 153 2002 233
- (2002) Res. Microbiol. , vol.153 , pp. 233
- Cowley, S.C.¹ Babakaiff, R.² Av-Gay, Y.³

26
- 78249286529
- K. Chandra, D. Dutta, A.K. Das, and A. Basak Bioorg. Med. Chem. 18 2010 8365
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 8365
- Chandra, K.¹ Dutta, D.² Das, A.K.³ Basak, A.⁴

27
- 9644285669
- K. Sonogashira, Y. Tohoda, and N. Hagihara Tetrahedron Lett. 16 1975 4467
- (1975) Tetrahedron Lett. , vol.16 , pp. 4467
- Sonogashira, K.¹ Tohoda, Y.² Hagihara, N.³

28
- 84989498349
- S. Takahashi, Y. Kuroyama, K. Sonogashira, and N. Hagihara Synthesis 1980 627
- (1980) Synthesis , pp. 627
- Takahashi, S.¹ Kuroyama, Y.² Sonogashira, K.³ Hagihara, N.⁴

29
- 0001248159
- L.F. Fieser, and M. Fieser Reagents Org. Synth. l1 1967 256
- (1967) Reagents Org. Synth. , vol.1 , pp. 256
- Fieser, L.F.¹ Fieser, M.²

30
- 79956208541
- S. Karger AG Basel
- W. Theilheimer Synthetic Methods of Organic Chemistry Vol. 20 1966 S. Karger AG Basel 52
- (1966) Synthetic Methods of Organic Chemistry , vol.20 , pp. 52
- Theilheimer, W.¹

31
- 3042741556
- D.B. Dess, and J.C. Martin J. Am. Chem. Soc. 113 1991 7277
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 7277
- Dess, D.B.¹ Martin, J.C.²

32
- 0001285003
- P.R. Schreiner Chem. Commun. 1998 483
- (1998) Chem. Commun. , pp. 483
- Schreiner, P.R.¹

33
- 79956207541
- K.C. Nicolaou Chem. Br. Jan. 1994 33
- (1994) Chem. Br. Jan. , pp. 33
- Nicolaou, K.C.¹

34
- 0037169037
- H. Wandel, and O. Wiest J. Org. Chem. 67 2002 388
- (2002) J. Org. Chem. , vol.67 , pp. 388
- Wandel, H.¹ Wiest, O.²

35
- 1542401458
- Huthig & Wepf Verlag Basel
- H.-G. Elias Macromolekule Vol. 1 1990 Huthig & Wepf Verlag Basel p 817
- (1990) Macromolekule , vol.1
- Elias, H.-G.¹

36
- 84985645263
- R.H. Grubbs, and D. Kratz Chem. Ber. 126 1993 149
- (1993) Chem. Ber. , vol.126 , pp. 149
- Grubbs, R.H.¹ Kratz, D.²

37
- 78249266638
- C. Madhurantakam, V.R.M. Chavali, and A.K. Das Proteins 2007 706
- (2007) Proteins , pp. 706
- Madhurantakam, C.¹ Chavali, V.R.M.² Das, A.K.³

38
- 11644261806
- G.M. Morris, D.S. Goodsell, R.S. Halliday, R. Huey, W.E. Hart, R.K. Belew, and A.J. Olson J. Comput. Chem. 19 1998 1639
- (1998) J. Comput. Chem. , vol.19 , pp. 1639
- Morris, G.M.¹ Goodsell, D.S.² Halliday, R.S.³ Huey, R.⁴ Hart, W.E.⁵ Belew, R.K.⁶ Olson, A.J.⁷

39
- 79956202084
- http://www.ebi.ac.uk/msd-srv/prot-int/pistart.html.

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