Formulation and characterization of gastroretentive discs containing famotidine

Brazilian Archives of Biology and Technology

Volumn 54, Issue 2, 2011, Pages 293-300

  Raval, Jignyasha Amitkumar ^a   Patel, Madhabhai M ^b  

^a GANPAT UNIVERSITY   (India)

^b GUJARAT TECHNOLOGICAL UNIVERSITY   (India)

Author keywords

Discs; Gastroretentive; Mucoadhesion; Polyethylene oxide; Polyvinylpyrrolidone

Indexed keywords

EID: 79955421808     PISSN: 15168913     EISSN: 15168913     Source Type: Journal    
DOI: 10.1590/S1516-89132011000200010     Document Type: Article

References (36)

1. Ali, J.; Hasan, S.; Ali, M. (2006), Formulation and development of gastroretentive drug delivery system for ofloxacin. Methods Find. Exp. Clin. Pharmacol., 28, 433-439.
2. Ali, J.; Tyagi, P.; Ahuja, A.; Baboota, S.; Hasan, S. (2007), Development and evaluation of a gastroretentive drug delivery system for the lowabsorption-window drug celecoxib., PDA J. Pharm. Sci. Technol., 61, 88-96.
3. Bamba, M.; Puisieux, F. (1979), Release mechanisms in gel forming sustained release preparation. Int. J. Pharm., 2, 307-315.
4. Basak, S.; Rahman, J.; Ramalingam, M. (2007), Design and in vitro testing of a floatable gastroretentive tablet of metformin hydrochloride. Pharmazie., 62, 145-148.
5. Chavanpatil, M.D.; Jain, P.; Chaudhari, S.; Shear, R.; Vavia, R.R. (2006), Novel sustained release, swellable and bioadhesive gastroretentive drug delivery system for ofloxacin, Int. J. Pharm., 316, 86-92.
6. Coffin, M.; Parr, A. (1995), Ranitidine solid dosage form. US Patent 5 407 687.
7. Dave, B.S.; Amin, A.F.; Patel, MM. (2004), Gastroretentive drug delivery system of ranitidine hydrochloride: formulation and in vitro evaluation, AAPS PharmSciTech., 5, e34.
8. Davis, S.S. (2005), Formulation strategies for absorption windows. Drug Discov. Today., 10, 249-257.
9. Deshpande, A.A., Shah, N.H., Rhodes, C.T., Malick, W. (1997), Development of a novel controlled release system for gastric retention, Pharm. Res., 14, 815-819.
10. Dhawan, S., Dhawan, K., Varma, M., Sinha, V.R. (2005), Application of poly (ethylene oxide) in drug delivery systems. Pharm Technol., 29, 72.
11. Goldsmith, J. A.; Randall, N.; Ross, S. D. (1978), Methods of expressing dissolution rate data. J. Pharm. Pharmacol., 30, 347-349.
12. Groning, R.; Cloer, C.; Muller, R.S. (2006), Development and in vitro evaluation of expandable gastroretentive dosage forms based on compressed collagen sponges. Pharmazie., 61, 608-612.
13. Gröninga, R.; Cloera, C.; Georgarakisb, M.; Müllera, R.S. (2007), Compressed collagen sponges as gastroretentive dosage forms: in vitro and in vivo studies. Eur. J.Pharm. Sci., 30, 1-6.
14. Harland, R. S.; Gazzaniga, A.; Sangalli, M. E., et al. (1988), Drug/polymer matrix: swelling and dissolution. Pharm. Res., 5, 488-494.
15. Higuchi, T. (1963), Mechanism of sustained-action medication: theoretical analysis of rate of release of solid drugs dispersed in solid matrices. J. Pharm. Sci., 52, 1145-1149.
16. Hixon, A. W.; Crowell, J. H. (1931), Dependence of reaction velocity upon surface and agitation. Ind. Eng. Chem., 23, 923-931.
17. Huang, Y.; Leobandung, W.; Foss, A.; Peppas, N.A. (2000), Molecular aspects of muco- and bioadhesion: tethered structures and site-specific surfaces. J. Control. Release., 65, 63-71.
18. Jaimini, M.; Rana, A. C.; Tanwar, Y. S. (2007), Formulation and evaluation of famotidine floating tablets. Curr. Drug Deliv., 4, 51-55.
19. Klausner, E.A.; Lavy, E.; Friedman, M.; Hoffman, A. (2003), Expandable gastroretentive dosage forms. J.Control. Release., 90, 143-162.
20. Korsmeyer, R.; Gurny, R.; Peppas, N. (1983), Mechanisms of solute release from porous hydrophilic polymers. Int. J. Pharm., 15, 25-35.
21. Langenbucher, F. (1972), Linearization of dissolution rate curves by the Weibull distribution. J. Pharm. Pharmacol., 24, 979-981.
22. Mahalingam, R.; Jasti, B.; Birudaraj, R.; Stefanidis, D.; Killion, R.; Alfredson, T.; Anne, P.; Li, X. (2009), Evaluation of Polyethylene Oxide Compacts as Gastroretentive Delivery Systems. AAPS PharmSciTech, 10, 98-103.
23. Marathe, P.H.; Arnold, M.E.; Meeker, J.; Greene, D.S.; Barbhaiya, R.H. (2000), Pharmacokinetics and bioavailability of a metformin/glyburide tablet administered alone and with food. J. Clin. Pharmacol., 40, 1494-1502.
24. Moes, A.J. (1993), Gastroretentive dosage forms. Crit. Rev. Ther. Drug Carrier. Syst., 10, 143-195.
25. Peppas, N. A. (1985), Analysis of Fickian and non-Fickian drug release from polymers. Pharm. Acta. Helv., 60, 110-111.
26. Ponchel, G.; Irache, J. (1998), Specific and non-specific bioadhesive particulate systems for oral delivery to the gastrointestinal tract. Adv. Drug. Deliv. Rev., 34, 191-219.
27. Raval, J.A.; Patel, J.K.; Naihong, LI, Patel, M.M. (2007), Ranitidine hydrochloride floating matrix tablets based on low density powder: effects of formulation and processing parameters on drug release. Asian J. Pharm. Sci., 2, 130-142.
28. Reynolds, J.E.F. (1996), Martindale the Extra Pharmacopoeia, The Royal Pharmaceutical Society: London, 1218-1220.
29. Rouge, N.; Alle?mann, E.; Gex-fabry, M.; Balant, L.; Cole, E.T.; Buri, P.; Doelker, E. (1998), Comparative pharmacokinetic study of a floating multiple-unit capsule, a high-density multiple-unit capsule and an immediate-release tablet containing 25 mg atenolol. Pharm. Acta Helv., 73, 81-87.
30. Streubel, A.; Siepmann, J.; Bodmeier, R. (2002), Floating microparticles based on low density foam powder. Int J Pharm., 241, 279-292.
31. Streubel, A.; Siepmann, J.; Bodmeier, R. (2003), Multiple unit gastroretentive drug delivery systems: a new preparation method for low density microparticles. J. Microencapsul., 20, 329-347.
32. Streubel, A.; Siepmann, J.; Bodmeier, R. (2006), Gastroretentive drug delivery systems. Expert. Opin. Drug Deliv., 3, 217-233.
33. Streubel, A.; Siepmann, J.; Bodmeier, R. (2006a), Drug delivery to the upper small intestine window using gastroretentive technologies. Curr. Opin. Pharmacol., 6, 501-508.
34. Talukder, R.; Fassihi, R. (2004), Gastroretentive delivery systems: hollow beads. Drug Dev. Ind. Pharm., 30, 405-412.
35. Tao, S.L.; Desai, T.A. (2005), Gastrointestinal patch systems for oral drug delivery. Drug Discov. Today., 10, 909-915.
36. Whitehead, L.; Fell, J.T.; Collett, J.H.; Sharma, H.L.; Smith, A.M. (1998), Floating dosage forms: an in vivo study demonstrating prolonged gastric retention. J. Control Release, 55, 3-12.