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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 10, 2011, Pages 2890-2893

SAR studies of pyridazinone derivatives as novel glucan synthase inhibitors

(18) Zhou, Gang a Ting, Pauline C a Aslanian, Robert a Cao, Jianhua a Kim, David W a Kuang, Rongze a Lee, Joe F a Schwerdt, John a Wu, Heping a Jason Herr, R b Zych, Andrew J b Yang, Jinhai b Lam, Sang b Wainhaus, Samuel a Black, Todd A a McNicholas, Paul M a Xu, Yiming a Walker, Scott S a

a MERCK RESEARCH LABORATORIES (United States)

b Albany Molecular Research (United States)

Author keywords

1,3 Glucan synthase inhibitors; Antifungal; Pyridazinone

Indexed keywords

5 [4 (BENZYLSULFONYL)PIPERAZIN 1 YL] 4 MORPHOLINO 2 PHENYLPYRIDAZIN 3(2H) ONE; ANIDULAFUNGIN; CASPOFUNGIN; GLUCAN SYNTHASE; PYRIDAZINONE DERIVATIVE; SULFONAMIDE; UNCLASSIFIED DRUG;

ANTIFUNGAL ACTIVITY; AREA UNDER THE CURVE; ARTICLE; CANDIDA ALBICANS; CANDIDA GLABRATA; DRUG STRUCTURE; FUNGAL STRAIN; NONHUMAN; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ANTIFUNGAL AGENTS; CANDIDA ALBICANS; CANDIDA GLABRATA; ENZYME INHIBITORS; GLUCOSYLTRANSFERASES; MOLECULAR STRUCTURE; PYRIDAZINES; STRUCTURE-ACTIVITY RELATIONSHIP;

CANDIDA ALBICANS; CANDIDA GLABRATA;

EID: 79955554707 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2011.03.083 Document Type: Article

Times cited : (28)

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