New and more efficient multivalent glyco-ligands for asialoglycoprotein receptor of mammalian hepatocytes

Bioorganic and Medicinal Chemistry

Volumn 19, Issue 8, 2011, Pages 2494-2500

  Lee, Reiko T ^a   Wang, Mei Hui ^b   Lin, Wuu Jyh ^b   Lee, Yuan C ^a  

^a JOHNS HOPKINS UNIVERSITY   (United States)

^b INSTITUTE OF NUCLEAR ENERGY RESEARCH   (Taiwan)

Author keywords

Endocytosis; Hepatocytes; Hexa valent glyco ligand; Liver targeting; Tri valent glyco ligand

Indexed keywords

AMINOGLYCOSIDE; ASIALOGLYCOPROTEIN RECEPTOR; ASPARTIC ACID DERIVATIVE; CARBOXYL GROUP; GLYCOPEPTIDE; GLYCOSIDE; INDIUM 111; IODINE 125; LACTOSE; LACTOSIDE; LIGAND; LYSINE; N ACETYLGALACTOSAMINE; NALPHA (TRIFLUOROACETAMIDO)HEXANOYL ASPARTIC ACID; PEPTIDE DERIVATIVE; TYROSYLASPARTYLGLUTAMIC ACID; TYROSYLGLUTAMYLGLUTAMIC ACID; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; CARBOHYDRATE ANALYSIS; CARBOHYDRATE SYNTHESIS; CONTROLLED STUDY; DRUG ACCUMULATION; DRUG DISTRIBUTION; LIVER CELL; MALE; MAMMAL CELL; MOUSE; NONHUMAN; RADIOACTIVITY; RAT;

ACETYLGALACTOSAMINE; ANIMALS; ASIALOGLYCOPROTEIN RECEPTOR; CELLS, CULTURED; GLYCOSIDES; HEPATOCYTES; LACTOSE; LIGANDS; LIVER; MICE; PROTEIN BINDING; RATS;

MAMMALIA; MUS; RATTUS;

EID: 79954417405     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2011.03.027     Document Type: Article

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