Solid dispersions of imidazolidinedione by PEG and PVP polymers with potential antischistosomal activities

AAPS PharmSciTech

Volumn 12, Issue 1, 2011, Pages 401-410

  Guedes, Francimary L ^a   De Oliveira, Boaz G ^a   Hernandes, Marcelo Z ^a   De Simone, Carlos A ^b   Veiga, Francisco J B ^c   De Lima, Maria Do Carmo A ^a   Pitta, Ivan R ^a   Galdino, Suely L ^a   Neto, Pedro José Rolim ^a  

^a FEDERAL UNIVERSITY OF PERNAMBUCO   (Brazil)

^b FEDERAL UNIVERSITY OF ALAGOAS   (Brazil)

^c UNIVERSITY OF COIMBRA   (Portugal)

Author keywords

dissolution profiles; imidazolidinedione; polyethyleneglycol; polyvinylpyrrolidone; solid dispersions

Indexed keywords

3 (4 CHLORO BENZYL) 5 (4 NITRO BENZYLIDENE) IMIDAZOLIDINE 2,4 DIONE; AMIDE; ANTISCHISTOSOMAL AGENT; CARBONYL DERIVATIVE; ETHER; HYDROGEN; IMIDAZOLIDINEDIONE; NITROGEN; OXYGEN; POLYETHYLENOGLYCOL; POLYMER; POVIDONE; UNCLASSIFIED DRUG; WATER;

ARTICLE; CONCENTRATION (PARAMETERS); DIFFERENTIAL SCANNING CALORIMETRY; DISSOLUTION; DRUG BIOAVAILABILITY; DRUG SOLUBILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROGEN BOND; MOLECULAR INTERACTION; PRIORITY JOURNAL; SCANNING ELECTRON MICROSCOPY; SOLID; THERMAL ANALYSIS; X RAY DIFFRACTION;

DOSAGE FORMS; DRUG CARRIERS; DRUG COMPOUNDING; DRUG DELIVERY SYSTEMS; HYDANTOINS; MODELS, MOLECULAR; POLYETHYLENE GLYCOLS; POLYMERS; POVIDONE; SCHISTOSOMICIDES; SOLUBILITY;

EID: 79954425113     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-010-9556-z     Document Type: Article

References (27)

1. WHO, Word Health Organization Disease Information, 2001
2. MCPA Albuquerque MGR Pitta JI Irmão CA Peixoto E Malagueño JV Santana, et al. 2007 Tegumental alterations in adult Schistosoma mansoni treated with imidazolidine derivatives Lat Am J Pharm 26 65 69 1:CAS:528:DC%2BD2sXotlektrs%3D (Pubitemid 47075245)
3. Pitta IR, Lima MCA, Albuquerque MCPA, Galdino SL. Novel compositions of imidazolidine derivatives useful in the treatment of intestinal schistosomiasis. Braz. Pedido PI, 2005
4. SM Oliveira MCPA Albuquerque MGR Pitta E Malagueño JV Santana MCA Lima, et al. 2004 Behavior of Schistosoma mansoni adult worms maintained in vitro towards imidazolidinone derivatives Acta Farm Bonaerense 23 343 348 1:CAS:528:DC%2BD2cXhtVCkt7jF (Pubitemid 39490576)
5. MCA Lima DLB Costa AJS Goes SL Galdino IR Pitta C Luu-Duc 1992 Synthesis and antimicrobial activity of chlorobenzyl benzylidene imidazolidinediones and thiazolidinediones Pharmazie 47 182 184 1615023 1:CAS:528:DyaK38Xkt1Knsbw%3D
6. SL Galdino MCA Lima AJS Goes IR Pitta LD Cuong 1991 Mass spectrometry of some benzylidene imidazolidinediones and thiazolidinediones. II. Chlorobenzyl imidazolidinedione and fluoro or chlorobenzyl thiazolidinedione compounds Spectrosc Lett 24 7-8 1013 1021 10.1080/00387019108020679 1:CAS:528: DyaK3MXms1GqtLs%3D
7. D Bikiaris GZ Parageorgiou A Stergiou E Pavlidou E Karavas F Kanaze, et al. 2005 Physicochemical studies on solid dispersions of poorly water-soluble drugs evaluation of capabilities and limitations of thermal analysis techniques Thermochem Acta 439 58 67 10.1016/j.tca.2005.09.011 1:CAS:528:DC%2BD2MXht1GlsrfM (Pubitemid 41688353)
8. S Verheyen N Blaton R Kinget GVD Mooter 2002 Mechanism of increased dissolution of diazepam and temazepam from polyethylene glycol 6000 solid dispersions Int J Pharm 249 45 58 12433433 10.1016/S0378-5173(02)00532-X 1:CAS:528:DC%2BD38XosFagtb0%3D (Pubitemid 35333431)
9. M Franco G Trapani A Latrofa C Tullio MR Provenzano M Serra, et al. 2001 Dissolution properties and anticonvulsant activity of phenytoin-polyethylene glycol 6000 and -polyvinylpyrrolidone K-30 solid dispersions Int J Pharm 225 63 73 11489555 10.1016/S0378-5173(01)00751-7 1:CAS:528:DC%2BD3MXlslant7g%3D (Pubitemid 32728200)
10. U.S, Department of Health and Human Services. Guidance for Industry: Dissolution Testing of Immediate Release Solid Oral Dosage Forms, August 1997. Available at: http://www.fda.gov/cder/guidance/1713 bp1.pdf. Accessed on: February 21, 2008.
11. KA Khan 1975 The concept of dissolution efficiency J Pharm Pharmacol 27 48 49 235616 1:CAS:528:DyaE2MXhsVCru7o%3D
12. L Ribeiro T Loftsson D Ferreira D Veiga 2003 Investigation and physicochemical characterization of vinpocetine-sulfobutyl ether β-cyclodextrins in solid binary and ternary complexes Chem Pharm Bull 51 914 922 12913228 10.1248/cpb.51.914 1:CAS:528:DC%2BD3sXnsFynsrg%3D (Pubitemid 41656773)
13. MD Veiga PJ Díaz F Ahsan 1998 Interactions of griseofulvin with cyclodextrins binary systems J Pharm Sci 87 891 900 9649360 10.1021/js970233x 1:CAS:528:DyaK1cXjsl2htLo%3D (Pubitemid 28319422)
14. BG Oliveira MCA Lima IR Pita SL Galdino MZ Hernandes 2010 J Mol Model 16 119 127 10.1007/s00894-009-0525-y 1:CAS:528:DC%2BC3cXlslGiur8%3D
15. Frisch MJ, Trucks GW, Schlegel HB, Scuseria GE, Robb MA, Cheeseman JR, et al. Gaussian 03. Wallingford CT: Gaussian, Inc.; 2004.
16. McQuarrie D. Estatística termodinâmica. New York: Harper & Row; 1973.
17. SB Boys F Bernardi 1970 Mol Phys 19 553 566 10.1080/00268977000101561 1:CAS:528:DC%2BD2sXht1alt7fM
18. GV Mooter P Augustijns N Blaton R Kinget 1998 Physico-chemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30 Int J Pharm 164 67 80 10.1016/S0378-5173(97)00401-8 (Pubitemid 28160099)
19. Z Naima T Siro GD Juan-Manuel C Chantal C René D Jerome 2001 Interactions between carbamazepine and polyethylene glycol (PEG) 6000: characterisations of the physical, solid dispersed and eutectic mixtures Eur J Pharm Sci 12 395 404 11231106 10.1016/S0928-0987(00)00168-8 1:CAS:528: DC%2BD3MXhsFSgsr8%3D (Pubitemid 32166738)
20. E Karavas G Ktistis A Xenakis E Georgarakis 2006 Effect of hydrogen bonding interactions on the release mechanism of felodipine from nanodispersions with polyvinylpyrrolidone Eur J Pharm Biopharm 63 103 114 16675209 10.1016/j.ejpb.2006.01.016 1:CAS:528:DC%2BD28XltFCgs78%3D (Pubitemid 43776203)
21. A Figueiras RA Carvalho L Ribeiro JJ Torres-Labandeira FJB Veiga 2007 Solid-state characterization and dissolution profiles of the inclusion complexes of omeprazole with native and chemically modified β-cyclodextrin Eur J Pharm Biopharm 67 531 539 17451924 10.1016/j.ejpb.2007.03.005 1:CAS:528:DC%2BD2sXovFyrsrc%3D (Pubitemid 47211912)
22. E Karavas E Georgarakis MP Sigalas K Avgoustakis D Bikiaris 2007 Investigations of the release mechanism of a sparingly water-soluble drug from solid dispersions in hydrophilic carries based on physical state of drug, particle size distribution and drug-polymer interactions Eur J Pharm Biopharm 66 334 347 17267194 10.1016/j.ejpb.2006.11.020 1:CAS:528:DC%2BD2sXlsFKmtLg%3D (Pubitemid 46778978)
23. LP Ruan BY Yu GM Fu D Zhu 2005 Improving the solubility of ampelopsin by solid dispersions and inclusion complexes J Pharm Biopharm Anal 38 457 464 1:CAS:528:DC%2BD2MXltVegtbo%3D (Pubitemid 40733182)
24. S Sethia E Squillante 2004 Solid dispersions of carbamazepine in PVP k30 by conventional solvent evaporation and supercritical methods Int J Pharm 272 1 10 15019063 10.1016/j.ijpharm.2003.11.025 1:CAS:528:DC%2BD2cXhs1Giurw%3D (Pubitemid 38293005)
25. DQM Craig 2002 The mechanisms of drug release from solid dispersions in water-soluble polymers Int J Pharm 231 131 144 11755266 10.1016/S0378-5173(01) 00891-2 1:CAS:528:DC%2BD3MXptlaitL0%3D (Pubitemid 34033673)
26. P Mura N Zerrouk N Mennini F Moestreli C Chemtob 2003 Development and characterization of naproxen-chitosan solid systems with improved drug dissolution properties Eur J Pharm Sci 19 67 75 12729863 10.1016/S0928-0987(03) 00068-X 1:CAS:528:DC%2BD3sXjt1Ogsrc%3D (Pubitemid 36506939)
27. L Marzocchi JR Moyano A Rossi P Muñoz MJ Arias F Giordano 2001 Current status of ATPase proton pump inhibitor complexation with cyclodextrins Biolog J Armenia 53 176 193 1:CAS:528:DC%2BD38XnvVOgt7g%3D